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  1. Ruxolitinib sulfate

    Catalog No. A11467
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    JAK1/2 inhibitor
    Ruxolitinib sulfate (INCB018424 sulfate) is the first potent, selective JAK1/2 inhibitor to enter the clinic with IC50s of 3.3 nM/2.8 nM, and has > 130-fold selectivity for JAK1/2 versus JAK3. 了解更多
  2. CYT387 sulfate salt

    Catalog No. A15056
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    JAK 抑制剂
    CYT387 sulfate salt是JAK1/JAK2的ATP竞争性抑制剂,IC50为11 nM/18 nM,是JAK3的约10倍选择性。 了解更多

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