“Tutalthromycin second gen”的搜索结果

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  1. Veledimex

    Catalog No. A21011
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    CYP3A4/5 inhibitor and substrate
    Veledimex is an oral activator ligand for a proprietary gene therapy promoter system, and a moderate inhibitor of and substrate for CYP3A4/5. 了解更多
  2. Seviteronel

    Catalog No. A20996
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    CYP17 lyase inhibitor
    Seviteronel (VT-464) is a potent CYP17 lyase inhibitor(h-Lyase IC50=69 nM) that demonstrated both exceptional in vitro lyase/hydroxylase selectivity (~10-fold) and oral activity in a hamster model of androgen biosynthesis inhibition. 了解更多
  3. Liarozole dihydrochloride

    Catalog No. A21853
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    CYP450 dependent inhibitor
    Liarozole dihydrochloride (R75251; R85246) is a cytochrome P450 (CYP450) dependent inhibitor, orally active, it also a potent inhibitor of estrogen (via inhibition of aromatase) and testicular androgen synthesis (inhibition of 17 ,20-lyase). 了解更多
  4. Sulfaphenazole

    Catalog No. A17283
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    CYP2C9 inhibitor
    Sulfaphenazole is a specific inhibitor of CYP2C9 which blocks atherogenic and pro-inflammatory effects of linoleic acid (increase in oxidative stress and activation of AP-1) mediated by CYP2C9. 了解更多
  5. TAK-700 Salt (Orteronel Salt)

    Catalog No. A13515
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    CYP17A1/androgen synthesis 抑制剂
    TAK-700 Salt (Orteronel Salt)是一种雄激素合成抑制剂。它选择性地抑制在睾丸,肾上腺和前列腺肿瘤组织中表达的酶CYP17A。 了解更多
  6. Baicalein

    Catalog No. A10120
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    Lipoxygenase 抑制剂
    Baicalein是一种类黄酮,最初从黄cut的根中分离出来。Baicalein抑制脂质过氧化 (通过TBARS的产生评估),IC50值为5 ?M。 了解更多
  7. Apigenin

    Catalog No. A10081
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    Protein kinase 抑制剂
    Apigenin是中央苯并二氮杂central受体的配体,其Ki为4μM竞争性抑制氟硝西epa的结合,发挥抗焦虑和轻微的镇静作用。 了解更多
  8. Cyproterone acetate

    Catalog No. A11409
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    Androgen Receptor 拮抗剂
    Cyproterone acetate是17-羟孕酮的合成衍生物,可作为雄激素受体拮抗剂以及具有弱孕激素和糖皮质激素活性的弱孕激素受体激动剂。 了解更多
  9. Naringenin

    Catalog No. A10625
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    Naringenin是一种黄烷酮,是一种类黄酮,被认为具有抗氧化剂,自由基清除剂,消炎,碳水化合物代谢促进剂和免疫系统调节剂等对人体健康的生物活性。 了解更多

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