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  1. GDC-0834 Racemate

    Catalog No. A12706
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    BTK 抑制剂
    GDC-0834 Racemate是一种有效且选择性的Bruton酪氨酸激酶(BTK)抑制剂,被研究用作类风湿关节炎的潜在治疗剂。 了解更多
  2. Vandetanib trifluoroacetate

    Catalog No. A15272
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    VEGFR/EGFR 抑制剂
    Vandetanib trifluoroacetate是一种有效的VEGFR2抑制剂,IC50为40 nM。 了解更多
  3. Pyrotinib Racemate

    Catalog No. A17068
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    EGFR/HER2 dual 抑制剂
    Pyrotinib Racemate是吡罗替尼的外消旋体。吡罗替尼是一种有效的选择性EGFR/HER2双重抑制剂。 了解更多
  4. Ibrutinib Racemate

    Catalog No. A18022
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    Btk inhibitor
    Ibrutinib Racemate (PCI-32765 Racemate) is the racemate of Ibrutinib. Ibrutinib is a selective, irreversible Btk inhibitor with IC50 value of 0.5 nM. 了解更多
  5. (Rac)-PT2399

    Catalog No. A21376
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    HIF-2α inhibitor
    (Rac)-PT2399 (Compound 10e), the racemate of PT2399, acts as a potent and specific hypoxia-inducible factor 2a (HIF-2α) inhibitor with an IC50 of 0.01 μM. 了解更多

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