“A 300”的搜索结果

产品 201 到 250 共 17506个

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  1. RO5203648 hydrochloride

    Catalog No. A22118
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    partial agonist of Trace amine-associated receptor 1
    RO5203648 hydrochloride is a partial agonist of Trace amine-associated receptor 1 (TAAR1). 了解更多
  2. NSC-45586

    Catalog No. A22119
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    pan-PHLPP inhibitor
    NSC-45586 is a pan-PHLPP inhibitor selective for PHLPP1 and PHLPP2. 了解更多
  3. FLTX1

    Catalog No. A22120
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    antiestrogenic properties
    FLTX1 is a fluorescent Tamoxifen derivative that can specifically label intracellular Tamoxifen-binding sites (estrogen receptors) under permeabilized and non-permeabilized conditions. FLTX1 exhibits the potent antiestrogenic properties of Tamoxifen in breast cancer cells. FLTX1 is devoid of the estrogenic agonistic effect on the uterus. 了解更多
  4. Epiblastin A

    Catalog No. A22121
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    inhibitor of Casein Kinase 1 (CK1)
    Epiblastin A is an inhibitor of Casein Kinase 1 (CK1) that engages CK1 isoenzymes in cell lysate and induces efficient conversion of epiblast stem cells (EpiSCs) into embryonic stem cells (cESCs). 了解更多
  5. ML198

    Catalog No. A22122
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    activator and non-inhibitory chaperone of glucocerebrosidase
    ML198 is a novel activator and non-inhibitory chaperone of glucocerebrosidase. 了解更多
  6. R243

    Catalog No. A22123
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    inhibitor of CCR8 signaling and chemotaxis
    R243 is an inhibitor of CCR8 signaling and chemotaxis. 了解更多
  7. BMS-986188

    Catalog No. A22124
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    Positive Allosteric Modulator of the delta-Opioid Receptor
    BMS-986188 is a novel Potent and Selective Positive Allosteric Modulator of the delta-Opioid Receptor. 了解更多
  8. BMS-986187

    Catalog No. A22125
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    positive allosteric modulator (PAM) of the δ-opioid receptor and a G-protein-biased allosteric agonist
    BMS-986187 is a potent and selective positive allosteric modulator (PAM) of the δ-opioid receptor and a G-protein-biased allosteric agonist. 了解更多
  9. NCGC607

    Catalog No. A22126
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    noninhibitory chaperone
    NCGC607 is a a noninhibitory chaperone of glucocerebrosidase (GCase). 了解更多
  10. PythiDC

    Catalog No. A22127
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    inhibitor of collagen prolyl 4-hydroxylase
    PythiDC is a selective inhibitor of collagen prolyl 4-hydroxylase. 了解更多
  11. GSK3 Inhibitor XIII

    Catalog No. A22128
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    ATP-binding site inhibitor of GSK-3
    GSK3 Inhibitor XIII (GSK3i XIII) is an ATP-binding site inhibitor of GSK-3. 了解更多
  12. MN58b

    Catalog No. A22129
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    choline kinase α (CHKα) inhibitor
    MN58b is a selective choline kinase α (CHKα) inhibitor, and results in inhibition of phosphocholine synthesis. 了解更多
  13. BGC201531

    Catalog No. A22130
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    EP4 antagonist
    BGC201531, also known as GTPL3380 and AP-1531, is a EP4 antagonist for the treatment of acute migraine. 了解更多
  14. TTK21

    Catalog No. A22131
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    CBP/p300 histone acetyltransferase activator
    TTK21 is a CBP/p300 histone acetyltransferase activator. 了解更多
  15. Statil

    Catalog No. A22132
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    aldose reductase inhibitor
    Ponalrestat, also known as MK-538, is an aldose reductase inhibitor. 了解更多
  16. MDK-1088

    Catalog No. A22133
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    Trypanosoma cruzi inhibitor
    MDK-1088 (T.cruzi Inhibitor) is a Trypanosoma cruzi inhibitor. 了解更多
  17. HZ-1157

    Catalog No. A22134
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    inhibitor of hepatitis C virus (HCV)
    HZ-1157 is an inhibitor of hepatitis C virus (HCV) with inhibitory activities toward HCV NS3/4A protease. 了解更多
  18. RGW 611

    Catalog No. A22135
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    anti-infective agent
    RGW 611, a morpholine derivative, is an impurity of Nimorazole, which is an anti-infective agent against anaerobic bacteria and protozoa. 了解更多
  19. (Z)-JIB-04

