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Nomegestrol
Catalog No. A19235 full progesterone receptor agonistNomegestrol is a potent and orally available progestin, acts as a selective full progesterone receptor agonist, with a Kd of 5.44 nM for rat uterine progesterone receptor, and has moderate antiandrogenic activity and strong antiestrogenic activity. 了解更多 -
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N-[(4-Aminophenyl)methyl]adenosine
Catalog No. A12659 Adenosine receptor inhibitorN-[(4-Aminophenyl)methyl]adenosine is a adenosine receptor inhibitor, with Ki of 29 nM for Rat ecto-5??-Nucleotidase. IC50 value: 29.0 ± 1.7 nM (Ki) Target: Adenosine Receptor 了解更多 -
Cariprazine
Catalog No. A21202 D3 receptor and D2 receptor partial agonistCariprazine is a novel antipsychotic drug candidate that exhibits high affinity for the D3 (Ki=0.085 nM) and D2 (Ki=0.49 nM) receptors, and moderate affinity for the 5-HT1A receptor (Ki=2.6 nM). 了解更多 -
Dihydrexidine
Catalog No. A21949 D1-like dopamine receptor (D1/D5) agonistDihydrexidine (DAR-0100) is a high potent, selective and full efficacy D1-like dopamine receptor (D1/D5) agonist with an IC50 of 10 nM for D1 receptor. Dihydrexidine exhibits potent antiparkinsonian activity. 了解更多 -
AZD9496 maleate
Catalog No. A21726 estrogen receptor (ERα) antagonistAZD9496 maleate is a potent and selective estrogen receptor (ERα) antagonist with IC50 of 0.28 nM. AZD9496 maleate is an orally bioavailable selective oestrogen receptor degrader (SERD). 了解更多 -
Tarafenacin D-tartrate
Catalog No. A21477 M3 muscarinic receptor antagonistTarafenacin D-tartrate (SVT-40776 D-tartrate) is a highly selective M3 muscarinic receptor antagonist (Ki= 0.19 nM), ~200 fold selectivity over M2 receptor. 了解更多 -
JNJ-37822681 dihydrochloride
Catalog No. A21470 dopamine D2 receptor antagonistJNJ-37822681 dihydrochloride is a potent, specific, centrally active, fast-dissociating dopamine D2 receptor antagonist with a moderate binding affinity for the dopamine D2L receptor (Ki =158 nM), which has potential for the treatment of schizophrenia and bipolar disorder. 了解更多 -
Risperidone mesylate
Catalog No. A21463 dopamine D2 receptor antagonistRisperidone mesylate(R 64 766 mesylate) is a serotonin 5-HT2 receptor blocker(Ki= 0.16 nM) and a potent dopamine D2 receptor antagonist(Ki= 1.4 nM). 了解更多 -
Masupirdine mesylate
Catalog No. A21409 5-HT6 receptor antagonistMasupirdine mesylate (SUVN-502 mesylate) is a potent, selective, orally bioavailable, and brain penetrant 5-HT6 receptor antagonist (Ki of 2.04 nM for human 5-HT6 receptor). 了解更多 -
Ditolylguanidine
Catalog No. A21268 Sigma receptor agonistDitolylguanidine (1,3-Di-o-tolylguanidine) is an agonist of sigma receptor (??1/??2 receptor). 了解更多 -
Zonampanel
Catalog No. A21199 glutamate receptor subtype antagonistZonampanel (YM 872) is a selective antagonist of the glutamate receptor subtype, α-amino-3-hydroxy-5-methylisoxazole-4-propionic acid (AMPA) receptor. 了解更多 -
Toreforant
Catalog No. A21058 histamine H4 receptor (H4R) antagonistToreforant is a potent and selective histamine H4 receptor (H4R) antagonist, with a Ki at the human receptor of 8.4 nM. 了解更多 -
Pexacerfont
Catalog No. A14105 CRF1 receptor antagonistPexacerfont is a selective corticotropin-releasing factor (CRF1) receptor antagonist with IC50 of 6.1??0.6 nM for human CRF1 receptor. 了解更多 -
LY-2940094
Catalog No. A19125 NOP receptor antagonistLY-2940094 is a potent, selective and orally available nociceptin receptor (NOP receptor) antagonist with high affinity (Ki=0.105 nM) and antagonist potency (Kb=0.166 nM). LY-2940094 reduces ethanol self-administration in animal models. 了解更多 -
