“inhibitor”的搜索结果

产品 151 到 200 共 5361个

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  1. DNA2 inhibitor C5

    Catalog No. A19091
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    DNA2 inhibitor
    DNA2 inhibitor C5 is a potent, competitive and specific inhibitor of DNA2 nuclease activity with an IC50 of 20 μM. 了解更多
  2. Sodium Channel inhibitor 2

    Catalog No. A20453
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    sodium channel blocker
    Sodium Channel inhibitor 2 is a sodium channel blocker extracted from patent WO 2004011439 A2, compound 3c. 了解更多
  3. NAMPT inhibitor-linker 1

    Catalog No. A19922
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    NAMPT inhibitor-linker 1 is a drug-linker conjugates for ADC, composed of an NAMPT inhibitor as a payload, and a linker. 了解更多
  4. NAMPT inhibitor-linker 2

    Catalog No. A19912
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    drug-linker conjugates for ADC
    NAMPT inhibitor-linker 2 is a drug-linker conjugates for ADC, composed of an NAMPT inhibitor as a payload, and a linker. 了解更多
  5. IRAK inhibitor 3

    Catalog No. A11457
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    IL-1 receptor-associated kinase (IRAK) kinase modulator
    IRAK inhibitor 3 is an interleukin-1 (IL-I) receptor-associated kinase (IRAK) kinase modulator extracted from patent WO2008030579 A2. 了解更多
  6. Ubiquitin Isopeptidase Inhibitor I, G5

    Catalog No. A12293
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    apoptosis activator
    Ubiquitin Isopeptidase Inhibitor I, G5 (NSC 144303) is an apoptosome-independent caspase and apoptosis activator with IC50 values of 1.76 and 1.6 μM in E1A and E1A/C9DN cells, respectively. 了解更多
  7. Casein Kinase II Inhibitor IV

    Catalog No. A12624
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    Epidermal keratinocyte differentiation inducer
    Casein Kinase II Inhibitor IV is a small-molecule inducer of epidermal keratinocyte differentiation. 了解更多
  8. Apoptosis Inhibitor (M50054)

    Catalog No. A13058
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    Apoptosis 抑制剂
    Apoptosis Inhibitor (M50054)是细胞可渗透的凋亡诱导抑制剂。 了解更多
  9. RIP2 kinase inhibitor 2

    Catalog No. A16313
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    RIP2 kinase 抑制剂
    RIP2 kinase inhibitor 2 是从专利WO/2014043437 A1(化合物实施例9)中提取的受体相互作用蛋白2(RIP2)激酶抑制剂。 了解更多
  10. RIP2 kinase inhibitor 1

    Catalog No. A16312
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    RIP2 kinase 抑制剂
    RIP2 kinase inhibitor 1 是从专利WO/2014043446 A1(化合物实施例1)中提取的受体相互作用蛋白2(RIP2)激酶抑制剂。 了解更多
  11. PI3K-gamma inhibitor 1

    Catalog No. A16275
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    PI3Kγ 抑制剂
    PI3K-gamma inhibitor 1 是有效的PI3Kγ抑制剂。 了解更多
  12. PI3K-alpha inhibitor 1

    Catalog No. A16274
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    PI3Kα 抑制剂
    PI3K-alpha inhibitor 1 是从专利US/20120088764A1中提取的PI3Kα抑制剂,化合物243,IC50 <0.1uM,PI3Kα抑制剂1还抑制HDAC(0.1uM≤IC50≤1uM)。 了解更多
  13. Btk inhibitor 1

    Catalog No. A16260
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    BTK 抑制剂
    Btk inhibitor 1 是作为Btk激酶抑制剂的吡唑并[3,4-d]嘧啶衍生物。 了解更多
  14. c-Met inhibitor 2

    Catalog No. A16256
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    c-Met 抑制剂
    c-Met inhibitor 2 是有效的化合物,对依赖于Met激活的癌症具有活性,并且还具有作为VEGFR抑制剂的抗癌活性。 了解更多
  15. PDK1 inhibitor

    Catalog No. A16185
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    PDK1 抑制剂
    PDK1 inhibitor,强效,ATP竞争性和选择性双重PI3K和PDPK1抑制剂(PDK1和p-T308-PKB抑制的IC50值分别为34 nM和94 nM。 了解更多
  16. K+ Channel inhibitor

    Catalog No. A16182
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    K+ Channel 抑制剂
    K+ Channel inhibitor,Kv1.5(IKur)的二氢吡唑并嘧啶抑制剂的合成基础。 了解更多
  17. HIF-2a Translation Inhibitor

