“AZ 960”的搜索结果

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  1. Sancycline

    Catalog No. A13393
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    Sancycline像其他四环素类药物一样,三环素通过可逆地结合到30S核糖体亚单位并通过阻断氨酰tRNA进入核糖体A位点来抑制蛋白质翻译。 了解更多
  2. HCV-IN-3

    Catalog No. A20957
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    HCV NS3/4a protein inhibitor
    HCV-IN-3 is a hepatitis C virus (HCV) NS3/4a protein inhibitor, with an IC50 of 20 μM, a Kd of 29 μM. 了解更多
  3. Loviride

    Catalog No. A21996
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    non-nucleoside reverse transcriptase inhibitor
    Loviride (R 89439) is a non-nucleoside reverse transcriptase inhibitor (NNRTI), with an IC50 of 0.3 ?M for reverse transcriptase from HIV-1. Loviride (R 89439) inhibits HIV-1, HIV-2 and SIV replication in MT-4 cells. 了解更多
  4. PSI-6206 13CD3

    Catalog No. A21782
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    HCV NS5B polymerase inhibitor
    PSI-6206 13CD3 is the deuterium labeled PSI-6206. PSI-6206 is the deaminated derivative of PSI-6130, which is a potent and selective inhibitor of HCV NS5B polymerase. 了解更多
  5. Tenofovir maleate

    Catalog No. A21776
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    nucleotide reverse transcriptase inhibitor
    Tenofovir Disoproxil Fumarate is a nucleotide reverse transcriptase inhibitor to treat HIV and chronic Hepatitis B. 了解更多
  6. Delavirdine

    Catalog No. A21469
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    non-nucleoside reverse transcriptase inhibitor
    Delavirdine(U 90152) is a potent non-nucleoside reverse transcriptase inhibitor (NNRTI). 了解更多
  7. R-1479

    Catalog No. A11540
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    HCV replication inhibitor
    R-1479 is a specific inhibitor of HCV replication in the HCV subgenomic replicon system (IC50=1.28 μM). 了解更多
  8. Mericitabine

    Catalog No. A11539
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    HCV NS5B polymerase inhibitor
    Mericitabine (RG 7128; R-7128) is a nucleoside inhibitor of the HCV NS5B polymerase that acts as an RNA chain terminator and prevents elongation of RNA transcripts during replication. 了解更多
  9. MIV-150

    Catalog No. A12060
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    NNRT inhibitor
    MIV-150 is a nonnucleoside reverse transcriptase (NNRT) inhibitor, blocking HIV-1 and HIV-2 infections, with an EC50<1 nM against HIV-1/HIV-2MN. 了解更多
  10. Voxilaprevir

    Catalog No. A12067
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    HCV NS 3/4A protease inhibitor
    Voxilaprevir (GS-9857) is a fluorinated macrocyclic hepatitis C virus (HCV) nonstructural protein (NS) 3/4A protease inhibitor with potent in vitro antiviral activity against genotypes 1-6 HCV and broad coverage of NS3/4A protease polymorphisms. GS-9857 improves coverage against commonly encountered NS3 resistance-associated variants (RAVs). 了解更多
  11. CCR4 antagonist 2

    Catalog No. A18471
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    CCR4 拮抗剂
    CCR4 antagonist 2 (Compound 31) is a novel potent, orally bioavailable small molecule antagonists of CC chemokine receptor 4 (CCR4) that inhibits Treg trafficking into the Tumor Microenvironment without suppressing the number of Treg in healthy tissues. 了解更多
  12. AZ084

    Catalog No. A19143
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    CCR8 拮抗剂
    AZ084 is a potent, selective, allosteric and oral active CCR8 antagonist, with a Ki of 0.9 nM. Has potential to treat asthma. 了解更多
  13. Cyromazine

    Catalog No. A16473
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    Cyromazine是一种三嗪昆虫生长调节剂,用作杀虫剂和杀螨剂。 了解更多
  14. Climbazole

    Catalog No. A16457
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    Climbazole是广谱咪唑类抗真菌剂,可提供去头皮屑的功效。 了解更多
  15. Cefazolin Sodium

    Catalog No. A16434
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    Cefazolin Sodium是一种半合成的头孢菌素类似物,由于抑制细菌细胞壁的合成而具有广谱抗生素作用。它具有很高的血清水平,可通过尿液迅速排泄。 了解更多
  16. Azlocillin sodium salt

    Catalog No. A16422
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    Azlocillin sodium salt是一种具有广泛抗细菌作用的氨苄青霉素。 了解更多
  17. Azithromycin Dihydrate

    Catalog No. A16421
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    Azithromycin Dihydrate是一种酸稳定的口服大环内酯类抗菌药物,在结构上与红霉素有关。 了解更多
  18. Aminothiazole

    Catalog No. A16403
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    Thyroid 抑制剂
    Aminothiazole可用作甲状腺抑制剂,并具有抗菌活性。 了解更多
  19. Bacitracin

    Catalog No. A10960
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    Bacitracin是枯草芽孢杆菌var Tracy的地衣形生物产生的相关环状多肽的混合物,其通过干扰细胞壁和肽聚糖的合成破坏革兰氏阳性和革兰氏阴性细菌。 了解更多
  20. Sodium sulfadiazine

    Catalog No. A16160
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    Sodium sulfadiazine是磺胺嘧啶的钠盐形式,磺胺嘧啶是一种具有中间作用的抑菌合成磺胺衍生物。 了解更多
  21. Furazolidone

    Catalog No. A16011
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    Furazolidone是合成的硝基呋喃衍生物,当用于对抗革兰氏阳性和革兰氏阴性细菌时具有杀菌或抑菌活性。 了解更多
  22. Zidovudine

    Catalog No. A15428
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    NRTI 抑制剂
    Zidovudine是一种核苷类似物逆转录酶抑制剂(NRTI),是一种用于治疗HIV/AIDS感染的抗逆转录病毒药物。叠氮胸苷降低了CRISPR介导的同源性定向修复(HDR)的效率。 了解更多
  23. Isoconazole nitrate

    Catalog No. A10481
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    Isoconazole nitrate (Travogen)是一种唑类抗真菌剂。 了解更多
  24. Aztreonam (Azactam, Cayston)

    Catalog No. A10118
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    Aztreonam (Azactam,Cayston)是一种合成的单环β-内酰胺抗生素 (一种单bactam),其细胞核是基于一种从紫罗兰色杆菌中分离出来的更简单的单bactam。 了解更多
  25. Atazanavir

    Catalog No. A10097
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    HIV Protease 抑制剂
    Atazanavir是一种氮杂肽及HIV-蛋白酶抑制剂,常与其他抗HIV药物结合,用于治疗HIV感染以及获得性免疫缺乏综合征。 了解更多
  26. Atazanavir sulfate (BMS-232632-05)

    Catalog No. A10096
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    HIV Protease 抑制剂
    Atazanavir sulfate (BMS-232632-05)是蛋白酶抑制剂(PI)类的抗逆转录病毒药物。是一种高选择性的 HIV-1蛋白酶抑制剂。 了解更多
  27. BMS-707035

    Catalog No. A10156
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    HIV-1 integrase 抑制剂
    BMS-707035是HIV-1整合酶(IN)抑制剂。HIV-1整合酶(IN)代表临床上治疗HIV/AIDS的具有治疗优势的病毒靶标。 了解更多

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