Fimasartan
Catalog No. A17477 non-peptide angiotensin II receptor antagonistFimasartan is a non-peptide angiotensin II receptor antagonist (ARB) used for the treatment of hypertension and heart failure. Through oral administration, fimasartan blocks angiotensin II receptor type 1 (AT1 receptors), reducing pro-hypertensive actions of angiotensin II, such as systemic vasoconstriction and water retention by the kidneys. 了解更多 -
Lobeline hydrochloride
Catalog No. A17333 nicotinic receptor agonistLobeline hydrochloride, a nicotinic receptor agonist, acting as a potent antagonist at both α3β2 and α4β2 neuronal nicotinic receptor subtypes. 了解更多 -
Angiotensin III
Catalog No. A18943 angiotensin 1 (AT1) and AT2 receptor agonistAngiotensin III is an angiotensin 1 (AT1) and AT2 receptor agonist. 了解更多 -
BAY 2416964
Catalog No. A22067 aryl hydrocarbon receptor (AHR) antagonistBAY 2416964 is a potent and orally active aryl hydrocarbon receptor (AHR) antagonist extracted from patent WO2018146010A1, example 192, has an IC50 of 341 nM. BAY 2416964 has the potential for solid tumors treatment. 了解更多 -
WAY-169916
Catalog No. A22105 pathway-selective inhibitor of estrogen receptor (ER)WAY-169916 is a pathway-selective inhibitor of estrogen receptor (ER) that acts by inhibiting NF-kB transcriptional activity. 了解更多 -
Cytosporone B
Catalog No. A22115 nuclear orphan receptor Nur77/NR4A1 agonistCytosporone B (Csn-B; Dothiorelone G) is a naturally occurring nuclear orphan receptor Nur77/NR4A1 agonist with an EC50 of 0.278 nM. 了解更多 -
RO5203648 hydrochloride
Catalog No. A22118 partial agonist of Trace amine-associated receptor 1RO5203648 hydrochloride is a partial agonist of Trace amine-associated receptor 1 (TAAR1). 了解更多 -
BMS-986188
Catalog No. A22124 Positive Allosteric Modulator of the delta-Opioid ReceptorBMS-986188 is a novel Potent and Selective Positive Allosteric Modulator of the delta-Opioid Receptor. 了解更多 -
BMS-986187
Catalog No. A22125 positive allosteric modulator (PAM) of the δ-opioid receptor and a G-protein-biased allosteric agonistBMS-986187 is a potent and selective positive allosteric modulator (PAM) of the δ-opioid receptor and a G-protein-biased allosteric agonist. 了解更多 -
Adenosine amine congener
Catalog No. A22193 A1 adenosine receptor agonistAdenosine amine congener (ADAC) is a selective A1 adenosine receptor agonist, can ameliorate noise- and Cisplatin-induced cochlear injury. 了解更多 -
5-HT3 antagonist-4i
Catalog No. A22265 5-HT3 receptor antagonist5-HT3 antagonist-4i is a 5-HT3 receptor antagonist which modulates the serotonergic system. 了解更多 -
Amarogentin
Catalog No. A22286 bitter taste receptor TAS2R1 agonistAmarogentin (AG), a secoiridoid glycoside mainly extracted from Swertia and Gentiana roots, exhibits anti-oxidative, anti-tumour, and anti-diabetic activities. Amarogentin is an agonist for the bitter taste receptor TAS2R1 and inhibits in LAD-2 cells substance P-induced production of newly synthesized TNF-α. 了解更多 -
Emedastine
Catalog No. A22158 histamine H1 receptor antagonistEmedastine is an orally active, selective and high affinity histamine H1 receptor antagonist with a Ki value of 1.3 nM. 了解更多 -
SSD114 hydrochloride
Catalog No. A22188 GABAB receptor positive allosteric modulatorSSD114 hydrochloride is a novel GABAB receptor positive allosteric modulator. 了解更多 -
Cholesterol
Catalog No. A22211 endogenous estrogen-related receptor α (ERRα) agonistCholesterol is also an endogenous estrogen-related receptor α (ERRα) agonist. 了解更多
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