“AZ 960”的搜索结果

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  1. Nec-4

    Catalog No. A21033
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    RIP1 inhibitor
    Nec-4, a tricyclic derivative, is a potent receptor interacting protein 1 (RIP1) inhibitor, with an IC50 of 2.6 μM, Ki of 0.46 μM. 了解更多
  2. RIPK1-IN-3

    Catalog No. A19023
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    RIPK1 inhibitor
    RIPK1-IN-3 (Example 38), a RIPK1 inhibitor, extracted from patent WO2018148626A1, possesses anti-inflammatory proprieties. 了解更多
  3. GSK481

    Catalog No. A12615
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    RIP1 抑制剂
    GSK481是新型的RIP1抑制剂苯并a庚酮(BOAz)系列。受体相互作用蛋白激酶1(RIP1)已被认为是通过调节程序性坏死调节炎症的关键因素。已显示对该激酶的抑制作用可阻止细胞坏死,从而将RIP1确定为潜在治疗多种炎性疾病的可行靶标。 了解更多

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