“Gefitinib”的搜索结果

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  1. FAAH-IN-2

    Catalog No. A20528
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    FAAH inhibitor
    FAAH-IN-2 (O-Desmorpholinopropyl Gefitinib) is a potent FAAH(fatty acid amide hydrolase) inhibitor extracted from Patent WO/2008/100977A2. 了解更多
  2. Gefitinib hydrochloride

    Catalog No. A15093
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    EGFR 抑制剂
    Gefitinib hydrochloride是一种EGFR抑制剂,可通过靶细胞中的表皮生长因子受体(EGFR)中断信号传导。因此,它仅在EGFR突变和过度活跃的癌症中有效。 了解更多
  3. Gefitinib (Iressa)

    Catalog No. A10422
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    EGFR 抑制剂
    Gefitinib (Iressa)是一种EGFR抑制剂,可阻断靶细胞中表皮生长因子受体(EGFR)的信号传导。 了解更多
  4. Gefitinib-based PROTAC 3

    Catalog No. A19093
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    Gefitinib-based PROTAC 3, conjugating an EGFR binding element to a VHL ligand via a linker, induces EGFR degradation with DC50s of 11.7 nM and 22.3 nM in HCC827(exon 19 del) and H3255 (L858R mutantion) cells, respectively. 了解更多
  5. MC-Sq-Cit-PAB-Gefitinib

    Catalog No. A18521
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    MC-Sq-Cit-PAB-Gefitinib is a drug-linker conjugate for ADC with potent antitumor activity by using Gefitinib (an EGFR tyrosine kinase inhibitor), linked via the ADC linker MC-Sq-Cit-PAB. 了解更多

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