“jwh 250”的搜索结果

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  1. Nicorandil

    Catalog No. A10641
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    Kir6 (KATP) channel opener
    Nicorandil (SG-75) 钾离子通道活化剂。 了解更多
  2. PETCM

    Catalog No. A15308
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    Caspase-3 activator
    PETCM是caspase-3的激活剂,也是HeLa细胞质中凋亡小体形成的刺激物。 了解更多
  3. OAC2

    Catalog No. A15931
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    Oct4 activator
    OAC2是一种Oct4激活化合物,可通过Oct4基因启动子激活表达。 了解更多
  4. Carglumic Acid

    Catalog No. A17588
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    CPS1 activator
    Carglumic acid (N-Carbamyl-L-glutamic acid), a functional analogue of N-acetylglutamate (NAG) and a carbamoyl phosphate synthetase 1 (CPS1) activator, is used to treat acute and chronic hyperammonemia associated with NAG synthase (NAGS) deficiency. 了解更多
  5. PAC-1

    Catalog No. A11090
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    Caspase activator
    PAC-1是procaspase-3的激活剂,可诱导癌细胞凋亡,EC50为2.08μM。 了解更多
  6. NS 309

    Catalog No. A11934
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    KCa3.1 channel activator
    NS 309是小和中电导Ca2+激活的K+通道(KCa2和KCa3.1通道)的正调制器。 了解更多
  7. Tenovin-1

    Catalog No. A11943
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    p53 activator
    Tenovin-1是p53转录活性的小分子激活剂,可防止MDM2介导的p53降解。 了解更多
  8. YC-1 (Lificiguat)

    Catalog No. A12402
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    sGC activator
    YC-1 (Lificiguat)是可溶性胍基环化酶(sGC)的直接活化剂,独立于一氧化氮。 了解更多
  9. OAC1

    Catalog No. A12931
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    Oct4 Activator
    OAC1通过增强Oct4和Nanog驱动的基因表达来增强iPSC重编程效率。 了解更多
  10. PS 48

    Catalog No. A13484
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    PDK1 抑制剂
    PS 48是一种变构磷酸肌醇依赖性蛋白激酶-1(PDK1)激活剂(Kd = 10.3μM)。 了解更多
  11. PRIMA-1

    Catalog No. A13581
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    p53 reactivator
    PRIMA-1是一种小分子,因其p53再激活作用而被鉴定。 了解更多
  12. Cannabichromene

    Catalog No. A15497
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    TRPA1 activatior/TRPM8 blocker
    Cannabichromene是一种主要的非精神植物大麻素,可抑制内源性大麻素失活并激活瞬时受体电位锚蛋白1(TRPA1)。内源性大麻素和TRPA1均可调节肠胃蠕动。 了解更多
  13. GSK621

    Catalog No. A15896
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    AMPK 激活剂
    GSK621是有效的选择性AMPK激动剂。 了解更多
  14. (-)-Indolactam V

    Catalog No. A13043
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    PKC activator
    (-)-Indolactam V是一种蛋白激酶C激活剂,可将人ES细胞衍生的定形内胚层强有力地引导至胰腺内胚层中。 了解更多
  15. PK11007

    Catalog No. A16833
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    p53 activator
    PK11007是一种抗p53药物,可通过两个表面暴露的半胱氨酸的选择性烷基化来稳定野生型和突变型p53,而不会损害其DNA结合活性。它不仅通过重新激活p53发挥抗肿瘤功能,还通过其他细胞机制发挥作用,例如将细胞ROS升高至毒性水平并激活UPR。 了解更多
  16. CBL-0137

    Catalog No. A16836
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    p53 activator / NF-κB 抑制剂
    CBL0137 (CBL-0137)在基于细胞的p53和NF-kB报告基因检测中分别激活p53和抑制NF-kB,EC50为0.37 uM和0.47 uM。它还抑制组蛋白伴侣FACT(促进染色质转录复合物)。 了解更多
  17. CDN1163

    Catalog No. A16951
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    SERCA2 allosteric activator
    CDN1163是SERCA2变构激活剂。它增加了肥胖小鼠的ER微粒体的Ca2+-ATPase活性和Ca2+吸收。从ER应激诱导的细胞死亡中拯救HEK细胞。 了解更多
  18. HLY78

    Catalog No. A18402
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    Wnt/β-catenin 激活剂
    HLY78 is an activator of the Wnt/β-catenin signaling pathway, which targets the DIX domain of Axin and potentiates the Axin-LRP6 association to promote Wnt signaling transduction. 了解更多
  19. SBI-797812

    Catalog No. A19058
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    NAMPT activator
    SBI-797812 is a novel NAMPT activator, elevating liver NAD+, turning NAMPT into a "super catalyst" that more efficiently generates NMN. 了解更多
  20. Y-26763

    Catalog No. A12271
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    K+ (KATP) channel activator
    Y-26763 is a K+ channel opener and active metabolite of Y-27152. Y-26763 is an ATP-sensitive K+ (KATP) channel activator. 了解更多
  21. LYN-1604 hydrochloride

    Catalog No. A21449
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    ULK1 activator
    LYN-1604 hydrochloride is a potent ULK1 activator with an EC50 of 18.94 nM. 了解更多
  22. NS 11021

    Catalog No. A21710
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    KCa1.1 channels activator
    NS 11021 is a potent and specific Ca2-activated big-conductance K?? Channels (KCa1.1 channels) activator. 了解更多

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