“AZ 960”的搜索结果

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  1. Vilazodone

    Catalog No. A11116
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    Serotonin reuptake 抑制剂
    Vilazodone充当5-羟色胺再摄取抑制剂(IC50 = 0.5 nM)和5-HT1A受体部分激动剂(IC50 = 0.2 nM; IA =?60-70%)。 了解更多
  2. Atomoxetine HCl

    Catalog No. A13424
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    norepinephrine (NE) transporter 抑制剂
    Atomoxetine HCl是SLC6A2的一种竞争性特异性抑制剂,同时在大鼠下丘脑突触体中显示出微弱的ST和DAT抑制作用。 了解更多
  3. Antazoline HCl

    Catalog No. A16411
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    Histamine H1 receptor 抑制剂
    Antazoline HCl是第一代抗组胺药,可与组胺H1受体结合并阻断内源性组胺的作用。 了解更多
  4. Azatadine dimaleate

    Catalog No. A16418
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    Histamine/cholinergic 抑制剂
    Azatadine是一种组胺和胆碱能抑制剂,IC50分别为6.5 nM和10 nM。 了解更多
  5. Loxapine Succinate

    Catalog No. A17347
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    D2DR and D4DR inhibitor
    Loxapine Succinate is a D2DR and D4DR inhibitor and serotonergic receptor antagonist. Loxapine succinate is an antipsychotic agent used in schizophrenia. 了解更多
  6. Nefazodone hydrochloride

    Catalog No. A17622
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    5-HT2 receptors inhibitor
    Nefazodone HCl is an inhibitor of 5-HT2 receptors, SERT, NET, and hERG K+ channels used to treat mood disorders. It decreases immobility time in the forced swim test. 了解更多
  7. Promazine hydrochloride

    Catalog No. A17638
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    D2DR inhibitor
    Promazine Hydrochloride is a phenothiazine compound and D2DR inhibitor. Promazine Hydrochloride has been employed in studies investigating dopamine-stimulated glycosylation of brain proteins in vitro. It has actions similar to chlorpromazine but with less antipsychotic activity. 了解更多
  8. MHP 133

    Catalog No. A20058
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    AChE /M1/M2/5HT4/I2 inhibitor
    MHP 133 is a drug with multiple CNS targets, and inhibits acetylcholinesterase (AChE) with Ki of 69 μM; also active against muscarinic M1 and M2 receptors, serotonin 5HT4 receptors, and imidazole I2 receptors. 了解更多
  9. Pentiapine

    Catalog No. A12512
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    dopamine release inhibitor
    Pentiapine is a novel dopamine release inhibitor. 了解更多
  10. Loxapine

    Catalog No. A18073
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    D2DR/D4DR inhibitor
    Loxapine Succinate is a D2DR and D4DR inhibitor, serotonergic receptor antagonist and also a dibenzoxazepine anti-psychotic agent. 了解更多
  11. Vilazodone D8

    Catalog No. A21876
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    SSR inhibitor / 5-HT1A receptor partial agonist
    Vilazodone D8 is the a deuterium labeled vilazodone, which is a combined serotonin specific reuptake inhibitor (SSRI) and 5-HT1A receptor partial agonist. 了解更多
  12. Vanoxerine

    Catalog No. A21922
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    dopamine reuptake inhibitor
    Vanoxerine (GBR-12909) is a competitive, potent, and highly selective dopamine reuptake inhibitor (Ki=1 nM). 了解更多
  13. GBR 12935

    Catalog No. A21951
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    dopamine reuptake inhibitor
    GBR 12935 is a potent, and selective dopamine reuptake inhibitor. 了解更多

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