Endocrinology / Hormones

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  1. ROR gamma modulator 1

    Catalog No. A16291
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    RORγ modulator
    ROR gamma modulator 1 是类维生素A相关的孤儿受体γ(RORy)调节剂 了解更多
  2. AZD9567

    Catalog No. A18850
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    selective glucocorticoid receptor modulator
    AZD9567 is a potent, oral active, non-steroidal and selective glucocorticoid receptor modulator (SGRM), with an IC50 of 3.8 nM. 了解更多
  3. GPR120 modulator 1

    Catalog No. A15094
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    GPR120 modulator 1 可用于调节G蛋白偶联受体120(GPR120)。 了解更多
  4. GPR120 modulator 2

    Catalog No. A15095
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    GPR120 modulator 2 可用于调节G蛋白偶联受体120(GPR120)。 了解更多
  5. Ostarine (MK-2866, GTx-024)

    Catalog No. A10253
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    Androgen Receptor Modulators
    Ostarine (MK-2866,GTX-024)是一种雄激素受体调节剂(SARM)。 了解更多
  6. BMS564929

    Catalog No. A12805
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    Androgen receptor (AR) modulator
    BMS-564929是一种新型,高效,口服活性,非甾体组织选择性雄激素受体(AR)调节剂,结合到雄激素受体,Ki 为 2.11±0.16 nM。该化合物已被推进临床试验,以治疗与年龄相关的功能衰退。 了解更多
  7. GSK-2881078

    Catalog No. A12645
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    androgen receptor modulator
    GSK-2881078是一种选择性雄激素受体调节剂(SARM),正在针对肌肉萎缩以改善其身体功能的受试者的肌肉生长和力量进行评估。 了解更多
  8. MK-0773

    Catalog No. A15164
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    Androgen receptor modulator
    MK-0773是一种选择性雄激素受体调节剂(SARMs),是一种4-氮杂-类固醇,在人体中表现出组织选择性(IC50 = 6.6 nM)。 了解更多
  9. Asoprisnil

    Catalog No. A19030
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    Progesterone receptor modulator
    Asoprisnil (J867), a selective progesterone receptor modulator, exhibits mixed progesterone agonist and antagonist effects on various progesterone targeted tissues in animal and human. 了解更多
  10. Ulipristal acetate

    Catalog No. A21041
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    progesterone receptor modulator
    Ulipristal (acetate) is a novel selective progesterone receptor modulator (SPRM) for the treatment of benign gynecological conditions such as uterine myoma. 了解更多
  11. Acolbifene (EM 652, SCH57068)

    Catalog No. A12771
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    estrogen receptor modulator
    Acolbifene (EM 652,SCH57068)是第四代选择性的estrogen receptor拮抗剂,LC50 值为 22±3 nM。用于预防高乳腺癌女性的乳腺癌。 盐酸阿科比芬与体内雌激素受体结合,阻断雌激素对乳房的作用。 它是选择性雌激素受体调节剂(SERM)的一种。 了解更多
  12. Ospemifene

    Catalog No. A14261
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    estrogen receptor modulator
    Ospemifene是一种非激素选择性雌激素受体调节剂(SERM)。 了解更多
  13. Bazedoxifene

    Catalog No. A15019
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    Estrogen modulator
    Bazedoxifene是雌激素受体的第三代选择性调节剂。 了解更多
  14. Toremifene

    Catalog No. A15265
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    Estrogen receptor modulator
    Toremifene是正在开发中的第二代选择性雌激素受体调节剂(SERM),用于预防骨质疏松症。 了解更多
  15. Lasofoxifene Tartrate

    Catalog No. A18097
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    selective Estrogen receptor modulator
    Lasofoxifene tartrate is a third-generation selective estrogen receptor modulator. 了解更多
  16. Tamoxifen

    Catalog No. A16738
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    selective estrogen receptor modulator (SERM)
    Tamoxifen (ICI 47699) is a selective estrogen receptor modulator (SERM) which blocks estrogen action in breast cells and can activate estrogen activity in other cells, such as bone, liver, and uterine cells. 了解更多
  17. Estetrol

    Catalog No. A21291
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    nuclear estrogen receptor modulator
    Estetrol, a natural estrogen synthesized exclusively during pregnancy by the human fetal liver, is a selective nuclear estrogen receptor modulator. 了解更多
  18. Pipendoxifene hydrochloride

    Catalog No. A21623
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    estrogen receptor modulators
    Pipendoxifene hydrochloride is a selective estrogen receptor modulators (SERMs). 了解更多
  19. 4-Hydroxytamoxifen

    Catalog No. A20955
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    estrogen receptor modulator
    4-Hydroxytamoxifen is a selective estrogen receptor modulator (SERM). 了解更多

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