“jwh 370”的搜索结果

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  1. Mosapride citrate

    Catalog No. A10607
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    5-HT4-receptor 激动剂
    Mosapride citrate起5-HT4受体激动剂和5-HT3受体拮抗剂的作用。 了解更多
  2. Carbetocin

    Catalog No. A18080
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    peripheral oxytocin receptors agonist
    Carbetocin (Lonactene; Duratocin) is an obstetric drug used to control postpartum hemorrhage and bleeding after giving birth; an agonist at peripheral oxytocin receptors. 了解更多
  3. Pancopride

    Catalog No. A12967
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    5-HT3 receptor antagonist
    Pancopride is a new potent and selective 5-HT3 receptor antagonist. 了解更多
  4. PS372424

    Catalog No. A19421
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    Human CXCR3 拮抗剂
    PS372424, a three amino-acid fragment of CXCL10, is a specific human CXCR3 agonist with anti-inflammatory activity, which inhibits the binding of CXCR3 ligand CXCL10 to CXCR3 receptor with IC50 of 42 nM. 了解更多
  5. Alprenolol hydrochloride

    Catalog No. A17781
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    5-HT1A receptor antagonist
    Alprenolol (hydrochloride) is a non-selective beta blocker as well as 5-HT1A receptor antagonist. 了解更多
  6. VU6005649

    Catalog No. A17023
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    CNS penetrant mGlu7/8 receptor 激动剂
    VU6005649是一种CNS渗透性mGlu7/8受体激动剂,对mGlu7受体和mGlu8受体的EC50分别为0.65 μM和2.6 μM。 了解更多
  7. LY 334370 hydrochloride

    Catalog No. A17027
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    5-HT1F 激动剂
    LY 334370 hydrochloride是一种选择性的5-HT1F受体激动剂(Ki值为1.87、16.4,> 100 (IC50))。CAS:199673-74-0(LY 334370盐酸盐);182563-08-2(LY 334370游离碱) 了解更多
  8. Tradipitant

    Catalog No. A16918
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    NK1 receptor 拮抗剂
    Tradipitant,也称为VLY-686和LY686017,是第二代神经激肽1受体拮抗剂,在临床前焦虑模型中表现出活性。 了解更多
  9. Naloxegol Oxalate

    Catalog No. A15972
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    Opioid 拮抗剂
    Naloxegol Oxalate是用于治疗阿片类药物引起的便秘的外周选择性阿片类药物拮抗剂。 了解更多
  10. PF-3274167

    Catalog No. A13754
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    Oxytocin 拮抗剂
    PF-3274167是一种高亲和力非肽催产素受体(OTR)拮抗剂,Ki为9.5 nM。 了解更多
  11. SCH 563705

    Catalog No. A15234
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    CXCR2/CXCR1 拮抗剂
    SCH 563705是有效的双重CXCR2(IC50 = 1.3 nM)/CXCR1(IC50 = 7.3 nM)拮抗剂。 了解更多
  12. Bromocriptin mesylate

    Catalog No. A13705
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    dopamine D2 receptor 激动剂
    Bromocriptin mesylate是一种有效的多巴胺受体激动剂,它以最高的亲和力(Ki = 2.5 nM)与D2受体结合。 了解更多
  13. ESI-09

    Catalog No. A14233
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    EPAC1/EPAC2 抑制剂
    ESI-09是一种直接由cAMP(EPAC)抑制剂激活的特异性交换蛋白,对于EPAC1和EPAC2,IC50为3.2 uM和1.4 uM。 了解更多

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