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搜索结果：“receptor”

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JTV-519 free base

Catalog No. A21846
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Ca2+-dependent blocker

TV-519 free base (K201 free base) is a Ca2+-dependent blocker of sarcoplasmic reticulum Ca2+-stimulated ATPase (SERCA) and a partial agonist of ryanodine receptors in striated muscle. Antiarrhythmic and cardioprotective properties. 了解更多

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Ro 25-6981 maleate

Catalog No. A13144
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NMDA receptors Blocker

Ro 25-6981是N-甲基-D-天冬氨酸（NMDA）受体的高亲和力，强效选择性阻断剂。了解更多

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RO 25-6981 maleate

Catalog No. A16083
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NMDA receptors blocker

RO 25-6981 maleate是含有NR2B亚基的NMDA受体的强效和选择性活性依赖性阻断剂。克隆的受体亚基组合NR1C/NR2B和NR1C/NR2A的IC50值分别为0.009和52 uM。了解更多

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Trimethobenzamide hydrochloride

Catalog No. A17648
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D2 receptor blocker

Trimethobenzamide hydrochloride is a blocker of the D2 receptor. Trimethobenzamide is an antiemetic used to prevent nausea and vomiting. 了解更多

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Doxazosin

Catalog No. A17779
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α-1 adrenergic receptor blocker

Doxazosin is an α-1 adrenergic receptor blocker that inhibits the binding of norepinephrine, which is released from sympathetic nerve terminals, to the α-1 receptors on the membrane of vascular smooth muscle cells. Blockages of the alpha-1 adrenergic action on the vascular smooth muscles lead to a decrease in vascular resistance and antihypertensive activity. 了解更多

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Dicarbine

Catalog No. A18925
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Dopamine receptor blocker

Dicarbine blocks dopamine receptors in various brain parts and prevents the depression of the conditioned defence reflexes caused by stimulation of the mesencephalic portion of the reticular formation. Dicarbine could be used to treat patients with schizophrenia and alcoholic psychosis in clinical. 了解更多

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IEM 1754 Dihydrobromide

Catalog No. A14010
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AMPA Receptor Blocker

IEM 1754 Dihydrobromide是AMPA受体的电压依赖性明渠阻断剂。了解更多

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Nebivolol

Catalog No. A13738
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Beta-1 adrenergic receptor blocker

Nebivolol是一种选择性抑制β-1肾上腺素能受体，IC50为0.8 nM。了解更多

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Pindolol

Catalog No. A13422
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Beta adrenergic receptor blocker

Pindolol是一种非选择性β阻断剂，具有部分β肾上腺素能受体激动剂活性。了解更多

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Metoprolol tartrate

Catalog No. A11713
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Beta1 receptor blocker

Metoprolol tartrate是一种选择性β1受体阻滞剂，用于治疗多种心血管系统疾病，尤其是高血压。了解更多

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Orphenadrine citrate

Catalog No. A11712
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NMDA receptor 拮抗剂

Orphenadrine柠檬酸盐是NMDA受体拮抗剂，Ki为6.0μM，还是HERG钾离子通道阻断剂。了解更多

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Azilsartan (TAK-536)

Catalog No. A11775
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AT1 Receptor Blocker

Azilsartan (TAK-536)是一种用于治疗高血压的血管紧张素II受体拮抗剂。了解更多

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Bisoprolol fumarate

Catalog No. A10149
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β1 adrenergic receptor blocker

Bisoprolol fumarate是一种属于β受体阻滞剂的药物，β受体阻滞剂是一类主要用于心血管疾病的药物。更具体地说，它是一种选择性的β1肾上腺素能受体阻滞剂。了解更多

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