    Catalog No. A16181
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    HIF-2a translation 抑制剂
    HIF-2a Translation Inhibitor(IC50值为5 uM);独立于HIF-2a mRNA表达或HIF-2a蛋白稳定性,并独立于mTOR活性,降低常氧和低氧状态下HIF-2a蛋白和HIF-2a目标基因的表达。此外,翻译抑制剂76增强了IRP1与HIF-2a IRE(铁反应元件)的结合。 了解更多
  18. cGMP Dependent Kinase Inhibitor Peptid

    Catalog No. A16052
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    PKG/PKA 抑制剂
    cGMP Dependent Kinase Inhibitor Peptid是一种特定的cGKI(环GMP依赖性蛋白激酶)抑制剂。数据表明,它不阻断完整组蛋白的环状GMP依赖性蛋白激酶磷酸化,已被用于研究恶性疟原虫。 了解更多
  19. Cathepsin Inhibitor 1

    Catalog No. A11466
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    Cathepsin 抑制剂
    Cathepsin Inhibitor 1抑制剂1 是一种Cathepsin (L, L2, S, K, B)的抑制剂,pIC50分别为7.9、6.7、6.0、5.5和5.2。 了解更多
  20. PD1-PDL1 inhibitor 2

    Catalog No. A15906
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    PD-1/PD-L1 interaction 抑制剂
    PD1-PDL1 inhibitor 2 是PD-1/PD-L1相互作用抑制剂。 了解更多
  21. IRAK-1-4 Inhibitor I

    Catalog No. A11462
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    IRAK-1-4 Inhibitor I是一种苯并咪唑,它破坏IRAK-1和-4的活性,其IC50值分别为300和200 nM。 了解更多
  22. ALK inhibitor 2

    Catalog No. A14988
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    ALK 抑制剂
    ALK inhibitor 2 是ALK激酶的新型选择性抑制剂。 了解更多
  23. ALK inhibitor 1

    Catalog No. A14987
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    ALK 抑制剂
    ALK inhibitor 1 是ALK激酶的新型选择性抑制剂。 了解更多
  24. Bax inhibitor peptide V5

    Catalog No. A15337
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    Bax 抑制剂
    Bax inhibitor peptide V5,Bax易位至线粒体的细胞渗透性合成肽抑制剂;由Ku70设计的一种蛋白质,被认为可抑制Bax的线粒体易位。在体外抑制Bax介导的细胞凋亡。 了解更多
  25. Bax inhibitor peptide P5

    Catalog No. A15336
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    Bax 抑制剂
    Bax inhibitor peptide P5,Bax易位至线粒体的细胞渗透性合成肽抑制剂;由Ku70设计的一种蛋白质,被认为可抑制Bax的线粒体易位。在体外抑制Bax介导的细胞凋亡。 了解更多
  26. Sodium Channel inhibitor 1

    Catalog No. A15243
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    Sodium Channel 抑制剂
    Sodium Channel inhibitor 1 是一种新型的选择性电压门控钠通道,用于疼痛治疗。 了解更多
  27. ROCK inhibitor-1

    Catalog No. A15226
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    ROCK 抑制剂
  28. p53 and MDM2 proteins-interaction-inhibitor racemic

    Catalog No. A15202
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    p53-MDM2 interaction 抑制剂
    p53和MDM2蛋白相互作用抑制剂消旋体是p53和MDM2蛋白之间相互作用的抑制剂。 了解更多
  29. mTOR inhibitor (mTOR-IN-1)

    Catalog No. A15175
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    mTOR 抑制剂
    mTOR inhibitor (mTOR-IN-1)是mTOR的有效且选择性的ATP竞争性抑制剂,Ki为1.5 nM。 了解更多
  30. Lck inhibitor 2

    Catalog No. A15141
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    Lck 抑制剂
    Lck inhibitor 2 是酪氨酸激酶的双苯胺基嘧啶抑制剂,包括LCK,BTK,LYN,SYK和TXK。Lck,Btk,Lyn,Btk和Txk的IC50值分别为13nM,9nM,3nM,26nM和2nM。 了解更多
  31. DGAT-1 inhibitor 2

    Catalog No. A15067
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    DGAT-1 抑制剂
    DGAT-1 inhibitor 2 是有效的DGAT-1抑制剂。 了解更多
  32. c-Met inhibitor 1

    Catalog No. A15049
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    c-Met 抑制剂
    c-Met inhibitor 1 是c-Met受体信号传导途径的抑制剂,可作用于胃癌,胶质母细胞瘤和胰腺癌在内的癌症。 了解更多
  33. CDK9 inhibitor 2

    Catalog No. A15039
    CDK9 抑制剂
    CDK9 inhibitor 2 是一种新型的细胞周期蛋白依赖性激酶9(CDK9)抑制剂。 了解更多
  34. Carboxypeptidase G2 (CPG2) Inhibitor

    Catalog No. A15035
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    CPG2 抑制剂
    Carboxypeptidase G2 (CPG2) Inhibitor是一种新型的羧肽酶G2(CPG2)抑制剂。 了解更多
  35. Caspase-3/7 Inhibitor I

