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搜索结果：“tak”

“tak”的搜索结果

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TAK-875 (Fasiglifam)

Catalog No. A11018
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GPR 激动剂

TAK-875 (Fasiglifam)是一种有效的，选择性的GPR40激动剂。了解更多

Product Citations (3)

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- Ying Liu, .et al. A synthetic free fatty acid-regulated transgene switch in mammalian cells and mice, Nucleic Acids Res, 2018, Oct 12; 46(18): 9864-9874 PMID: 30219861
- Deborah A. Goldspink, .et al. Mechanistic insights into the detection of free fatty and bile acids by ileal glucagon-like peptide-1 secreting cells, Mol Metab, 2018, Jan; 7: 90-101 PMID: 29167062
- Hodaka Yamada, .et al. Potentiation of Glucose-stimulated Insulin Secretion by the GPR40-PLC-TRPC Pathway in Pancreatic β-Cells, Sci Rep, 2016, 6: 25912 PMID: 27180622
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Ramelteon (TAK-375)

Catalog No. A10777
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MT1/MT2-Receptor 激动剂

Ramelteon (TAK-375)是melatonin受体激动剂，对褪黑激素MT1（IC50 = 28.5±8.55 pM）和MT2（20.1±9.25 pM）受体均具有高亲和力，并且相对于MT3受体具有选择性。了解更多

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Mosapride citrate

Catalog No. A10607
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5-HT4-receptor 激动剂

Mosapride citrate起5-HT4受体激动剂和5-HT3受体拮抗剂的作用。了解更多

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Vilazodone D8

Catalog No. A21876
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SSR inhibitor / 5-HT1A receptor partial agonist

Vilazodone D8 is the a deuterium labeled vilazodone, which is a combined serotonin specific reuptake inhibitor (SSRI) and 5-HT1A receptor partial agonist. 了解更多

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YL-0919

Catalog No. A16337
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5-HT1A receptor 激动剂/serotonin reuptake 抑制剂

YL0919，具有5-HT1A受体激动剂和选择性5-羟色胺再摄取抑制剂双重活性的新型抗抑郁候选药物，YL-0919抑制5-HT被大鼠大脑皮层突触小体和人重组细胞摄取的IC50值为1.78±0.34 nM和1.93±0.18 nM。了解更多

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