“2c c hcl”的搜索结果

产品 401 到 450 共 16088个

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  1. Solamargine

    Catalog No. A22357
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    anticancer agent
    Solamargine, a derivative from the steroidal solasodine in Solanum species, exhibits anticancer activities in numerous types of cancer. Solamargine induces non-selective cytotoxicity and P-glycoprotein inhibition. 了解更多
  2. Skatole

    Catalog No. A22359
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    bacteriostatic agent
    Skatole (3-methylindole, Scatole) is a mildly toxic white crystalline organic compound that occurs naturally in feces. It has a fairly broad bacteriostatic effect.. 了解更多
  3. 3BDO

    Catalog No. A22360
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    mTOR activator
    3BDO is a new mTOR activator which can also inhibit autophagy. 了解更多
  4. TG-89

    Catalog No. A22361
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    JAK2 inhibitor
    TG-89 is an inhibitor of JAK2 with IC50 of 11.2 μM. 了解更多
  5. BMP signaling agonist sb4

    Catalog No. A22362
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    BMP4 signaling agonist
    BMP signaling agonist sb4 is a potent benzoxazole bone morphogenetic protein 4 (BMP4) signaling agonist with a EC50 value of 74 nM, activates BMP signaling by stabilizing intracellular p-SMAD-1/5/9. 了解更多
  6. 5-Bromoindole

    Catalog No. A22363
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    inhibitor of glycogen synthase kinase 3
    5-bromoindole is an important pharmaceutical chemical intermediate and a potential inhibitor of glycogen synthase kinase 3 (GSK-3). 了解更多
  7. Remimazolam

    Catalog No. A22200
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    benzodiazepine derivative drug
    Remimazolam, also known as CNS-7056, is a benzodiazepine derivative drug, developed by PAION, in collaboration with Japanese licensee Ono Pharmaceutical as an alternative to the short-acting imidazobenzodiazepine midazolam, for use in induction of anaesthesia and conscious sedation for minor invasive procedures. 了解更多
  8. Avacopan

    Catalog No. A22202
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    selective C5aR antagonist
    Avacopan (CCX168) is an orally administered and selective C5a receptor (C5aR) antagonist. 了解更多
  9. Perlapine

    Catalog No. A22204
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    hM3Dq DREADD agonist
    Perlapine is a potent and selective hM3Dq DREADD agonist (EC50 = 2.8 nM). This drug exhibits >10,000-fold selectivity for hM3Dq over hM3. 了解更多
  10. Durlobactam sodium

    Catalog No. A13801
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    beta-lactamase inhibitor drug candidate
    Durlobactam, also known as ETX2514, is a beta-lactamase inhibitor drug candidate. 了解更多
  11. Ozogamicin

    Catalog No. A12672
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    antibody-drug conjugate Linker
    Ozogamicin is an antibody-drug conjugate Linker. 了解更多
  12. Etanercept

    Catalog No. A12009
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    TNF inhibitor
    Etanercept, a dimeric fusion protein that binds TNF, acts as a TNF inhibitor. 了解更多
  13. Dehydroascorbic acid

    Catalog No. A12366
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    potent cerebroprotection
    Dehydroascorbic acid, a blood-brain barrier transportable form of vitamin C, mediates potent cerebroprotection in experimental stroke. 了解更多
  14. Emedastine

    Catalog No. A22158
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    histamine H1 receptor antagonist
    Emedastine is an orally active, selective and high affinity histamine H1 receptor antagonist with a Ki value of 1.3 nM. 了解更多
  15. IACS-13909

    Catalog No. A22159
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    SHP2 allosteric inhibitor
    IACS-13909 is a selective, potent and orally active SHP2 allosteric inhibitor with an IC50 of 15.7 nM and a Kd of 32 nM. 了解更多
  16. CB-103

    Catalog No. A22160
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    protein-protein interaction (PPI) inhibitor
    CB-103 is a first-in-class, orally active protein-protein interaction (PPI) inhibitor of the NOTCH transcriptional activation complex. CB-103 has anti-tumor activity. 了解更多
  17. CRBN modulator-1

    Catalog No. A22161
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    CRBN modulator
    CRBN modulator-1, a Thalidomide analog and a CRBN modulator extracted from WO2020006262A1, compound 10, has an IC50 of 3.5 μM and a Ki of 0.98 μM. 了解更多
  18. ATR inhibitor 2