    Catalog No. A22137
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    Jumonji histone demethylase inihibitor
    Z-JIB-04 (NSC 693627, JIB-04 Z-isomer) is an isomer of JIB-04. JIB-04 is a pan-selective Jumonji histone demethylase inihibitor with IC50 of 230 nM, 340 nM, 855 nM, 445 nM, 435 nM, 1100 nM and 290 nM for JARID1A, JMJD2E, JMJD3, JMJD2A, JMJD2B, JMJD2C, and JMJD2D, respectively. 了解更多
  20. DS-1205b free base

    Catalog No. A22138
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    inhibitor of AXL kinase
    DS-1205b free base is a potent and selective inhibitor of AXL kinase, with an IC50 of 1.3 nM. 了解更多
  21. MSA-2

    Catalog No. A22139
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    non-nucleotide STING agonist
    MSA-2, a potent and orally available non-nucleotide STING agonist, is bound to STING as a noncovalent dimer with nanomolar affinity. 了解更多
  22. ASLAN003

    Catalog No. A22140
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    Dihydroorotate Dehydrogenase (DHODH) inhibitor
    ASLAN003 is an orally active and potent Dihydroorotate Dehydrogenase (DHODH) inhibitor with an IC50 of 35 nM for human DHODH enzyme. 了解更多
  23. (Rac)-JBJ-04-125-02

    Catalog No. A22141
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    EGFR inhibitor
    (Rac)-JBJ-04-125-02 is the racemate of JBJ-04-125-02. JBJ-04-125-02 is a potent, mutant-selective, allosteric and orally active EGFR inhibitor with an IC50 of 0.26 nM for EGFRL858R/T790M. 了解更多
  24. Takeda103A

    Catalog No. A22142
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    bovine tubulin oxidation inhibitor
    Takeda103A is a potent GRK2-dependent bovine tubulin oxidation inhibitor. 了解更多
  25. GSK199

    Catalog No. A22143
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    inhibitor of PAD4
    GSK199 is a selective inhibitor of PAD4 with IC50 of 200 nM in the absence of calcium. 了解更多
  26. Pyrimorph

    Catalog No. A22144
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    fungicide
    Pyrimorph is a fungicide with high activity against the plant pathogen Phytophthora capsici. 了解更多
  27. Soporidine

    Catalog No. A22145
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    strigolactone (SL) antagonist
    Soporidine is a strigolactone (SL) antagonist and inhibitor of germination in their biological assays. It binds AtHTL and specifically interferes with SL signaling. 了解更多
  28. GNE-140 racemic

    Catalog No. A22146
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    lactate dehydrogenase (LDHA) inhibitor
    GNE-140 racemic is a novel potent lactate dehydrogenase (LDHA) inhibitor. 了解更多
  29. AA41612

    Catalog No. A22147
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    antagonist of melanopsin-mediated phototransduction
    AA41612 is an antagonist of melanopsin-mediated phototransduction. 了解更多
  30. KLH45

    Catalog No. A22148
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    DDHD2 inhibitor
    KLH45 is a potent and selective DDHD2 inhibitor, with an IC50 of 1.3 nM. 了解更多
  31. WWL229

    Catalog No. A22149
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    Ces3 inhibitor
    WWL229 is a selective inhibitor of Ces3 that acts by inhibiting recombinant Ces3 and recapitulating the effects of WWL113 in adipocytes. 了解更多
  32. ERDRP-0519

    Catalog No. A22150
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    inhibitor of polymerase
    ERDRP-0519 is an orally available inhibitor of polymerase that shows efficacy against a lethal morbillivirus infection in a large animal model. 了解更多
  33. SGC2085 hydrochloride

    Catalog No. A22151
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    inhibitor of coactivator associated arginine methyltransferase 1 (CARM1)
    SGC2085 hydrochloride is a potent and selective inhibitor of coactivator associated arginine methyltransferase 1 (CARM1) with IC50 of 50 nM. 了解更多
  34. Aka Lumine

    Catalog No. A22152
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    luciferin analogue
    Aka Lumine, a luciferin analogue, is a luciferase substrate emitting red, green, and blue light. The longest emission wavelength of Aka Lumine is recorded at 675 nm, which is within the NIR region. 了解更多
  35. Simetride

    Catalog No. A22153
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    non-narcotic analgesic
    Simetride, a non-narcotic analgesic, is an ingredient of Kyorin AP2 which is used to treat low back pain, symptomatic neuralgia, headache, menstrual pain and etc. 了解更多
  36. Nicomol

