“kinase inhibitor”的搜索结果

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  1. AKT Kinase Inhibitor

    Catalog No. A11285
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    Akt kinase inhibitor
    AKT Kinase Inhibitor is an Akt kinase inhibitor with anti-tumor activity. 了解更多
  2. Multi-kinase inhibitor 1

    Catalog No. A22645
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    multi-kinase inhibitor
    Multi-kinase inhibitor 1 is a potent multi-kinase inhibitor. Multi-kinase inhibitor 1 has the potential for diseases or disorders associated with abnormal or deregulated tyrosine kinase activity, particularly diseases associated with the activity of PDGF-R, c-Kit and Bcr-abl. 了解更多
  3. Src Inhibitor 1

    Catalog No. A12299
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    Src tyrosine kinase inhibitor
    Src Inhibitor 1 is a potent and selective dual site Src tyrosine kinase inhibitor with IC50 values of 44 nM for Src and 88nM for Lck. 了解更多
  4. Kinase inhibitor-1

    Catalog No. A20661
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    Kinase inhibitor-1 (Compound 5) is a kinase inhibitor. 了解更多
  5. RIP1 kinase inhibitor 1

    Catalog No. A20154
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    RIP1 kinase inhibitor
    RIP1 kinase inhibitor 1 (compound 22) is a highly potent, orally available, and brain-penetrating RIP1 kinase inhibitor (pKi=9.04). 了解更多
  6. PDGFRα kinase inhibitor 1

    Catalog No. A19632
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    type II PDGFRα kinase inhibitor
    PDGFRα kinase inhibitor 1 is a highly selective type II PDGFRα kinase inhibitor with IC50s of 132 nM and 6115 nM for PDGFRα and PDGFRβ, respectively. 了解更多
  7. Aurora Kinase Inhibitor 3

    Catalog No. A19448
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    Aurora A kinase inhibitor
    Aurora Kinase Inhibitor 3 is a strong and selective Aurora A kinase inhibitor with an IC50 of 42 nM, and weakly inhibits EGFR with an IC50>10 μM. 了解更多
  8. Tie2 kinase inhibitor

    Catalog No. A10932
    Tie2 kinase inhibitor
    Tie2 kinase inhibitor是一种有效的选择性Tie2抑制剂,IC50为0.25μM。 了解更多
  9. Histone Acetyltransferase Inhibitor II

    Catalog No. A12331
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    cell permeable p300 inhibitor
    Histone Acetyltransferase Inhibitor II is a potent and cell permeable p300 inhibitor, with an IC50 of 5 ?M; Histone Acetyltransferase Inhibitor II can be used in cancer research. 了解更多
  10. CPA inhibitor

    Catalog No. A11369
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    CPA inhibitor
    CPA inhibitor is a potent inhibitor for carboxypeptidase A (CPA). 了解更多
  11. IRAK inhibitor 2

    Catalog No. A11456
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    interleukin-1 receptor associated kinase inhibitor
    IRAK inhibitor 2 is interleukin-1 receptor associated kinase inhibitor . 了解更多
  12. RIP2 Kinase Inhibitor 3

    Catalog No. A20109
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    RIP2 inhibitor
    RIP2 Kinase Inhibitor 3 is a highly potent and selective inhibitor of receptor interacting protein-2 (RIP2) Kinase with an IC50 of 1 nM . 了解更多
  13. Btk inhibitor 1 R enantiomer hydrochloride

    Catalog No. A21865
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    BTK inhibitor
    Btk inhibitor 1 R enantiomer hydrochloride (Ibrutinib analog hydrochloride) (Compound 14) is a covalent and irreversible Bruton??s tyrosine kinase (BTK) inhibitor and can be used in synthesis of Ibrutinib and ibrutinib-based activity-based probes (ABPs). 了解更多
  14. Btk inhibitor 1 (R enantiomer)

    Catalog No. A21861
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    BTK inhibitor
    Btk inhibitor 1 R enantiomer (Ibrutinib analog) (Compound 14) is a covalent and irreversible Bruton??s tyrosine kinase (BTK) inhibitor and can be used in synthesis of Ibrutinib and ibrutinib-based activity-based probes (ABPs). 了解更多
  15. IRAK inhibitor 4

    Catalog No. A11458
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    IRAK4 inhibitor
    IRAK inhibitor 4 is an interleukin-1 receptor associated kinase 4(IRAK4) inhibitor. 了解更多
  16. MARK4 inhibitor 1

    Catalog No. A18695
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    (MARK4 inhibitor
    MARK4 inhibitor 1 is a potent microtubule affinity-regulating kinase 4 (MARK4) inhibitor, with an IC50 of 1.54 μM. MARK4 inhibitor 1 inhibits cancer cell proliferation, metastasis and induces apoptosis. 了解更多
  17. Casein Kinase II Inhibitor IV

