“azd”的搜索结果

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  1. AZD-0284

    Catalog No. A18766
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    RORγ 激动剂
    AZD-0284 is a potent, selective, inverse agonist of the nuclear receptor RORγ for the potential treatment of Plaque psoriasis. 了解更多
  2. AZD9496 maleate

    Catalog No. A21726
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    estrogen receptor (ERα) antagonist
    AZD9496 maleate is a potent and selective estrogen receptor (ERα) antagonist with IC50 of 0.28 nM. AZD9496 maleate is an orally bioavailable selective oestrogen receptor degrader (SERD). 了解更多
  3. AZD2906

    Catalog No. A18936
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    glucocorticoid receptor agonist
    AZD2906 is a selective glucocorticoid receptor (GR) agonist, increases micronucleated immature erythrocytes in the bone marrow of rats. AZD2906 shows IC50s of 2.2, 0.3, 41.6 and 7.5 nM at GR in human, rat PBMC and human, rat whole blood, respectively. 了解更多
  4. AZD9567

    Catalog No. A18850
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    selective glucocorticoid receptor modulator
    AZD9567 is a potent, oral active, non-steroidal and selective glucocorticoid receptor modulator (SGRM), with an IC50 of 3.8 nM. 了解更多
  5. AZD9496

    Catalog No. A15822
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    estrogen receptor downregulator and 拮抗剂
    AZD9496是一种有效的生物选择性雌激素受体下调剂和拮抗剂。 了解更多
  6. AZD1981

    Catalog No. A13186
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    CRTH2 receptor 拮抗剂
    AZD1981作为疾病相关细胞系统的有效拮抗剂,可抑制DK-PGD2诱导的人嗜酸性粒细胞CD11b表达,IC50为10 nM。 了解更多
  7. AZD5423

    Catalog No. A13249
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    nonsteroidal glucocorticoid receptor 激动剂
    AZD5423是新型的非甾体类糖皮质激素受体激动剂。 了解更多
  8. AZD3514

    Catalog No. A12396
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    AR 抑制剂 downregulator
    AZD3514是一种有效的雄激素受体下调剂,具有潜在的抗癌活性。 了解更多

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