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搜索结果：“betaine hydrochloride”

“betaine hydrochloride”的搜索结果

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AR-M 1000390 hydrochloride

Catalog No. A21911
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δ opioid receptor agonist

AR-M 1000390 hydrochloride is an exceptionally selective, potent δ opioid receptor agonist with an EC50 of 7.2??0.9 nM for δ agonist potency. 了解更多

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GSK1521498 free base (hydrochloride)

Catalog No. A21792
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μ-opioid receptor (MOR) antagonist

GSK1521498 free base (hydrochloride) is a potent and selective μ-opioid receptor (MOR) antagonist. 了解更多

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CYT-1010 hydrochloride

Catalog No. A21348
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mu-opioid receptor agonist

CYT-1010 hydrochloride is a mu-opioid receptor agonist extracted from patent WO2013173730A2, with EC50s of 13.1 nM and 0.0053 nM on beta-arrestin recruitment and inhibition of cAMP production, respectively. 了解更多

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Nalmefene hydrochloride

Catalog No. A13843
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dopamine receptor 激动剂

Nalmefene hydrochloride是opioid receptor拮抗剂。了解更多

Product Citations (1)

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- Mark G Papich, .et al. Naloxone and nalmefene absorption delivered by hollow microneedles compared to intramuscular injection, Drug Deliv Transl Res, 2022, Feb;12(2):376-383 PMID: 34817831
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Nalfurafine hydrochloride

Catalog No. A12579
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opioid κ-selective 激动剂

Nalfurafine hydrochloride是一种κ-opioid激动剂。了解更多

Product Citations (6)

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- Alexander R French, .et al. Sex- and β-arrestin-dependent effects of kappa opioid receptor-mediated ethanol consumption, Pharmacol Biochem Behav, 2022, May;216:173377 PMID: 35364122
- Wen-Wen Zhang, .et al. Peripheral ablation of type III adenylyl cyclase induces hyperalgesia and eliminates KOR-mediated analgesia in mice, JCI Insight, 2022, Feb 8;7(3):e153191 PMID: 34914639
- A Dunn, .et al. Modulation of Cocaine-Related Behaviors by Low Doses of the Potent KOR Agonist Nalfurafine in Male C57BL6 Mice, Psychopharmacology (Berl), 2020, May 20 PMID: 32435819
- Dunn AD, .et al. Signaling Properties of Structurally Diverse Kappa Opioid Receptor Ligands: Toward in Vitro Models of in Vivo Responses, ACS Chem Neurosci, 2019, Aug 21;10(8):3590-3600 PMID: 31313902
- Anika Mann, .et al. Agonist-selective NOP receptor phosphorylation correlates in vitro and in vivo and reveals differential post-activation signaling by chemically diverse agonists, Sci Signal, 2019, Mar 26;12(574). pii: eaau8072 PMID: 30914485
- Snyder LM, .et al. Kappa Opioid Receptor Distribution and Function in Primary Afferents, Neuron, 2018, Sep 19;99(6):1274-1288.e6 PMID: 30236284
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MCOPPB 3HCl

Catalog No. A10561
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NOP receptor 激动剂

MCOPPB 3HCl是一种用作伤害感受器受体的有效和选择性激动剂的化合物，pKi为10.07。了解更多

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BRL 52537 HCl

Catalog No. A11210
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Opioid Receptors 激动剂

BRL 52537 hydrochloride是一种高度选择性和有效的κ阿片类激动剂（Ki = 0.24 nM）。比吗啡强25倍。了解更多

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