    Catalog No. A12624
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    Epidermal keratinocyte differentiation inducer
    Casein Kinase II Inhibitor IV is a small-molecule inducer of epidermal keratinocyte differentiation. 了解更多
  18. RIP2 kinase inhibitor 2

    Catalog No. A16313
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    RIP2 kinase 抑制剂
    RIP2 kinase inhibitor 2 是从专利WO/2014043437 A1(化合物实施例9)中提取的受体相互作用蛋白2(RIP2)激酶抑制剂。 了解更多
  19. RIP2 kinase inhibitor 1

    Catalog No. A16312
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    RIP2 kinase 抑制剂
    RIP2 kinase inhibitor 1 是从专利WO/2014043446 A1(化合物实施例1)中提取的受体相互作用蛋白2(RIP2)激酶抑制剂。 了解更多
  20. GSK3 Inhibitor XIII

    Catalog No. A22128
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    ATP-binding site inhibitor of GSK-3
    GSK3 Inhibitor XIII (GSK3i XIII) is an ATP-binding site inhibitor of GSK-3. 了解更多
  21. ATR inhibitor 2

    Catalog No. A22162
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    ATR inhibitor
    ATR inhibitor 2 is an ATP-competitive, orally active, and selective ATR inhibitor, with a Ki of <150 pM. 了解更多
  22. LMPTP INHIBITOR 1 dihydrochloride

    Catalog No. A22227
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    LMPTP inhibitor
    LMPTP INHIBITOR 1 (dihydrochloride) is a selective inhibitor of low molecular weight protein tyrosine phosphatase (LMPTP), with an IC50 of 0.8 μM LMPTP-A. 了解更多
  23. VPS34 inhibitor 1 (Compound 19)

    Catalog No. A22378
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    VPS34 inhibitor
    VPS34 inhibitor 1 (Compound 19, PIK-III analogue) is a potent and selective inhibitor of VPS34 with an IC50 of 15 nM. 了解更多
  24. Selective PI3Kδ Inhibitor 1 (compound 7n)

    Catalog No. A22381
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    PI3Kδ inhibitor
    Selective PI3Kδ Inhibitor 1 (compound 7n) is an inhibitor of PI3Kδ with an IC50 of 0.9 nM and >1000-fold selectivity against other class I PI3K isoforms [PI3K α/γ/β=3670/1460/21300 nM]. 了解更多
  25. BTK inhibitor 1 (Compound 27)

    Catalog No. A22445
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    BTK inhibitor
    BTK inhibitor 1 (compound 27) is an inhibitor of BTK with an IC50 of 0.11 nM for Btk and inhibits B cell activation in hWB with an IC50 of 2 nM. 了解更多
  26. Diacylglycerol acyltransferase inhibitor-1

    Catalog No. A20315
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    DGAT1 inhibitor
    Diacylglycerol acyltransferase inhibitor-1 is a diacylglycerol acyltransferase (DGAT1) inhibitor. 了解更多
  27. MAT2A inhibitor 2

    Catalog No. A20171
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    MAT2A inhibitor
    MAT2A inhibitor 2 is a methionine adenosyltransferase 2A (MAT2A) inhibitor. 了解更多
  28. DAAO inhibitor-1

    Catalog No. A20117
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    DAAO inhibitor
    DAAO inhibitor-1 is a potent D-amino acid oxidase (DAAO) inhibitor with an IC50 of 0.12 μM. 了解更多
  29. Grp94 Inhibitor-1

    Catalog No. A20073
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    Grp94 inhibitor
    Grp94 Inhibitor-1 is a potent, selective Grp94 inhibitor with an IC50 value of 2 nM, and over 1000-fold selectivity to Grp94 against Hsp90α. 了解更多
  30. mTOR inhibitor-1

    Catalog No. A20029
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    mTOR inhibitor
    mTOR inhibitor-1 is a novel mTOR pathway inhibitor which can suppress cells proliferation and inducing autophagy. 了解更多
  31. Tubulin inhibitor 1

    Catalog No. A19998
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    tubulin inhibitor
    Tubulin inhibitor 1 is a tubulin inhibitor, inhibits tubulin polymerization. 了解更多
  32. YAP/TAZ inhibitor-1

    Catalog No. A19976
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    YAP/TAZ inhibitor
    YAP/TAZ inhibitor-1 is a YAP/TAZ inhibitor extracted from patent WO2017058716A1, Compound 1, has an IC50 of <0.100 μμ in firefly luciferase assay. 了解更多
  33. SIRT5 inhibitor 1

