“betaine hydrochloride”的搜索结果

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  1. Niraparib hydrochloride

    Catalog No. A18018
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    PARP1 and PARP2 inhibitor
    Niraparib hydrochloride (MK-4827 hydrochloride) is a highly potent and orally bioavailable PARP1 and PARP2 inhibitor with IC50s of 3.8 and 2.1 nM, respectively. 了解更多
  2. Resminostat hydrochloride

    Catalog No. A15220
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    HDAC 抑制剂
    Resminostat hydrochloride是HDAC1/3/6的有效抑制剂(IC50 = 43-72 nM);对HDAC8的效力较低,IC50为877 nM。 了解更多
  3. Givinostat hydrochloride

    Catalog No. A21487
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    HDAC inhibitor
    Givinostat hydrochloride (ITF-2357 hydrochloride) is a HDAC inhibitor with an IC50 of 198 and 157 nM for HDAC1 and HDAC3, respectively. 了解更多
  4. CX-6258 hydrochloride hydrate

    Catalog No. A15055
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    Pim 抑制剂
    CX-6258 hydrochloride hydrate是一种有效的,口服有效的Pim 1/2/3激酶(IC50 = 5 nM/25 nM/16 nM)抑制剂,具有出色的生化效能和激酶选择性。 了解更多
  5. SCH-1473759 hydrochloride

    Catalog No. A21711
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    Aurora inhibitor
    SCH-1473759 hydrochloride is an aurora inhibitor with IC50s of 4 and 13 nM for aurora A and B, respectively. 了解更多
  6. SRT 1720 Hydrochloride

    Catalog No. A21143
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    SIRT1 activator of
    SRT 1720 Hydrochloride is a selective activator of SIRT1 with an EC50 of 0.10 μM, and shows less potent activities on SIRT2 and SIRT3. 了解更多
  7. NS-018 hydrochloride

    Catalog No. A16225
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    JAK2 抑制剂
    NS-018 hydrochloride是一种新型的高选择性JAK2抑制剂。 了解更多
  8. PJ 34 hydrochloride

    Catalog No. A12665
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    PARP 抑制剂
    PJ 34 hydrochloride是聚(ADP-核糖)聚合酶(PARP)(EC50 = 20 nM)的有效抑制剂。 了解更多
  9. T-3775440 hydrochloride

    Catalog No. A18340
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    LSD1 inhibitor
    T-3775440 (hydrochloride) is an irreversible lysine-specific histone demethylase (LSD1) inhibitor with an IC50 value of 2.1 nM. 了解更多
  10. Tranylcypromine hydrochloride

    Catalog No. A13358
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    LSD1/BHC110 & MAO 抑制剂
    Tranylcypromine hydrochloride是一种非选择性的MAO-A/B抑制剂。 了解更多
  11. Veliparib dihydrochloride

    Catalog No. A21356
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    PARP inhibitor
    Veliparib dihydrochloride is a potent PARP inhibitor, inhibiting PARP1 and PARP2 with Kis of 5.2 and 2.9 nM, respectively. 了解更多
  12. GSK-LSD1 dihydrochloride

    Catalog No. A21815
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    LSD1 inhibitor
    GSK-LSD1 dihydrochloride is a potent, selective and irreversible lysine specific demethylase 1 (LSD1) inhibitor with an IC50 of 16 nM. 了解更多
  13. NVP-BSK805 dihydrochloride

    Catalog No. A21406
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    JAK2 inhibitor
    NVP-BSK805 dihydrochloride (BSK805 dihydrochloride) is an ATP-competitive JAK2 inhibitor, with IC50s of 0.48 nM, 31.63 nM, 18.68 nM, and 10.76 nM for JAK2 JH1 (JAK homology 1), JAK1 JH1, JAK3 JH1, and TYK2 JH1, respectively. 了解更多
  14. Amodiaquine dihydrochloride dihydrate

    Catalog No. A16405
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    Amodiaquine dihydrochloride dihydrate是人红细胞中组胺N-甲基转移酶的有效,非竞争性抑制剂,也用作抗疟疾和抗炎药。 了解更多
  15. HLCL-61

    Catalog No. A15870
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    PRMT5 抑制剂
    HLCL-61 hydrochloride是一种有效的选择性PRMT5抑制剂,可用于治疗急性髓细胞性白血病。 了解更多
  16. UNC 926 hydrochloride

    Catalog No. A15367
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    MBT Domain (L3MBTL1) 抑制剂
    UNC 926 hydrochloride是甲基赖氨酸阅读器域抑制剂。 了解更多

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