“tak”的搜索结果

18 个项目

每页

设置降序顺序
  1. TAK 259

    Catalog No. A16186
    Quick View
    α1D Adrenoceptor 拮抗剂
    TAK-259是一种新型的,选择性的,口服活性的α1D肾上腺素受体拮抗剂(α1D,Ki = 1.1 nM),具有抗尿频效应并减少人类以太相关基因(hERG)的责任。 了解更多
  2. Ramelteon (TAK-375)

    Catalog No. A10777
    Quick View
    MT1/MT2-Receptor 激动剂
    Ramelteon (TAK-375)是melatonin受体激动剂,对褪黑激素MT1(IC50 = 28.5±8.55 pM)和MT2(20.1±9.25 pM)受体均具有高亲和力,并且相对于MT3受体具有选择性。 了解更多
  3. Mosapride citrate

    Catalog No. A10607
    Quick View
    5-HT4-receptor 激动剂
    Mosapride citrate起5-HT4受体激动剂和5-HT3受体拮抗剂的作用。 了解更多
  4. GBR 12935

    Catalog No. A21951
    Quick View
    dopamine reuptake inhibitor
    GBR 12935 is a potent, and selective dopamine reuptake inhibitor. 了解更多
  5. Eplivanserin mixture

    Catalog No. A21987
    Quick View
    serotonin reuptake inhibitor/5-HT2A receptor antagonist
    Eplivanserin mixture is a selective serotonin reuptake inhibitor and a 5-HT2A receptor antagonist, extracted from patent WO 2005/002578 A1. 了解更多
  6. Vanoxerine

    Catalog No. A21922
    Quick View
    dopamine reuptake inhibitor
    Vanoxerine (GBR-12909) is a competitive, potent, and highly selective dopamine reuptake inhibitor (Ki=1 nM). 了解更多
  7. Vilazodone D8

    Catalog No. A21876
    Quick View
    SSR inhibitor / 5-HT1A receptor partial agonist
    Vilazodone D8 is the a deuterium labeled vilazodone, which is a combined serotonin specific reuptake inhibitor (SSRI) and 5-HT1A receptor partial agonist. 了解更多
  8. SPD-473 citrate

    Catalog No. A12617
    Quick View
    serotonin/dopamine/norepinephrine reuptake inhibitior
    SPD-473 citrate is a serotonin/dopamine/norepinephrine reuptake inhibitior. 了解更多
  9. YL-0919

    Catalog No. A16337
    Quick View
    5-HT1A receptor 激动剂/serotonin reuptake 抑制剂
    YL0919,具有5-HT1A受体激动剂和选择性5-羟色胺再摄取抑制剂双重活性的新型抗抑郁候选药物,YL-0919抑制5-HT被大鼠大脑皮层突触小体和人重组细胞摄取的IC50值为1.78±0.34 nM和1.93±0.18 nM。 了解更多
  10. Desvenlafaxine succinate hydrate

    Catalog No. A15491
    Quick View
    serotonin (5-HT)/norepinephrine (NE) reuptake 抑制剂
    Desvenlafaxine succinate hydrate是一种新型5-羟色胺(5-HT)转运蛋白 和去甲肾上腺素(NE)转运蛋白重吸收抑制剂,Ki值分别为40.2 nM和558.4 nM 了解更多
  11. Phenylpiracetam

    Catalog No. A15211
    Quick View
    Dopamine reuptake 抑制剂
    Phenylpiracetam是促智药物吡乙酰胺的苯基化衍生物。它被用作促智药物,效力比吡乙酰胺高30-60倍。 了解更多
  12. Norfluoxetine

    Catalog No. A13458
    Quick View
    serotonin uptake 抑制剂
    Norfluoxetine是抗抑郁药氟西汀的活性代谢物,抑制5-羟色胺的摄取,pKi值为7.35.1氟西汀的S-对映体的5-羟色胺再摄取阻断能力是R-对映体的20倍(pKis分别为7.86和6.51)。 了解更多
  13. Edivoxetine HCl

    Catalog No. A13865
    Quick View
    norepinephrine reuptake 抑制剂
    Edivoxetine HCl是一种选择性去甲肾上腺素再摄取抑制剂。 了解更多
  14. Levomilnacipran HCl

    Catalog No. A14391
    Quick View
    serotonin/NE reuptake 抑制剂
    Levomilnacipran HCl是一种选择性的5-羟色胺和去甲肾上腺素再摄取抑制剂。 了解更多
  15. GBR 12783 dihydrochloride

    Catalog No. A13128
    Quick View
    dopamine uptake 抑制剂
    GBR 12783 dihydrochloride是一种非常有效的选择性多巴胺摄取抑制剂(抑制大鼠纹状体突触体中[3H]-多巴胺摄取的IC50为1.8 nM)。 了解更多
  16. Maprotiline hydrochloride

    Catalog No. A10555
    Quick View
    noradrenalin re-uptake 抑制剂
    Maprotiline hydrochloride是选择性去甲肾上腺素再摄取抑制剂。 了解更多
  17. Vanoxerine 2HCl (GBR-12909)

    Catalog No. A10725
    Quick View
    dopamine re-uptake 抑制剂
    Vanoxerine 2HCl (GBR-12909)是哌嗪衍生物,是一种有效的、选择性的多巴胺摄取(dopamine uptake)抑制剂。 了解更多
  18. Vilazodone

    Catalog No. A11116
    Quick View
    Serotonin reuptake 抑制剂
    Vilazodone充当5-羟色胺再摄取抑制剂(IC50 = 0.5 nM)和5-HT1A受体部分激动剂(IC50 = 0.2 nM; IA =?60-70%)。 了解更多

18 个项目

每页

设置降序顺序
Rewards