“jwh 073”的搜索结果

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  1. AMG 073 (Cinacalcet)

    Catalog No. A11314
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    CaSR activator
    AMG 073 (Cinacalcet)是一类治疗甲状旁腺功能亢进的新型化合物。 了解更多
  2. AMG-073 HCl (Cinacalcet HCl)

    Catalog No. A10219
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    CaSR activator
    AMG-073 HCl(Cinacalcet HCl)是一种用于治疗甲状旁腺功能亢进的化合物,称为拟钙剂,通过增加甲状旁腺钙敏感受体(CaR)对细胞外钙的敏感性来减少甲状旁腺激素(PTH)的合成和分泌 。 了解更多
  3. Cenerimod

    Catalog No. A20913
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    S1P1 agonist
    Cenerimod (ACT-334441) is a potent and orally available sphingosine 1-phosphate 1 receptor (S1P1) agonist extracted from patent WO 2016184939 A1 and WO 2011007324 A1, example 1, with an EC50 of 2.7 nM. 了解更多
  4. Loxapine

    Catalog No. A18073
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    D2DR/D4DR inhibitor
    Loxapine Succinate is a D2DR and D4DR inhibitor, serotonergic receptor antagonist and also a dibenzoxazepine anti-psychotic agent. 了解更多
  5. Rauwolscine

    Catalog No. A13426
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    α2-adrenergic receptor 拮抗剂
    Rauwolscine是一种天然生物碱,具有选择性和可逆性α2肾上腺素能受体拮抗剂(Ki = 12 nM)。 了解更多
  6. Clemizole

    Catalog No. A13073
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    H1 histamine receptor 拮抗剂.
    Clemizole是H1组胺受体拮抗剂。 了解更多

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