    Catalog No. A19841
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    SIRT5 inhibitor
    SIRT5 inhibitor 1 is a potent Human Sirtuin 5 deacylase inhibitor, with an IC50 of 0.11 μM. 了解更多
  34. BET bromodomain inhibitor

    Catalog No. A19831
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    BET inhibitor
    BET bromodomain inhibitor is a potent BET inhibitor extracted from patent WO/2015/153871A2, compound example 11. 了解更多
  35. TRAF-STOP inhibitor 6877002

    Catalog No. A19758
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    CD40-TRAF6 interaction inhibitor
    TRAF-STOP inhibitor 6877002, is a selective inhibitor of CD40-TRAF6 interaction, compound VII, shows inhibition of NF-κB activation in RAW cells, extracted from patent WO2014033122A1. 了解更多
  36. Glutaminyl Cyclase Inhibitor 1

    Catalog No. A19723
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    glutaminyl cyclase inhibitor
    Glutaminyl Cyclase Inhibitor 1 is a glutaminyl cyclase inhibitor with an IC50 of 0.5 μM. 了解更多
  37. PKC-theta inhibitor

    Catalog No. A19712
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    PKC-θ inhibitor
    PKC-theta inhibitor is a selective PKC-θinhibitor, with an IC50 of 12 nM. 了解更多
  38. LRRK2 inhibitor 1

    Catalog No. A19701
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    LRRK2 inhibitor
    LRRK2 inhibitor 1 is a potent, selective and oral LRRK2 inhibitor with an pIC50 of 6.8 nM. 了解更多
  39. HIV-1 integrase inhibitor 3

    Catalog No. A19628
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    INST inhibitor
    HIV-1 integrase inhibitor 3 is a HIV-1 integrase strand transfer (INST) inhibitor with an IC50 of 2.7 nM. 了解更多
  40. PI3K/mTOR Inhibitor-2

    Catalog No. A19621
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    dual pan-PI3K/mTOR inhibitor
    PI3K/mTOR Inhibitor-2 is a potent dual pan-PI3K/mTOR inhibitor with IC50s of 3.4/34/16/1 nM for PI3Kα/PI3Kβ/PI3Kδ/PI3Kγ and 4.7 nM for mTOR. Antitumor activity. 了解更多
  41. HIV-1 integrase inhibitor 4

    Catalog No. A19617
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    INST inhibitor
    HIV-1 integrase inhibitor 4 is a HIV-1 integrase strand transfer (INST) inhibitor with an IC50 of 3.7 nM. 了解更多
  42. Neurotoxin Inhibitor

    Catalog No. A19507
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    neurotoxin inhibitor
    Neurotoxin Inhibitor is a neurotoxin inhibitor. 了解更多
  43. p38α inhibitor 1

    Catalog No. A19182
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    p38α inhibitor
    p38α inhibitor 1 is a p38α inhibitor extracted from patent WO 2008076265 A1. 了解更多
  44. Bromodomain inhibitor-8

    Catalog No. A19161
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    BET bromodomain inhibitor
    Bromodomain inhibitor-8 (Intermediate 21) is a BET bromodomain inhibitor for treating autoimmune and inflammatory diseases. 了解更多
  45. FAAH inhibitor 1

    Catalog No. A21841
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    FAAH inhibitor
    FAAH inhibitor 1 (Benzothiazole analog 3) is a potent fatty acid amide hydrolase (FAAH) inhibitor with an IC50 of 18??8 nM. 了解更多
  46. Notch inhibitor 1

    Catalog No. A21591
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    Notch inhibitor
    Notch inhibitor 1 is a potent Notch inhibitor, with IC50s of 7.8 and 8.5 nM for Notch 1 and Notch 3, respectively. Used in the research of cancer. 了解更多
  47. β-Secretase Inhibitor IV

    Catalog No. A21346
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    BACE-1 inhibitor
    β-Secretase Inhibitor IV is a potent, cell-active BACE-1 inhibitor with IC50s of 15.6 and 16.3nM under BACE-1 concentrations of 2 nM and 100 pM, respectively. 了解更多
  48. HIV-1 integrase inhibitor 2

    Catalog No. A11447
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    HIV-1 integrase inhibitor
    HIV-1 integrase inhibitor 2, in the treatment of human immunodeficiency virus (HIV) infection. 了解更多
  49. HIV-1 integrase inhibitor

    Catalog No. A11446
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    HIV-1 integrase inhibitor
    HIV-1 integrase inhibitor is uesful for anti-HIV. 了解更多
  50. P-gp inhibitor 1

    Catalog No. A13384
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    P-gp inhibitor
    P-gp inhibitor 1 is a novel inhibitor reversing P-glycoprotein-mediated multidrug resistance. 了解更多

产品 1 到 50 共 5606个

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