“MK-2206 dihydrochloride”的搜索结果

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  1. GDC-0575 dihydrochloride

    Catalog No. A21567
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    CHK1 inhibitor
    GDC-0575 dihydrochloride (ARRY-575 dihydrochloride) is an orally bioavailable CHK1 inhibitor, with an IC50 of 1.2 nM, and has antitumor activity. 了解更多
  2. Lerociclib dihydrochloride

    Catalog No. A21577
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    CDK4/CDK6 inhibitor
    Lerociclib dihydrochloride (G1T38 dihydrochloride) is a potent and selective inhibitor of CDK4/CDK6, with IC50s of 1 nM and 2 nM for CDK4/CyclinD1 and CDK6/CyclinD3, respectively. 了解更多
  3. H-1152 dihydrochloride

    Catalog No. A15102
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    ROCK 抑制剂
    H-1152 dihydrochloride是一种异喹啉磺酰胺衍生物,是Rho激酶的一种更特异,更强且可透过膜的抑制剂,Ki值为1.6 nM,但对其他丝氨酸/苏氨酸激酶的抑制作用较弱。 了解更多
  4. HA-1077 dihydrochloride

    Catalog No. A13785
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    ROCK 抑制剂
    HA-1077 dihydrochloride通过充当细胞内Ca2+拮抗剂来抑制血管平滑肌收缩。 了解更多
  5. SR 3677 dihydrochloride

    Catalog No. A12674
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    ROCK 抑制剂
    SR 3677 dihydrochloride是一种有效的选择性Rho激酶抑制剂(ROCK-II和ROCK-I的IC50值分别为3和56 nM)。 了解更多
  6. Y-33075 dihydrochloride

    Catalog No. A11611
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    ROCK inhibitor
    Y-33075 dihydrochloride is a selective ROCK inhibitor with an IC50 of 3.6 nM. 了解更多

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