“AZ 960”的搜索结果

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  1. Dienogest

    Catalog No. A10308
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    Dienogest是一种口服抗孕激素,具有抗雄激素活性,因此可以改善雄激素症状。 了解更多
  2. Benazepril HCl

    Catalog No. A10123
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    RAAS 抑制剂
    Benazepril hydrochloride是一种非肽血管紧张素转化酶(ACE)抑制剂。降低自发性高血压大鼠的血压和心肌肥大。 了解更多
  3. Bazedoxifene acetate

    Catalog No. A11665
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    Bazedoxifene Acetate是第三代选择性雌激素受体调节剂(SERM)。 了解更多
  4. Azilsartan (TAK-536)

    Catalog No. A11775
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    AT1 Receptor Blocker
    Azilsartan (TAK-536)是一种用于治疗高血压的血管紧张素II受体拮抗剂。 了解更多
  5. 17 alpha-propionate

    Catalog No. A10009
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    Androgen 拮抗剂
    17 alpha-propionate是一种新型的局部和外周选择性雄激素拮抗剂。 了解更多
  6. Cilazapril monohydrate

    Catalog No. A11747
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    ACE 抑制剂
    Cilazapril monohydrate是哒嗪血管紧张素转换酶抑制剂(ACE抑制剂),用于治疗高血压和充血性心力衰竭。 了解更多
  7. Deflazacort

    Catalog No. A10294
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    Deflazacort是一种糖皮质激素,用作抗炎和免疫抑制剂。 了解更多
  8. AZD3514

    Catalog No. A12396
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    AR 抑制剂 downregulator
    AZD3514是一种有效的雄激素受体下调剂,具有潜在的抗癌活性。 了解更多
  9. AZD5423

    Catalog No. A13249
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    nonsteroidal glucocorticoid receptor 激动剂
    AZD5423是新型的非甾体类糖皮质激素受体激动剂。 了解更多
  10. (Glp1)-Apelin-13

    Catalog No. A13215
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    Apelin Receptor activator
    (Glp1)-Apelin-13是Apelin受体的激活剂。 了解更多
  11. AZD1981

    Catalog No. A13186
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    CRTH2 receptor 拮抗剂
    AZD1981作为疾病相关细胞系统的有效拮抗剂,可抑制DK-PGD2诱导的人嗜酸性粒细胞CD11b表达,IC50为10 nM。 了解更多
  12. Bazedoxifene

    Catalog No. A15019
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    Estrogen modulator
    Bazedoxifene是雌激素受体的第三代选择性调节剂。 了解更多
  13. AZD9496

    Catalog No. A15822
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    estrogen receptor downregulator and 拮抗剂
    AZD9496是一种有效的生物选择性雌激素受体下调剂和拮抗剂。 了解更多
  14. Desogestrel

    Catalog No. A16173
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    Desogestrel是一种合成的孕激素,通常用作联合口服避孕药的孕激素成分。 了解更多
  15. Azilsartan Medoxomil

    Catalog No. A16420
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    angiotensin II receptor type 1 拮抗剂
    Azilsartan medoxomil是一种口服给药的1型血管紧张素II受体拮抗剂,IC50为0.62 nM。 了解更多
  16. AZD9567

    Catalog No. A18850
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    selective glucocorticoid receptor modulator
    AZD9567 is a potent, oral active, non-steroidal and selective glucocorticoid receptor modulator (SGRM), with an IC50 of 3.8 nM. 了解更多
  17. AZD-0284

    Catalog No. A18766
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    RORγ 激动剂
    AZD-0284 is a potent, selective, inverse agonist of the nuclear receptor RORγ for the potential treatment of Plaque psoriasis. 了解更多
  18. AZD2906

    Catalog No. A18936
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    glucocorticoid receptor agonist
    AZD2906 is a selective glucocorticoid receptor (GR) agonist, increases micronucleated immature erythrocytes in the bone marrow of rats. AZD2906 shows IC50s of 2.2, 0.3, 41.6 and 7.5 nM at GR in human, rat PBMC and human, rat whole blood, respectively. 了解更多
  19. PROTAC ERRα Degrader-1

    Catalog No. A18910
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    ERRα Degrader
    PROTAC ERRα Degrader-1 comprises a MDM2 ligand binding group, a linker and an estrogen-related receptor alpha (ERRa) binding group. PROTAC ERRα Degrader-1 is an estrogen-related receptor alpha (ERRa) degrader. 了解更多
  20. Betamethasone acibutate

    Catalog No. A18697
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    glucocorticoid
    Betamethasone acibutate, derives from Betamethasone, is an acetate ester. Betamethasone acibutate is a glucocorticoid. 了解更多
  21. ROR agonist-1

    Catalog No. A18569
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    ROR 激动剂
    ROR agonist-1 is a potent and orally bioavailable inverse agonist of the retinoic acid receptor-related orphan receptor C2 (RORC2), inhibition of IL-17A production from human primary TH 17 cells with a pIC50 of 7.5. 了解更多
  22. Glucocorticoid receptor agonist

    Catalog No. A11431
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    Glucocorticoid receptor agonist
    Glucocorticoid receptor agonist is a potent Glucocorticoid receptor agonist. 了解更多
  23. Imidaprilate

    Catalog No. A20003
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    ACE inhibitor
    Imidaprilate is an active metabolite of TA-6366, acts as a potent angiotensin converting enzyme (ACE) inhibitor, with an IC50 of 2.6 nM, and is used in the research of hypertensive disease. 了解更多
  24. Azilsartan medoxomil monopotassium

    Catalog No. A20860
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    angiotensin II receptor type 1 antagonist
    Azilsartan medoxomil monopotassium is an orally administered angiotensin II receptor type 1 antagonist with IC50 of 0.62 nM, which used in the treatment of adults with essential hypertension. 了解更多
  25. Fosdagrocorat

    Catalog No. A21303
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    dissociated glucocorticoid receptor agonist
    Fosdagrocorat (PF-04171327) is a dissociated glucocorticoid receptor agonist. 了解更多
  26. Dagrocorat

    Catalog No. A21312
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    glucocorticoid receptor agonist
    Dagrocorat (PF-00251802) is a novel and dissociated glucocorticoid receptor agonist. 了解更多
  27. Losartan (D4 Carboxylic Acid)

    Catalog No. A21578
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    angiotensin II receptor antagonist
    Losartan D4 Carboxylic Acid is the deuterium labeled Losartan(EXP-3174), which is an angiotensin II receptor antagonist. 了解更多
  28. Azilsartan D5

    Catalog No. A21600
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    angiotensin II type 1 receptor antagonist
    Azilsartan D5 is the deuterium labeled Azilsartan(TAK-536), which is a specific and potent angiotensin II type 1 receptor antagonist. 了解更多
  29. Pipendoxifene hydrochloride

    Catalog No. A21623
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    estrogen receptor modulators
    Pipendoxifene hydrochloride is a selective estrogen receptor modulators (SERMs). 了解更多
  30. H3B-6545 Hydrochloride

    Catalog No. A21629
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    estrogen receptor covalent antagonist
    H3B-6545 Hydrochloride is an oral, selective estrogen receptor covalent antagonist (SERCA). 了解更多
  31. AZD9496 maleate

    Catalog No. A21726
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    estrogen receptor (ERα) antagonist
    AZD9496 maleate is a potent and selective estrogen receptor (ERα) antagonist with IC50 of 0.28 nM. AZD9496 maleate is an orally bioavailable selective oestrogen receptor degrader (SERD). 了解更多

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