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搜索结果：“jwh 250”

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Flavoxate

Catalog No. A12900
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muscarinic AChR antagonist

Flavoxate结合并抑制毒蕈碱受体，从而通过改变脑干的排尿中心来抑制排尿反射并增加膀胱容量。了解更多

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CGS19755

Catalog No. A15791
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NMDA 拮抗剂

CGS 19755（顺式-4-膦酰基甲基-2-哌啶羧酸）是一种有效的立体定向抑制剂，由N-甲基-D-天冬氨酸（NMDA）诱发，但不是由KCl诱发的[3H]乙酰胆碱释放大鼠纹状体的切片。了解更多

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PF-3635659

Catalog No. A13548
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muscarinic M(3) receptor 拮抗剂

PF-3635659是有效的毒蕈碱M3受体拮抗剂。了解更多

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SDZ 220-581

Catalog No. A12426
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NMDA receptor 拮抗剂

SDZ 220-581是一种竞争性NMDA受体拮抗剂（pKi = 7.7）。了解更多

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NF 279

Catalog No. A11972
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P2X1 拮抗剂

NF279是一种苏拉明类似物，可作为P2X受体的高选择性，竞争性和可逆性ATP拮抗剂（平滑肌中IC50/KB1μM）。了解更多

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A 740003

Catalog No. A11316
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P2X7 receptor 拮抗剂

A740003是P2X7受体的新型竞争性拮抗剂（人的IC50值= 40 nM，大鼠的IC50值= 18 nM）。了解更多

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Flumazenil

Catalog No. A10397
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Benzodiazepine 拮抗剂

Flumazenil是竞争性抑制GABA/苯二氮卓受体复合物上苯二氮卓识别位点的活性。Flumazenil在一些活性动物模型中是弱部分激动剂，但在人类中很少或没有激动剂活性。了解更多

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Biperiden HCl

Catalog No. A10147
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Muscarinic receptor antagonist

Biperiden HCl是毒蕈碱受体拮抗剂，对M1亚型表现出一定的选择性。了解更多

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(+)-Bicuculline

Catalog No. A12590
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GABAA 拮抗剂

(+)-Bicuculline是一种经典的GABAA拮抗剂。了解更多

Product Citations (1)

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- Maryam Adenike Salaudeen, .et al. Anticonvulsant Activity of Tapinanthus dodoneifolius (DC.) Danser in Chicks and Mice: A Potential Source of Novel Anticonvulsant Agent, J Pharmacy and Drug Innovations, 2022, 3(4)
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Phenoxybenzamine hydrochloride

Catalog No. A10719
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α-adrenergic (AR) 拮抗剂/CaM 抑制剂

Phenoxybenzamine hydrochloride是一种细胞可渗透的，非特异性的，不可逆的α-肾上腺素（AR）拮抗剂，也可作为CaM抑制剂。了解更多

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Ipratropium bromide

Catalog No. A10476
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Ipratropium bromide是毒蕈碱拮抗剂、支气管扩张剂、阿托品的N-异丙基盐。了解更多

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