mAChR

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  1. AF-DX 384

    Catalog No. A13856
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    mAChR 拮抗剂
    AF-DX 384是充当毒蕈碱乙酰胆碱受体的选择性拮抗剂的药物。 了解更多
  2. PF-3635659

    Catalog No. A13548
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    muscarinic M(3) receptor 拮抗剂
    PF-3635659是有效的毒蕈碱M3受体拮抗剂。 了解更多
  3. Umeclidinium bromide

    Catalog No. A15268
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    Muscarinic receptor 拮抗剂
    Umeclidinium bromide (GSK573719A)是毒蕈碱受体拮抗剂,可用于治疗慢性阻塞性肺疾病(COPD)。 了解更多
  4. Revefenacin

    Catalog No. A15986
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    muscarinic receptor 拮抗剂
    Revefenacin是正在研发中的有效,选择性毒蕈碱受体拮抗剂,可用于治疗COPD。 了解更多
  5. Glycopyrrolate

    Catalog No. A12641
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    muscarinic 拮抗剂
    Glycopyrrolate是一种毒蕈碱竞争性拮抗剂,可用作解痉挛药。 了解更多
  6. Flavoxate

    Catalog No. A12900
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    muscarinic AChR antagonist
    Flavoxate结合并抑制毒蕈碱受体,从而通过改变脑干的排尿中心来抑制排尿反射并增加膀胱容量。 了解更多
  7. Atropine methyl bromide

    Catalog No. A18026
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    mAChR antagonist
    Atropine methyl bromide, a muscarinic receptor (mAChR) antagonist, is a quaternary ammonium salt of atropine and a mydriatic for dilation of the pupil during ophthalmic examination. It is introduced for relieving pyloric spasm in infants for its highly polar nature. It penetrates less readily into the central nervous system than atropine. 了解更多
  8. Cimetropium Bromide

    Catalog No. A18290
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    mAChR antagonist
    Cimetropium Bromide (DA-3177) is a mAChR antagonist for long-term treatment of irritable bowel syndrome. 了解更多
  9. Tiotropium Bromide

    Catalog No. A10934
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    muscarinic acetylcholine receptor (mAChR) antagonist
    Tiotropium Bromide (BA679 BR) is a muscarinic acetylcholine receptor (mAChR) antagonist that blocks the binding of the acetylcholine ligand and subsequent opening of the ligand-gated ion channel. 了解更多
  10. mAChR-IN-1 hydrochloride

    Catalog No. A21398
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    mAChR antagonist
    mAChR-IN-1 hydrochloride is a potent muscarinic cholinergic receptor (mAChR) antagonist, with an IC50 of 17 nM. 了解更多
  11. mAChR-IN-1

    Catalog No. A21518
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    mAChR antagonist
    mAChR-IN-1 is a potent muscarinic cholinergic receptor(mAChR) antagonist with IC50 of 17 nM. 了解更多
  12. Diphenidol HCl

    Catalog No. A14244
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    M2/M3 拮抗剂
    Diphenidol HCl是毒蕈碱M2和M3受体的有效拮抗剂,pKb为6.72和7.02。 了解更多
  13. Fesoterodine fumarate (Toviaz)

    Catalog No. A10386
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    AChR 拮抗剂
    Fesoterodine fumarate是一种用于尿急的药物,可减少尿液通过的频率并促使尿失禁。 了解更多
  14. 5-hydroxymethyl tolterodine (PNU 200577)

    Catalog No. A11166
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    muscarinic receptor 拮抗剂
    5-hydroxymethyl tolterodine (PNU 200577)是托特罗定的代谢产物,tolterodine是一种用于治疗尿失禁的毒蕈碱受体拮抗剂。 了解更多
  15. Rocuronium bromide

    Catalog No. A10803
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    AchR 拮抗剂
    Rocuronium Bromide是一种竞争性AchR拮抗剂,用于现代麻醉中。 了解更多
  16. Biperiden HCl

    Catalog No. A10147
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    Muscarinic receptor antagonist
    Biperiden HCl是毒蕈碱受体拮抗剂,对M1亚型表现出一定的选择性。 了解更多
  17. Tolterodine tartrate (Detrol LA)

    Catalog No. A10937
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    muscarinic receptor 拮抗剂
    Tolterodine tartrate (Detrol LA)是毒蕈碱受体拮抗剂。 了解更多
  18. Solifenacin succinate

    Catalog No. A11215
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    muscarinic M3 receptor antagoinst
    Solifenacin succinate是毒蕈碱M3受体拮抗剂,用于治疗尿失禁。 了解更多
  19. Atropine

    Catalog No. A10098
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    mAChR 拮抗剂
    Atropine是M1,M2,M3,M4和M5型毒蕈碱乙酰胆碱受体的竞争性拮抗剂。 了解更多
  20. SVT-40776 (Tarafenacin)

    Catalog No. A10808
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    muscarinic receptor 拮抗剂
    SVT-40776 (Tarafenacin)是新型M3毒蕈碱受体拮抗剂,用于治疗膀胱过度活动症。 了解更多
  21. Orphenadrine citrate

    Catalog No. A11712
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    NMDA receptor 拮抗剂
    Orphenadrine柠檬酸盐是NMDA受体拮抗剂,Ki为6.0μM,还是HERG钾离子通道阻断剂。 了解更多
  22. Gallamine triethiodide

    Catalog No. A10417
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    mAChR M2 拮抗剂
    Gallamine Triethiodide是一种具有显著心脏选择性的mAChR M2拮抗剂。 了解更多
  23. Ipratropium bromide

    Catalog No. A10476
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    Ipratropium bromide是毒蕈碱拮抗剂、支气管扩张剂、阿托品的N-异丙基盐。 了解更多

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