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搜索结果：“Ligand-gated Ion Channels”

“Ligand-gated Ion Channels”的搜索结果

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(-)-BAY-1251152

Catalog No. A21570
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PTEF/CDK9 inhibitor

(-)-BAY-1251152 is an enanthiomer of BAY-1251152 with rotation (-). BAY-1251152 is a potent and highly selective PTEF/CDK9 inhibitor. 了解更多

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CDK9-IN-1

Catalog No. A21552
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CDK9 inhibitor

CDK9-IN-1 is a novel, selective CDK9 inhibitor for the treatment of HIV infection, with an IC50 of 39 nM for CDK9/CycT1, extracted from reference, compound 87. 了解更多

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Ca2+ channel agonist 1

Catalog No. A12186
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Ca2+ channel agonist/CDK2 inhibitor

Ca2+ channel agonist 1 is an agonist of N-type Ca2+ channel and an inhibitor of Cdk2, with EC50s of 14.23 μM and 3.34 μM, respectively, and is used as a potential treatment for motor nerve terminal dysfunction. 了解更多

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bio-THZ1

Catalog No. A18559
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covalent CDK7 inhibitor

bio-THZ1 is a biotinylated version of THZ1 and binds irreversibly to CDK7. THZ1 is a selective and potent covalent CDK7 inhibitor with an IC50 of 3.2 nM. 了解更多

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PD 0332991 Isethionate

Catalog No. A13811
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CDK4/6 抑制剂

PD 0332991 Isethionate是CDK4/6的高选择性抑制剂，IC50分别为11 nM/16 nM。了解更多

Product Citations (1)

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- K Keegan ,etc. Preclinical evaluation of AMG 925, a FLT3/CDK4 dual kinase inhibitor for treating acute myeloid leukemia. Molecular cancer therapeutics, 2014, 13(4), 880-889.