“MK-2206 dihydrochloride”的搜索结果

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  1. MW-150 dihydrochloride dihydrate

    Catalog No. A21860
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    p38α MAPK inhibitor
    MW-150 dihydrochloride dihydrate (MW01-18-150SRM dihydrochloride dihydrate) is a selective, CNS penetrant, and orally active inhibitor of p38α MAPK with a Ki of 101 nM. 了解更多
  2. B-Raf inhibitor 1 dihydrochloride

    Catalog No. A21834
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    Raf kinase inhibitor
    B-Raf inhibitor 1 dihydrochloride is a potent Raf kinase inhibitor with Kis of 1 nM, 1 nM, and 0.3 nM for B-RafWT, B-RafV600E, and C-Raf, respectively. 了解更多
  3. ML 786 dihydrochloride

    Catalog No. A11211
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    Raf 抑制剂
    ML 786 dihydrochloride是一种有效的Raf激酶抑制剂(B-RafV600E,C-Raf和野生型B-Raf的IC50值分别为2.1、2.5和4.2 nM)。 了解更多
  4. SKF 86002 Dihydrochloride

    Catalog No. A11101
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    p38 MAPK 抑制剂
    SKF 86002 Dihydrochloride是p38 MAP激酶的抑制剂(IC50 = 0.1-1 uM)。有效抑制人单核细胞中LPS诱导的IL-1和TNF-α的产生(IC50 = 1 uM)。 了解更多
  5. DBM 1285 dihydrochloride

    Catalog No. A16058
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    p38 MAPK 抑制剂
    DBM 1285 dihydrochloride是p38 MAPK抑制剂。在巨噬细胞和体内抑制p38磷酸化和LPS诱导的TNF-α产生。 了解更多

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