    Catalog No. A22154
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    antilipidemic agent
    Nicomol is a niacin derivative that exhibits antilipidemic activity. 了解更多
  37. Cetraxate Hydrochloride

    Catalog No. A22155
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    mucosal protective agent and an anti-ulcer drug
    Cetraxate (DV-1006) Hydrochloride (HCl) is a mucosal protective agent and an anti-ulcer drug candidate. Cetraxate raises levels of calcitonin gene-related peptide and substance P in human plasma. 了解更多
  38. Prexasertib HCl

    Catalog No. A22156
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    ATP-competitive CHK1 inhibitor
    Prexasertib (LY2606368) is an ATP-competitive CHK1 inhibitor with a Ki value of 0.9 nmol/L. For CHK2 and RSK, its IC50 values are 8 nM and 9 nM respectively in cell-free assay. 了解更多
  39. JBSNF-000088

    Catalog No. A22190
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    NNMT inhibitor
    JBSNF-000088 (6-Methoxynicotinamide), a analog of nicotinamide (NA), is a potent Nicotinamide N-methyltransferase (NNMT) inhibitor with IC50s of 1.8 ?M, 2.8 ?M, and 5.0??M for human NNMT, monkey NNMT and mouse NNMT, respectively. 了解更多
  40. (Rac)-Benpyrine

    Catalog No. A22192
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    TNF-α inhibitor
    (Rac)-Benpyrine, a racemate of Benpyrine, is a potent and orally active TNF-α inhibitor. (Rac)-Benpyrine has the potential for TNF-α mediated inflammatory and autoimmune disease research. 了解更多
  41. Adenosine amine congener

    Catalog No. A22193
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    A1 adenosine receptor agonist
    Adenosine amine congener (ADAC) is a selective A1 adenosine receptor agonist, can ameliorate noise- and Cisplatin-induced cochlear injury. 了解更多
  42. Enpp-1-IN-1

    Catalog No. A22194
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    Ectonucleotide pyrophosphatase-phosphodiesterase 1 (enpp-1) inhibitor
    Enpp-1-IN-1 is a Ectonucleotide pyrophosphatase-phosphodiesterase 1 (enpp-1) inhibitor extracted from patent WO2019046778, Example 55. 了解更多
  43. PNU112455A hydrochloride

    Catalog No. A22195
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    ATP-competitive CDK2 and CDK5 inhibitor
    PNU112455A hydrochloride is an ATP-competitive CDK2 and CDK5 inhibitor. 了解更多
  44. FOY 251

    Catalog No. A22196
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    proteinase inhibitor
    FOY 251, an anti-proteolytic active metabolite Camostate (HY-13512), acts as a proteinase inhibitor. FOY 251 inhibits SARS-CoV-2 infection in cells assay. 了解更多
  45. TH-263

    Catalog No. A22197
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    inactive analog control for the type III allosteric LIM-kinase (LIMK) inhibitors TH-257, TH-255 and TH-251
    TH-263 is an inactive analog control for the type III allosteric LIM-kinase (LIMK) inhibitors TH-257, TH-255 and TH-251. 了解更多
  46. Remimazolam besylate

    Catalog No. A22198
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    ultra short-acting benzodiazepine
    Remimazolam besylate is an ultra short-acting benzodiazepine used in the induction and maintenance of sedation during short (<30 minute) procedures. 了解更多
  47. SR-31747 free base

    Catalog No. A22199
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    immunosuppressive and anti-inflammatory properties
    SR-31747 free base is a sigma ligand with immunosuppressive and anti-inflammatory properties. 了解更多
  48. Zebularine

    Catalog No. A12721
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    DNA methyltransferase inhibitor
    Zebularine (NSC309132; 4-Deoxyuridine) is a DNA methyltransferase inhibitor. 了解更多
  49. Clobenpropit dihydrobromide

    Catalog No. A22263
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    histamine H3R antagonist/inverse agonist
    Clobenpropit dihydrobromide is a potent histamine H3R antagonist/inverse agonist with a pEC50 of 8.07 for histamine H3LR. 了解更多
  50. A 784168

    Catalog No. A22264
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    antagonist of Vanilloid receptor type 1
    A-784168 is a potent and selective antagonist of Vanilloid receptor type 1 (TRPV1). 了解更多

产品 201 到 250 共 17506个

每页
页面:
  1. 3
  2. 4
  3. 5
  4. 6
  5. 7

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