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￥ 0.00 “Ligand-gated Ion Channels”的搜索结果
16 个项目
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ML418
Catalog No. A18426 Kir7.1 potassium channels blockerML418 is a selective, sub-micromolar pore blocker of Kir7.1 potassium channels. The inward rectifier potassium (Kir) channel Kir7.1 (KCNJ13) is a key regulator of melanocortin signaling in the brain, electrolyte homeostasis in the eye, and uterine muscle contractility during pregnancy. 了解更多 -
Vernakalant HCl
Catalog No. A15275 Ion channel blockerVernakalant hydrochloride是一种研究性混合离子通道阻滞剂，可以以2至5 mg/kg的剂量终止人的急性心房纤颤（AF），并且与现有药物相比，对房颤的选择性更高。在抗心律不齐的治疗中。 了解更多 -
Nicardipine hydrochloride
Catalog No. A16634 calcium channel blockerNicardipine hydrochloride (YC-93) is a calcium channel blocker with an IC50 of 1 μM for blocking cardiac calcium channels. 了解更多 -
Mibefradil
Catalog No. A12478 Calcium channel blockerMibefradil is a calcium channel blocker with moderate selectivity for T-type Ca2+ channels displaying IC50s of 2.7 μM and 18.6 μM for T-type and L-type currents, respectively. 了解更多 -
Efonidipine
Catalog No. A17478 Calcium channel blockerEfonidipine is a dihydropyridine calcium channel blocker that blocks both T-type and L-type calcium channels. It has also been studied in atherosclerosis and acute renal failure. 了解更多 -
Ralfinamide mesylate
Catalog No. A22002 Na+ channel blockerRalfinamide mesylate (FCE-26742A mesylate) is an orally available Na+ channel blocker derived from α-aminoamide, with function of suppressing pain. 了解更多 -
Levamlodipine besylate
Catalog No. A21418 Calcium channel blockerLevamlodipine besylate ((S)-Amlodipine besylate) is a powerful dihydropyridine calcium channel blocker, possessing vasodilation properties and used in the treatment of hypertension and angina. 了解更多 -
Dicarbine
Catalog No. A18925 Dopamine receptor blockerDicarbine blocks dopamine receptors in various brain parts and prevents the depression of the conditioned defence reflexes caused by stimulation of the mesencephalic portion of the reticular formation. Dicarbine could be used to treat patients with schizophrenia and alcoholic psychosis in clinical. 了解更多 -
Senicapoc (ICA-17043)
Catalog No. A11568 Gardos channel blockerSenicapoc (ICA-17043) is a potent and selective Gardos channel blocker with IC50 value of 11 nM. It blocks Ca2+-induced rubidium flux from human RBCs with an IC50 value of 11 nM and inhibits RBC dehydration with IC50 of 30 nM. 了解更多 -
Doxazosin
Catalog No. A17779 α-1 adrenergic receptor blockerDoxazosin is an α-1 adrenergic receptor blocker that inhibits the binding of norepinephrine, which is released from sympathetic nerve terminals, to the α-1 receptors on the membrane of vascular smooth muscle cells. Blockages of the alpha-1 adrenergic action on the vascular smooth muscles lead to a decrease in vascular resistance and antihypertensive activity. 了解更多 -
Nicardipine
Catalog No. A17571 Calcium channel blockersNicardipine(YC-93) is a calcium channel blocker that has been widely used to control blood pressure in severe hypertension following events such as ischemic stroke, traumatic brain injury, and intracerebral hemorrhage. 了解更多 -
Imeglimin hydrochloride
Catalog No. A16283 oxidative phosphorylation blockerImeglimin hydrochloride是新型含四氢三嗪的口服降糖药中的第一个，即glimins。已证明它可作用于肝脏，肌肉和胰腺γ-细胞，以独特地靶向2型糖尿病的关键缺陷。 了解更多 -
Gap 27
Catalog No. A14866 -
Gap 26
Catalog No. A14865
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