“leukotriene receptor”的搜索结果
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Ca2+-dependent blocker
TV-519 free base (K201 free base) is a Ca2+-dependent blocker of sarcoplasmic reticulum Ca2+-stimulated ATPase (SERCA) and a partial agonist of ryanodine receptors in striated muscle. Antiarrhythmic and cardioprotective properties.
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NMDA receptors Blocker
Ro 25-6981是N-甲基-D-天冬氨酸(NMDA)受体的高亲和力,强效选择性阻断剂。
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NMDA receptors blocker
RO 25-6981 maleate是含有NR2B亚基的NMDA受体的强效和选择性活性依赖性阻断剂。克隆的受体亚基组合NR1C/NR2B和NR1C/NR2A的IC50值分别为0.009和52 uM。
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D2 receptor blocker
Trimethobenzamide hydrochloride is a blocker of the D2 receptor. Trimethobenzamide is an antiemetic used to prevent nausea and vomiting.
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α-1 adrenergic receptor blocker
Doxazosin is an α-1 adrenergic receptor blocker that inhibits the binding of norepinephrine, which is released from sympathetic nerve terminals, to the α-1 receptors on the membrane of vascular smooth muscle cells. Blockages of the alpha-1 adrenergic action on the vascular smooth muscles lead to a decrease in vascular resistance and antihypertensive activity.
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Dopamine receptor blocker
Dicarbine blocks dopamine receptors in various brain parts and prevents the depression of the conditioned defence reflexes caused by stimulation of the mesencephalic portion of the reticular formation. Dicarbine could be used to treat patients with schizophrenia and alcoholic psychosis in clinical.
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AMPA Receptor Blocker
IEM 1754 Dihydrobromide是AMPA受体的电压依赖性明渠阻断剂。
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Beta-1 adrenergic receptor blocker
Nebivolol是一种选择性抑制β-1肾上腺素能受体,IC50为0.8 nM。
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Beta adrenergic receptor blocker
Pindolol是一种非选择性β阻断剂,具有部分β肾上腺素能受体激动剂活性。
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Beta1 receptor blocker
Metoprolol tartrate是一种选择性β1受体阻滞剂,用于治疗多种心血管系统疾病,尤其是高血压。
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NMDA receptor 拮抗剂
Orphenadrine柠檬酸盐是NMDA受体拮抗剂,Ki为6.0μM,还是HERG钾离子通道阻断剂。
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AT1 Receptor Blocker
Azilsartan (TAK-536)是一种用于治疗高血压的血管紧张素II受体拮抗剂。
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β1 adrenergic receptor blocker
Bisoprolol fumarate是一种属于β受体阻滞剂的药物,β受体阻滞剂是一类主要用于心血管疾病的药物。更具体地说,它是一种选择性的β1肾上腺素能受体阻滞剂。
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