“ab fubinaca”的搜索结果

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  1. Pyridostatin hydrochloride

    Catalog No. A21727
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    G-quadruplexe stabilizer
    Pyridostatin hydrochloride (RR82 hydrochloride) is a G-quadruplexe stabilizer, with a Kd of 490 nM. 了解更多
  2. Tafamidis meglumine

    Catalog No. A18045
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    transthyretin (TTR) stabilizer
    Tafamidis meglumine (Fx-1006A) is a potent and selective transthyretin (TTR) stabilizer, shows comparable potency and efficacy to the mutumant homotetramers V30M-TTR, V122I-TTR and wild type WT-TTR, with EC50s of 2.7-3.2 μM. 了解更多
  3. Nedocromil

    Catalog No. A10950
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    mast cell stabilizer
    Nedocromil is a medication considered as mast cell stabilizer which act to prevent wheezing, shortness of breath, and other breathing problems caused by asthma. It is administered by an inhaler under the brand name Tilade. 了解更多
  4. JI051

    Catalog No. A18774
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    Hes1-PHB2 interaction stabilizer
    JI051 is a stabilizer for the Hes1-PHB2 interaction, interacts with a cancer-associated protein chaperone prohibitin 2 (PHB2), induces cell-cycle arrest by inhibiting the Notch downstream effector gene Hes1. Anti-cancer activity. 了解更多
  5. ACR 16 hydrochloride

    Catalog No. A16074
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    dopaminergic stabilizer
    ACR 16 hydrochloride是一种多巴胺能稳定剂(对于D2(低)和D2(高),Ki值分别为17550 nM和7521),通过功能性多巴胺D2受体拮抗作用和皮质谷氨酸功能的双重作用,稳定地稳定精神运动活动。在各种情况下神经传递受到干扰。 了解更多
  6. PhiKan 083

    Catalog No. A15350
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    p53 stabilizer
    PhiKan 083是p53稳定剂;在与功能性DNA/蛋白质相互作用区域不同的位点,突变型(Y220C)p53优先结合野生型p53。 了解更多
  7. CP 31398 dihydrochloride

    Catalog No. A15346
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    p53 stabilizer
    CP 31398 dihydrochloride是p53稳定剂。在具有突变型或野生型p53的癌细胞系中稳定p53的活性构象并提高p53的活性。在体内抑制小的人类肿瘤异种移植物的生长。 了解更多
  8. CP 31398 2HCl

    Catalog No. A13522
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    p53 stabilizer
    CP 31398 2HCl已显示出可作为p53的稳定剂,并促进癌细胞系中p53的活性。 了解更多
  9. Sagopilone

    Catalog No. A14328
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    microtubule stabilizer
    Sagopilone是一种具有潜在抗肿瘤活性的全合成低分子量埃博霉素。 了解更多

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