    Catalog No. A14919
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    Caspase-3/7 抑制剂
    Caspase-3/7 Inhibitor I是caspase-3(Ki = 60 nM)和caspase-7(Ki = 170 nM)的有效,细胞可渗透且可逆的有效抑制剂。 了解更多
  36. Elastase Inhibitor, SPCK

    Catalog No. A14913
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    HLE 抑制剂
    Elastase Inhibitor,SPCK是一种有效的不可逆的人类白细胞弹性蛋白酶(HLE)抑制剂(Ki = 10 uM)。 了解更多
  37. Calpain Inhibitor II, ALLM

    Catalog No. A14911
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    Calpain 抑制剂
    Calpain Inhibitor II, ALLM是钙蛋白酶I,钙蛋白酶II,组织蛋白酶L和组织蛋白酶B的细胞可渗透抑制剂,Ki值分别为120 nM,230 nM,0.6 nM和100 nM。 了解更多
  38. PKA inhibitor fragment (6-22) amide

    Catalog No. A14868
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    PKA 抑制剂
    PKA inhibitor fragment (6-22) amide是一种合成肽,可作为蛋白激酶抑制剂。 了解更多
  39. EGFR Inhibitor

    Catalog No. A13673
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    EGFR 抑制剂
    EGFR inhibitor是一种可透过细胞的4,6-二取代嘧啶化合物,可选择性抑制EGFR激酶,在体外的IC50值为21 nM,可阻断细胞中的受体自身磷酸化。 了解更多
  40. K-Ras(G12C) inhibitor 12

    Catalog No. A14227
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    K-Ras(G12C) 抑制剂
    K-Ras(G12C) inhibitor 12 是致癌性K-Ras(G12C)的变构抑制剂。 了解更多
  41. PI3k-delta inhibitor 1

    Catalog No. A14109
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    PI3Kδ 抑制剂
    PI3k-delta inhibitor 1是有效的选择性PI3Kδ抑制剂,IC50为3.8 nM。 了解更多
  42. K-Ras(G12C) inhibitor 6

    Catalog No. A14103
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    K-Ras(G12C) 抑制剂
    K-Ras(G12C) inhibitor 6 是致癌性K-Ras(G12C)的不可逆抑制剂,颠覆了天然核苷酸的偏爱性,使GDP优于GTP。 了解更多
  43. NSC 42834(JAK2 Inhibitor V, Z3)

    Catalog No. A14132
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    JAK2 抑制剂
    NSC 42834(JAK2 Inhibitor V,Z3)是一种新型的Jak2酪氨酸激酶特异性抑制剂。 了解更多
  44. HPGDS inhibitor 1

    Catalog No. A12258
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    HPGDS 抑制剂
    HPGDS inhibitor 1是一种新的选择性造血前列腺素d合酶(HPGDS)抑制剂,IC50值为0.7 nM。 了解更多
  45. MDM2 Inhibitor

    Catalog No. A13582
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    MDM2 抑制剂
    MDM2 Inhibitor是一种细胞可渗透的硼烷基查尔酮,表现出与MDM2的强结合,并不可逆地破坏MDM2/p53蛋白复合物。 了解更多
  46. Lavendustin B

    Catalog No. A22298
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    GLUT1 inhibitor
    Lavendustin B is an inhibitor of HIV-1 integrase interaction with LEDGF/p75 with an IC50 of 94.07 μM. Lavendustin B is an ATP-competitive GLUT1 inhibitor with a Ki of 15 ?M. Lavendustin B is also a weak inhibitor of tyrosine kinases. 了解更多
  47. GSK1940029

    Catalog No. A20820
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    SCD inhibitor
    GSK1940029 (SCD inhibitor 1) is a stearoyl-coa desaturase (SCD) inhibitor extracted from patent WO/2009060053 A1, compound example 16. 了解更多
  48. IACS-8968

    Catalog No. A20020
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    dual IDO/TDO inhibitor
    IACS-8968 (IDO/TDO Inhibitor) is a dual IDO and TDO inhibitor, with pIC50s of 6.43 for IDO and <5 for TDO, respectively. 了解更多
  49. Upamostat

    Catalog No. A21035
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    serine protease inhibitor
    Upamostat is a serine protease inhibitor. Upamostat is the orally available prodrug of the WX-UK1, which is a urokinase plasminogen activator (uPA) inhibitor. 了解更多
  50. X-376

    Catalog No. A20971
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    ALK tyrosine kinase inhibitor
    X-376 is a potent and highly specific ALK tyrosine kinase inhibitor (TKI) (IC50=0.61 nM). X-376 is a less potent inhibitor of MET (IC50=0.69 nM). X-376 displays potent anti-tumor activity. 了解更多

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