    Catalog No. A22162
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    ATR inhibitor
    ATR inhibitor 2 is an ATP-competitive, orally active, and selective ATR inhibitor, with a Ki of <150 pM. 了解更多
  19. Cenobamate

    Catalog No. A22163
    antiepileptic drug
    Cenobamate (YKP-3089) is a novel antiepileptic drug candidate with broad-spectrum anticonvulsant activity. 了解更多
  20. JSH-150

    Catalog No. A22164
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    CDK9 inhibitor
    JSH-150 is a highly selective and potent CDK9 inhibitor with an IC50 of 1 nM. 了解更多
  21. Molnupiravir

    Catalog No. A22165
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    broad-spectrum antiviral activity
    Molnupiravir (EIDD-2801, MK-4482) is an orally bioavailable prodrug of the ribonucleoside analog β-d-N4-hydroxycytidine (NHC; EIDD-1931) with broad-spectrum antiviral activity against SARS-CoV-2, MERS-CoV, SARS-CoV, and the causative agent of COVID-19. 了解更多
  22. Laninamivir octanoate

    Catalog No. A22166
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    neuraminidase (NA) inhibitor
    Laninamivir octanoate (CS-8958), a prodrug of Laninamivir, is a long-acting neuraminidase (NA) inhibitor with anti-influenza virus activity. 了解更多
  23. Conoidin A

    Catalog No. A22167
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    cell permeable inhibitor
    Conoidin A is a cell permeable inhibitor of T. gondii enzyme peroxiredoxin II (TgPrxII). 了解更多
  24. ML382

    Catalog No. A22168
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    MRGPRX1 positive allosteric modulator
    ML382 is a potent and selective MRGPRX1 (Mas-related G protein-coupled receptor X1, MrgX1) positive allosteric modulator, with an EC50 of 190 nM. 了解更多
  25. GRP-60367

    Catalog No. A22169
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    rabies virus (RABV) entry inhibitor
    GRP-60367 is a first-in-class small-molecule rabies virus (RABV) entry inhibitor with nanomolar potency against some RABV strains. 了解更多
  26. Lycorine

    Catalog No. A22170
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    SCAP inhibitor
    Lycorine is a natural alkaloid extracted from the Amaryllidaceae plant. Lycorine is a potent and orally active SCAP inhibitor with a Kd value 15.24 nM. 了解更多
  27. Eurycomanone

    Catalog No. A22171
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    Eurycomanone could increases spermatogenesis by inhibiting the activity of phosphodiesterase and aromatase in steroidogenesis. 了解更多
  28. Gentiopicroside

    Catalog No. A22172
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    antianti-inflammatoryand antioxidative effects
    Gentiopicroside, a naturally occurring iridoid glycoside, inhibits P450 activity, with an IC50 and a Ki of 61 ?M and 22.8 ?M for CYP2A6; Gentiopicroside has antianti-inflammatoryand antioxidative effects. 了解更多
  29. Eleutheroside B1

    Catalog No. A22173
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    anti-human influenza virus efficacy
    Eleutheroside B1, a coumarin compound, has a wide spectrum of anti-human influenza virus efficacy, with an IC50 value of 64-125 ?g/ml. Antiviral and anti-inflammatory activities. 了解更多
  30. Periplogenin

    Catalog No. A22174
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    anti-psoriatic agent
    Periplogenin is a naturally occurring furanocoumarin found in Angelica dahurica roots, with potent anti-psoriatic effects. Periplogenin induces adipocyte differentiation. 了解更多
  31. Groenlandicine

    Catalog No. A22176
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    protoberberine alkaloid
    Groenlandicine is a protoberberine alkaloid isolated from Coptidis Rhizoma. Groenlandicine exhibits moderate inhibitory effect with IC50 value of 154.2 μM for human recombinant aldose reductase (HRAR). 了解更多
  32. 6-Methoxydihydroavicine

    Catalog No. A22177
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    antiplatelet activities
    6-Methoxydihydroavicine is an alkaloid isolated from Zanthoxylum integrifoliolum. 6-Methoxydihydroavicine has antiplatelet activities and inhibits AA-, collagen- and PAF-induced platelet aggregation in vitro. 了解更多
  33. S-23

