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  • 搜索结果：“Ligand-gated Ion Channels”

“Ligand-gated Ion Channels”的搜索结果

17 个项目

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  1. RI-2
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    RI-2

    Catalog No. A20992
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    RAD51 inhibitor
    RI-2 is a reversible RAD51 inhibitor, with an IC50 of 44.17 μM, and specifically inhibits homologous recombination repair in human cells. 了解更多
  2. (-)-BAY-1251152
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    (-)-BAY-1251152

    Catalog No. A21570
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    PTEF/CDK9 inhibitor
    (-)-BAY-1251152 is an enanthiomer of BAY-1251152 with rotation (-). BAY-1251152 is a potent and highly selective PTEF/CDK9 inhibitor. 了解更多
  3. CDK9-IN-1
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    CDK9-IN-1

    Catalog No. A21552
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    CDK9 inhibitor
    CDK9-IN-1 is a novel, selective CDK9 inhibitor for the treatment of HIV infection, with an IC50 of 39 nM for CDK9/CycT1, extracted from reference, compound 87. 了解更多
  4. Ca2+ channel agonist 1
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    Ca2+ channel agonist 1

    Catalog No. A12186
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    Ca2+ channel agonist/CDK2 inhibitor
    Ca2+ channel agonist 1 is an agonist of N-type Ca2+ channel and an inhibitor of Cdk2, with EC50s of 14.23 μM and 3.34 μM, respectively, and is used as a potential treatment for motor nerve terminal dysfunction. 了解更多
  5. AAPK-25
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    AAPK-25

    Catalog No. A19085
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    Aurora/PLK dual 抑制剂
    AAPK-25 is a potent and selective Aurora/PLK dual inhibitor with anti-tumor activity, which can cause mitotic delay and arrest cells in a prometaphase, reflecting by the biomarker histone H3Ser10 phosphorylation and followed by a surge in apoptosis. 了解更多
  6. ZT-12-037-01
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    ZT-12-037-01

    Catalog No. A18395
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    ATP-competitive STK19 inhibitor
    ZT-12-037-01 is a potent, selective, ATP-competitive STK19 inhibitor. ZT-12-037-01 effectively blocks oncogenic NRAS-driven melanocyte malignant transformation and melanoma growth in vitro and in vivo. 了解更多
  7. bio-THZ1
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    bio-THZ1

    Catalog No. A18559
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    covalent CDK7 inhibitor
    bio-THZ1 is a biotinylated version of THZ1 and binds irreversibly to CDK7. THZ1 is a selective and potent covalent CDK7 inhibitor with an IC50 of 3.2 nM. 了解更多
  8. R-10015
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    R-10015

    Catalog No. A18806
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    LIMK inhibitor
    R-10015, a broad-spectrum antiviral compound for HIV infection, acts as a potent and selective inhibitor of LIM domain kinase (LIMK) and binds to the ATP-binding pocket, with an IC50 of 38 nM for human LIMK1. 了解更多
  9. MRTX1257
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    MRTX1257

    Catalog No. A17223
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    KRAS-G12C inhibitor
    MRTX1257 is a potent, selective, covalent and irreversible inhibitor of KRAS G12C, MRTX1257 inhibited KRAS dependent ERKphosphorylation in the H358cell assay with an IC50= 900 pM. 了解更多
  10. CCT245737
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    CCT245737

    Catalog No. A17239
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    CHK1 inhibitor
    CCT245737 is a potent, selective and orally active checkpoint kinase 1 (CHK1) inhibitor. CCT245737 showed CHK1 IC50 = 1.3 nM, CHK2 IC50 = 2440 nM, G2 check point abrogation IC50 = 30 nM. Mouse F (oral)=100%. 了解更多
  11. Ripasudil
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    Ripasudil

    Catalog No. A15888
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    ROCK inhibitor
    Ripasudil (K-115) is potent ROCK inhibitor with IC50 of 51 nM and 19 nM for ROCK1 and ROCK2, respectively, used for the treatment of glaucoma and ocular hypertension. 了解更多
  12. PD 0332991 Isethionate
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    PD 0332991 Isethionate

    Catalog No. A13811
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    CDK4/6 抑制剂
    PD 0332991 Isethionate是CDK4/6的高选择性抑制剂，IC50分别为11 nM/16 nM。 了解更多
  13. NSC-23766 HCl
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    NSC-23766 HCl

    Catalog No. A13975
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    Rac GTPase 抑制剂
    NSC 23766是Rac特异性GEF TrioN和Tiam 1（IC50 = 50 uM）引起的Rac1激活的细胞可渗透性可逆抑制剂。 了解更多
  14. EHop-016
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    EHop-016

    Catalog No. A12740
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    Rac GTPase Inhibitor
    EHop-016 is a potent and specific inhibitor of Rac1 and Rac3 GTPase activity that inhibits Vav2 interaction with Rac, Rac-activated PAK1, lamellipodia formation, and cell migration. 了解更多
  15. Kobe0065
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    Kobe0065

    Catalog No. A13135
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    Ras-Raf interaction 抑制剂
    Kobe0065抑制锚定依赖性和非依赖性生长，阻断MEK / ERK活性并诱导H-rasG12V转化的NIH3T3细胞凋亡。 了解更多
  16. NSC 23766
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    NSC 23766

    Catalog No. A12546
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    Rac1 activation 抑制剂
    SC 23766是Rac1-GEF相互作用的选择性抑制剂。通过Rac特异性鸟嘌呤核苷酸交换因子（GEF）TrioN和Tiam1（IC50为50 μM）阻止Rac1激活，而不影响Cdc42或RhoA激活。 了解更多
  17. Zoledronic Acid
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    Zoledronic Acid

    Catalog No. A11010
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    osteoclastic bone resorption 抑制剂
    Zoledronic acid, 破骨细胞抑制剂，通过抑制甲羟戊酸途径诱导破骨细胞凋亡。 了解更多

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  1. Chk (2)
  2. CDK (5)
  3. Aurora Kinase (1)
  4. PLK (1)
  5. ROCK (2)
  6. Ras (7)
  7. RAD51 (1)
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