“tak”的搜索结果

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  1. TAK 259

    Catalog No. A16186
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    α1D Adrenoceptor 拮抗剂
    TAK-259是一种新型的,选择性的,口服活性的α1D肾上腺素受体拮抗剂(α1D,Ki = 1.1 nM),具有抗尿频效应并减少人类以太相关基因(hERG)的责任。 了解更多
  2. TAK-779

    Catalog No. A13846
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    CCR5 拮抗剂
    TAK-779是一种新颖,有效和选择性的CCR5小分子拮抗剂,在结合试验中IC50值为1.4nM。 了解更多
  3. Relugolix

    Catalog No. A17783
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    GnRH antagonist
    Relugolix is a novel, non-peptide, orally active gonadotropin-releasing hormone (GnRH) antagonist with IC50 of 0.33 nM in the presence of 40% fetal bovine serum, TAK-385 possesses higher affinity and potent antagonistic activity compared with TAK-013. 了解更多
  4. Azilsartan D5

    Catalog No. A21600
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    angiotensin II type 1 receptor antagonist
    Azilsartan D5 is the deuterium labeled Azilsartan(TAK-536), which is a specific and potent angiotensin II type 1 receptor antagonist. 了解更多
  5. Azilsartan medoxomil monopotassium

    Catalog No. A20860
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    angiotensin II receptor type 1 antagonist
    Azilsartan medoxomil monopotassium is an orally administered angiotensin II receptor type 1 antagonist with IC50 of 0.62 nM, which used in the treatment of adults with essential hypertension. 了解更多
  6. Azilsartan Medoxomil

    Catalog No. A16420
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    angiotensin II receptor type 1 拮抗剂
    Azilsartan medoxomil是一种口服给药的1型血管紧张素II受体拮抗剂,IC50为0.62 nM。 了解更多
  7. BX471 hydrochloride

    Catalog No. A21886
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    non-peptide CCR1 antagonist
    BX471 hydrochloride (ZK-811752 hydrochloride) is a potent, selective non-peptide CCR1 antagonist with Ki of 1 nM for human CCR1, and exhibits 250-fold selectivity for CCR1 over CCR2, CCR5 and CXCR4. 了解更多
  8. Eplivanserin mixture

    Catalog No. A21987
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    serotonin reuptake inhibitor/5-HT2A receptor antagonist
    Eplivanserin mixture is a selective serotonin reuptake inhibitor and a 5-HT2A receptor antagonist, extracted from patent WO 2005/002578 A1. 了解更多

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