    Catalog No. A22178
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    selective androgen receptor modulator
    S-23 is an orally active selective androgen receptor modulator (SARM) with a Ki of 1.7 nM. 了解更多
  34. AC-262536

    Catalog No. A22179
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    selective androgen receptor (SAR) molecule
    AC-262536 is a selective androgen receptor (SAR) molecule. It has partial agonist activity with respect to testosterone and suppresses luteinizing hormone. 了解更多
  35. NSC23005 free acid

    Catalog No. A22180
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    p18INK inhibitor
    NSC23005 is a p18INK inhibitor. NSC23005 potently promotes hematopoietic stem cell (HSC) expansion (ED50 = 5.21 nM). 了解更多
  36. MQAE

    Catalog No. A22181
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    fluorescent indicator
    MQAE is a fluorescent indicator that is quenched via collision with chloride, and is more sensitive and selective than 36Cl and microelectrode-based methods for chloride measurement in cells. 了解更多
  37. ML346

    Catalog No. A22182
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    activator of Hsp70 expression and HSF-1 activity
    ML346 is an activator of Hsp70 expression and HSF-1 activity, with an EC50 of 4.6 μM for Hsp70. 了解更多
  38. ALK2-IN-1

    Catalog No. A22183
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    inhibitor of Activin receptor-like kinase (ALK2) mutant R206H
    ALK2-IN-1 (BLU-782) is a potent and selective inhibitor of Activin receptor-like kinase (ALK2) mutant R206H with binding IC50 of <10 nM. 了解更多
  39. OTSSP167 hydrochloride

    Catalog No. A22184
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    MELK inhibitor
    OTSSP167 (hydrochloride) is a highly potent MELK inhibitor with IC50 value of 0.41 nM. 了解更多
  40. BIO-013077-01

    Catalog No. A22185
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    antagonist of the TGFbeta family type I receptors, Alk5 and/or Alk4
    BIO-013077-01, Novel potent antagonist of the TGFbeta family type I receptors, Alk5 and/or Alk4. 了解更多
  41. Practolol

    Catalog No. A22186
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    β1-adrenergic receptor antagonist
    Practolol is a potent and selective β1-adrenergic receptor antagonist. Practolol can be used for the research of cardiac arrhythmias. 了解更多
  42. Thiambutosine

    Catalog No. A22187
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    candidate for treatment of lepromatous leprosy
    Thiambutosine was a candidate for treatment of lepromatous leprosy. 了解更多
  43. SSD114 hydrochloride

    Catalog No. A22188
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    GABAB receptor positive allosteric modulator
    SSD114 hydrochloride is a novel GABAB receptor positive allosteric modulator. 了解更多
  44. GR 125743

    Catalog No. A22189
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    5-HT1B/1D receptor antagonis
    GR 125743 is a selective 5-HT1B/1D receptor antagonist, with pKis of 8.85 and 8.31 for wild-type h5-HT1B and wild-type h5-HT1D, respectively. 了解更多
  45. Isocyclosporin A

    Catalog No. A22205
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    Isocyclosporin A is a rearranged degradation product formed by acid treatment of cyclosporin A under aqueous and non-aqueous conditions. 了解更多
  46. Levobupivacaine hydrochloride

    Catalog No. A22206
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    sodium channel blocker
    Levobupivacaine hydrochloride is a sodium channel blocker. 了解更多
  47. Apcin-A

    Catalog No. A22207
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    anaphase-promoting complex (APC) inhibitor
    Apcin-A, an Apcin derivative, is an anaphase-promoting complex (APC) inhibitor. 了解更多
  48. ICCB280

    Catalog No. A22208
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    inducer of C/EBPα
    ICCB280 is a potent inducer of C/EBPα. 了解更多
  49. SBP-7455

    Catalog No. A22209
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    dual ULK1/ULK2 autophagy inhibitor
    SBP-7455 is a potent, high affinity and orally active dual ULK1/ULK2 autophagy inhibitor with IC50s of 13 nM and 476 nM in the ADP-Glo assays, respectively. 了解更多
  50. FIDAS-5

    Catalog No. A22210
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    MAT2A inhibitor
    FIDAS-5 is a potent and orally active methionine S-adenosyltransferase 2A (MAT2A) inhibitor with an IC50 of 2.1 μM. 了解更多

产品 401 到 450 共 16088个

每页
页面:
  1. 7
  2. 8
  3. 9
  4. 10
  5. 11

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