“MK 1775”的搜索结果

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  1. MK-0354

    Catalog No. A22008
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    GPR109a receptor agonist
    MK-0354 is a partial agonist of GPR109a receptor, for hGPR109a/ mGPR109a with EC50 of 1.65/1.08 μM, showed no activation of GPR109b. 了解更多
  2. LY 344864 hydrochloride

    Catalog No. A21748
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    5-HT1F agonist
    LY 344864 hydrochloride is a selective 5-HT1F agonist with a Ki of 6 nM. 了解更多
  3. Taranabant ((1R,2R)stereoisomer)

    Catalog No. A21705
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    CB1 receptor inverse agonist
    Taranabant (1R,2R)stereoisomer is the R-enantiomer of Taranabant. Taranabant is a highly potent and selective cannabinoid 1 (CB1) receptor inverse agonist. 了解更多
  4. MK-5046

    Catalog No. A21214
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    BRS-3 agonist
    MK-5046 is a novel BRS-3 agonist, binds to BRS-3 with high affinity (mouse Ki = 1.6 nM, human Ki = 25 nM). 了解更多
  5. Taranabant

    Catalog No. A11578
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    CB1 receptor inverse agonist
    Taranabant is a highly potent and selective cannabinoid 1 (CB1) receptor inverse agonist that inhibits the binding and functional activity of various agonists, with a binding Ki of 0.13 nM for the human CB1R in vitro. 了解更多
  6. MK-6913

    Catalog No. A12311
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    Estrogen receptor β agonist
    Tetrahydrofluoroene 52 is a potent and selective estrogen receptor β agonist. 了解更多
  7. TPA 023

    Catalog No. A20140
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    GABAA α2/α3 agonist
    TPA 023 is a GABAA α2/α3 subtype-selective agonist, with Ki of 0.19-0.41 nM. 了解更多
  8. Midodrine

    Catalog No. A17758
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    adrenergic alpha-1 agonist
    Midodrine is an ethanolamine derivative that is an adrenergic alpha-1 agonist. It is used as a vasoconstrictor agent in the treatment of HYPOTENSION. 了解更多
  9. Midodrine hydrochloride

    Catalog No. A17757
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    Adrenergic alpha-1 agonist
    Midodrine hydrochloride is an ethanolamine derivative that is an adrenergic alpha-1 agonist. It is used as a vasoconstrictor agent in the treatment of hypotension. It improves clinical outcome of chronic hypotension. 了解更多
  10. MK-6892

    Catalog No. A12982
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    GPR109A 激动剂
    MK-6892是高亲和力烟酸(NA)受体GPR109A的有效,选择性和完全激动剂。人GPR109A的MK-6892的Ki和GTPγSEC 50分别为4 nM和16 nM。 了解更多

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