Cannabinoid Receptors

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  1. AM630

    Catalog No. A14993
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    CB2 拮抗剂
    AM630是一种选择性CB2拮抗剂,Ki为31.2 nM,选择性是CB1受体的150倍以上。 了解更多
  2. Otenabant

    Catalog No. A15200
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    CB1 receptor 拮抗剂
    Otenabant是最近发现的选择性,高亲和力,竞争性CB1受体拮抗剂,Ki为0.7 nM。 了解更多
  3. AM251

    Catalog No. A12914
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    CB1 receptor 拮抗剂
    AM251是有效的CB1受体拮抗剂(IC50 = 8 nM,Ki = 7.49 nM),其选择性是CB2受体的306倍。 了解更多
  4. CP 945598 HCl (Otenabant HCl)

    Catalog No. A11942
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    CB1 拮抗剂
    CP 945598 HCl (Otenabant HCl)是一种有效且高度选择性的CB1拮抗剂。 了解更多
  5. Taranabant racemate

    Catalog No. A21699
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    CB1 antagonist/inverse agonist
    Taranabant racemate is an antagonist and/or inverse agonist of the Cannabinoid-1 (CB1) receptor extracted from patent WO 2004048317 A1. 了解更多
  6. (±)-Ibipinabant

    Catalog No. A21439
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    CB-1 receptor antagonist
    (±)-Ibipinabant ((±)-SLV319) is the racemate of SLV319. (±)-Ibipinabant ((±)-SLV319) is a potent and selective cannabinoid-1 (CB-1) receptor antagonist with an IC50 of 22 nM. 了解更多
  7. JD-5037

    Catalog No. A20837
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    CB1R antagonist
    JD-5037 is a novel, peripherally restricted CB1R antagonist with an IC50 of 1.5 nM. 了解更多
  8. CB1 antagonist 2

    Catalog No. A18810
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    CB1 antagonist
    CB1 antagonist 2 is caimabinoid 1 (CB1) antagonist extracted from patent WO2016184310A1, compound 3, inhibits CB1 in vivo with an IC50 of 25.5 nM. 了解更多

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