“Tutalthromycin second gen”的搜索结果

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  1. Nomegestrol acetate

    Catalog No. A21829
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    progesterone receptor agonist
    Nomegestrol acetate is a potent, highly selective progestogen, which is characterized as a full agonist at the progesterone receptor, with no or minimal binding to other steroid receptors, including the androgen and glucocorticoid receptors. 了解更多
  2. DMCM hydrochloride

    Catalog No. A21755
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    Benzodiazepine inverse agonist
    DMCM (hydrochloride) is Benzodiazepine inverse agonist that displays anxiogenic and potent convulsant activity. 了解更多
  3. diABZI STING agonist-1 trihydrochloride

    Catalog No. A21694
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    STING receptor agonist
    diABZI STING agonist-1 (trihydrochloride) is a selective stimulator of interferon genes (STING) receptor agonist, with an EC50s of 130 for human PBMCs. 了解更多
  4. diABZI STING agonist-1

    Catalog No. A21688
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    STING receptor agonist
    diABZI STING agonist-1 is a selective stimulator of interferon genes (STING) receptor agonist, with an EC50s of 130 nM for human PBMCs. 了解更多
  5. RGX-104 free Acid

    Catalog No. A21513
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    LXR agonist
    RGX-104 free Acid is an orally bioavailable and potent liver-X nuclear hormone receptor (LXR) agonist that modulates innate immunity via transcriptional activation of the ApoE gene. 了解更多
  6. Kynurenic acid sodium

    Catalog No. A20000
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    GPR35/CXCR8 agonist
    Kynurenic acid sodium, an endogenous tryptophan metabolite, is a broad-spectrum antagonist targeting NMDA, glutamate, α7 nicotinic acetylcholine receptor. Kynurenic acid sodium is also an agonist of GPR35/CXCR8. 了解更多
  7. Propyl pyrazole triol

    Catalog No. A13329
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    ERα agonist
    Propyl pyrazole triol (PPT) is an estrogen receptor alpha (ERα) agonist. 了解更多
  8. ITE

    Catalog No. A12565
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    AhR agonist
    ITE is a potent endogenous agonist of aryl hydrocarbon receptor (AhR), binding directly to AHR, with a Ki of 3 nM. ITE also has immunosuppressive activity. 了解更多
  9. MK-6913

    Catalog No. A12311
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    Estrogen receptor β agonist
    Tetrahydrofluoroene 52 is a potent and selective estrogen receptor β agonist. 了解更多
  10. PROTAC ERRα ligand 2

    Catalog No. A18939
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    ERRα inverse agonist
    PROTAC ERRα ligand 2 is an estrogen-related receptor α (ERRα) inverse agonist with an IC50 of 5.67 nM. PROTAC ERRα ligand 2 (IC50=5.67 nM) displays a ~11-fold improved potency than XCT790 (IC50=61.3 nM). 了解更多
  11. STING agonist-4

    Catalog No. A19074
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    STING receptor agonist
    STING agonist-4 is an stimulator of Interferon Genes (STING) receptor agonist with an apparent inhibitory constant (IC50) of 20 nM. 了解更多
  12. GSK5182

    Catalog No. A19383
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    ERRγ agonist
    GSK5182 is a highly selective inverse agonist of estrogen-related receptor γ (ERRγ) with an IC50 of 79 nM and does not interact with other nuclear receptors, including ERRα or ERα. 了解更多
  13. Kynurenic acid

    Catalog No. A16581
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    GPR35/CXCR8 拮抗剂
    Kynurenic acid, an endogenous tryptophan metabolite, is a broad-spectrum antagonist targeting NMDA, glutamate, α7 nicotinic acetylcholine receptor. Kynurenic acid is also an agonist of GPR35/CXCR8. 了解更多
  14. KAG-308

    Catalog No. A18389
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    EP4 激动剂
    KAG-308, a newly-identified EP4-selective agonist shows efficacy for treating ulcerative colitis and can bring about lower risk of colorectal carcinogenesis by oral administration. 了解更多
  15. Beclometasone

    Catalog No. A18177
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    glucocorticoid receptor agonist
    Beclometasone, also known as Beclomethasone, is an anti-inflammatory, synthetic glucocorticoid. It is used topically as an anti-inflammatory agent and in aerosol form for the treatment of asthma. 了解更多
  16. Nylidrin Hydrochloride

    Catalog No. A17947
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    beta-adrenergic agonist
    Nylidrin hydrochloride is a beta-adrenergic agonist. Nylidrin hydrochloride is shown to be an effective inhibitor of IgE-mediated release of histamine from human basophils, and thus can be used as antiallergic agent. 了解更多
  17. Midodrine

    Catalog No. A17758
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    adrenergic alpha-1 agonist
    Midodrine is an ethanolamine derivative that is an adrenergic alpha-1 agonist. It is used as a vasoconstrictor agent in the treatment of HYPOTENSION. 了解更多
  18. Midodrine hydrochloride

    Catalog No. A17757
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    Adrenergic alpha-1 agonist
    Midodrine hydrochloride is an ethanolamine derivative that is an adrenergic alpha-1 agonist. It is used as a vasoconstrictor agent in the treatment of hypotension. It improves clinical outcome of chronic hypotension. 了解更多
  19. Canrenone

    Catalog No. A17574
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    Na/K ATPase partial agonist
    Canrenone is a metabolite of spironolactone, Na/K ATPase partial agonist and aldosterone and androgen receptor antagonist used as a diuretic. 了解更多
  20. GW-870086

    Catalog No. A18343
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    Glucocorticoid receptor agonist
    GW-870086 is a potent anti-inflammatory agent, acting as a glucocorticoid receptor agonist, with a pIC50 of 10.1 in A549 cells expressing NF-κB. 了解更多
  21. (R)-Equol

    Catalog No. A16986
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    Estrogen receptor 激动剂
    (R)-Equol是ER&alpha和ER&beta的激动剂,Kis分别为27.4和15.4 nM。 了解更多
  22. Galanin (1-30) (human)

    Catalog No. A16890
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    Endogenous galanin receptor 激动剂
    Galanin (1-30) (human)是具有多种内分泌,代谢和行为作用的内源肽。 了解更多
  23. Andarine (GTX-007)

    Catalog No. A10076
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    Androgen Receptor 激动剂
    Andarine (GTX-007)是研究性的选择性雄激素受体调节剂(SARM)。 了解更多
  24. Hexestrol

    Catalog No. A10451
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    Estrogen/progestogen Receptor 激动剂
    Hexestrol是一种致癌的合成雌激素,可抑制微管聚合和带状结构的形成。它是脂质过氧化的抑制剂。 了解更多

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