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搜索结果：“jwh 018”

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CP-640186 hydrochloride

Catalog No. A21808
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ACC inhibitor

CP-640186 hydrochloride is a potent and cell-permeable Acetyl-CoA carboxylase (ACC) inhibitor with IC50s of 53 nM and 61 nM for rat liver ACC1 and rat skeletal muscle ACC2 respectively. 了解更多

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CVT-12012

Catalog No. A21447
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SCD inhibitor

CVT-12012 is a potent and orally bioavailable stearoyl-coA desaturase (SCD) inhibitor, with IC50s of 38 nM, 6.1 nM for rat microsomal and human HEPG2, respectively. 了解更多

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IDO-IN-3

Catalog No. A20898
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IDO inhibitor

IDO-IN-3 is a potent indoleamine 2,3-dioxygenase (IDO) inhibitor with an IC50 of 290 nM. 了解更多

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TPN171

Catalog No. A18464
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PDE5 inhibitor

TPN171 is potent PDE5 inhibitor with subnanomolar potency for PDE5 and good selectivity over PDE6. 了解更多

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4-Chloro-DL-phenylalanine

Catalog No. A16424
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Tryptophan hydroxylase 抑制剂

4-Chloro-DL-phenylalanine是色氨酸羟化酶的选择性和不可逆抑制剂，色氨酸羟化酶是5-羟色胺（5-羟色胺）生物合成中的限速酶。了解更多

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CGP 3466B maleate

Catalog No. A12385
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GAPDH 抑制剂

CGP 3466B maleate是口服活性甘油醛-3-磷酸脱氢酶(gapdh)抑制剂。了解更多

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JZL184

Catalog No. A12747
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MAGL 抑制剂

JZL184是一种有效的选择性单酰基甘油脂肪酶（MAGL）抑制剂。体内阻断内源性大麻素2-花生四烯酸甘油酯（2-AG）的水解（IC50 = 8 nM）。了解更多

Product Citations (4)

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- Lakhan S Khara, .et al. Inhibiting the endocannabinoid degrading enzymes FAAH and MAGL during zebrafish embryogenesis alters sensorimotor function, J Exp Biol, 2022, May 1;225(9):jeb244146 PMID: 35438163
- Md Shah Sufian, .et al. Early suppression of the endocannabinoid degrading enzymes FAAH and MAGL alters locomotor development in zebrafish, J Exp Biol, 2021, 21 JUNE
- Toshihiko Tsutsumi, .et al. Identification of human glycerophosphodiesterase 3 as an ecto phospholipase C that converts the G protein-coupled receptor 55 agonist lysophosphatidylinositol to bioactive monoacylglycerols in cultured mammalian cells, Biochim Biophys Acta Mol Cell Biol Lipids, 2020, Sep;1865(9):158761 PMID: 32629025
- Rea Pihlaja, .et al. The Anti-Inflammatory Effects of Lipoxygenase and Cyclo-Oxygenase Inhibitors in Inflammation-Induced Human Fetal Glia Cells and the Aβ Degradation Capacity of Human Fetal Astrocytes in an Ex vivo Assay, Front Neurosci, 2017, 11: 299 PMID: 28611577
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Carbidopa

Catalog No. A10181
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aromatic-L-amino-acid decarboxylase 抑制剂

Carbidopa是一种芳香族-L-氨基酸脱羧酶抑制剂，这是一种在L-色氨酸生物合成5-羟色胺和L-DOPA生物合成多巴胺（DA）中重要的酶。了解更多

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