“leukotriene receptor”的搜索结果
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NMDA receptor 拮抗剂
Orphenadrine柠檬酸盐是NMDA受体拮抗剂,Ki为6.0μM,还是HERG钾离子通道阻断剂。
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AMPA Receptor 拮抗剂
NBQX是一种有效,选择性和竞争性的AMPA受体拮抗剂。
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NMDA receptor 拮抗剂
DNQX是一种非N-甲基-D-天冬氨酸(非NMDA)受体复合物拮抗剂。
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TRPV1 receptor 拮抗剂
A-889425是选择性TRPV1受体拮抗剂。A-889425阻断TRPV1通道,IC50为335 nM(大鼠)和34 nM(人)。
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AMPA/kainate receptor 拮抗剂
Talampanel是AMPA受体的非竞争性拮抗剂,具有抗癫痫活性。
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TRPV1 receptor 拮抗剂
SB-366791是新颖,有效且选择性的肉桂酰胺TRPV1拮抗剂。
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TRPM8 antagonist
AMG2850 is a potent, orally bioavailable and selective transient receptor potential melastatin 8 (TRPM8) antagonist.
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AMPA receptor antagonist
SYM 2206 is a novel, potent, non-competitive AMPA receptor antagonist.
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CP-AMPA receptors antagonist
Naspm trihydrochloride (1-Naphthylacetyl spermine trihydrochloride), a synthetic analogue of Joro spider toxin, is a calcium permeable AMPA (CP-AMPA) receptors antagonist.
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AMPA (CP-AMPA) receptors antagonist
Naspm (1-Naphthyl acetyl spermine), a synthetic analogue of Joro spider toxin, is a calcium permeable AMPA (CP-AMPA) receptors antagonist.
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L-type calcium antagonist
Barnidipine (Mepirodipine) is an L-type calcium antagonist (CaA) with high affinity for [3H] initrendipine binding sites (Ki=0.21 nmol/l), has selective action against CaA receptors.
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