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￥ 0.00 “AG 013736”的搜索结果
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2-Methoxycinnamaldehyde
Catalog No. A12965 antitumor agent2-Methoxycinnamaldehyde (o-Methoxycinnamaldehyde) is a natural compound of Cinnamomum cassia, with antitumor activity. 了解更多 -
Ginsenoside Rc
Catalog No. A15565 anti-cancer agentGinsenoside Rc, isolated from Panax ginseng, may exert various activities including anti-cancer, anti-inflammatory, antiobesity, and anti-diabetic effects. 了解更多 -
Methyl protodioscin
Catalog No. A15690 antitumor agentMethyl protodioscin(NSC-698790) is a furostanol bisglycoside with antitumor properties; shows to reduce proliferation, cause cell cycle arrest. 了解更多 -
L-SelenoMethionine
Catalog No. A17926 cancer chemopreventive agentL-SelenoMethionine, an L-isomer of Selenomethionine, is a major natural food-form of selenium. L-SelenoMethionin is a cancer chemopreventive agent that can reduce cancer incidence by dietary supplementation and induce apoptosis of cancer cells. 了解更多 -
Ketoprofen
Catalog No. A10499 non-steroidal antiinflammatory agentKetoprofen (RP-19583) is a non-steroidal antiinflammatory agent, acting as a potent inhibitor of COX, with IC50s of 2 nM and 26 nM for COX-1 and COX-2 in human blood monocytes, respectively. 了解更多 -
Geniposidic acid
Catalog No. A11630 anticancer and radioprotection agentGeniposidic acid is an effective anticancer and radioprotection agent. 了解更多 -
Lonidamine
Catalog No. A11633 antitumor agentLonidamine (AF-1890), an antitumor agent, is a hexokinase, mitochondrial pyruvate carrier (Ki 2.5 μM in isolated rat liver mitochondria) and plasma membrane monocarboxylate transporters inhibitor, which also inhibits mitochondrial complex II. 了解更多 -
Fenoprofen Calcium hydrate
Catalog No. A16547 nonsteroidal, anti-inflammatory antiarthritic agentFenoprofen Calcium hydrate is a nonsteroidal, anti-inflammatory antiarthritic agent. 了解更多 -
L-Ascorbic acid
Catalog No. A15465 elastogenesis inhibitorL-Ascorbic acid (L-Ascorbate), an electron donor, is an endogenous antioxidant agent. L-Ascorbic acid inhibits selectively Cav3.2 channels with an IC50 of 6.5 μM. L-Ascorbic acid is also a collagen deposition enhancer and an elastogenesis inhibitor. 了解更多 -
Sodium Salicylate
Catalog No. A16716 S6K inhibitorSodium Salicylate (Salicylic acid sodium salt) inhibits cyclo-oxygenase-2 (COX-2) activity independently of transcription factor (NF-κB) activation. Sodium Salicylate is also a S6K inhibitor.Sodium Salicylate is a NF-κB inhibitor that decreases inflammatory gene expression and improves repair in aged muscle. 了解更多 -
Diammonium Glycyrrhizinate
Catalog No. A17257 anti-inflammatory agentDiammonium Glycyrrhizinate, isolated from the licorice root, is a widely used anti-inflammatory agent. 了解更多 -
Levofloxacin
Catalog No. A10528 Levofloxacin is a fluoroquinolone antibiotic. It is active against S. aureus, S. epidermidis, B. subtilis, E. coli, P. aeruginosa, and K. pneumoniae (MICs = 0.25, 0.25, 0.5, 0.03, 4, and 0.25 μg/ml, respectively). 了解更多 -
Blarcamesine (AVex-73)
Catalog No. A21095 muscarinic M1 agonistBlarcamesine, also known as AVex-73 and AE-37, is a muscarinic M1 agonist potentially for the treatment of Alzheimer's disease. It is an σ receptor ligand. 了解更多 -
ML-9 hydrochloride
Catalog No. A17856 MLCK inhibitorML-9 is a selective and potent inhibitor of Akt kinase, inhibits myosin light-chain kinase (MLCK) and stromal interaction molecule 1 (STIM1) activity. ML-9 inhibits inhibits MLCK, PKA and PKC activity with Ki values of 4, 32 and 54 μM, respectively. ML-9 induces autophagy by stimulating autophagosome formation and inhibiting their degradation. 了解更多 -
IT1t dihydrochloride
Catalog No. A22027 CXCR4 antagonistIT1t dihydrochloride is a potent CXCR4 antagonist; inhibits CXCL12/CXCR4 interaction with an IC50 of 2.1 nM. 了解更多 -
Sograzepide
Catalog No. A22020 Gastrin/CCK-B antagonistSograzepide (Netazepide; YF 476; YM-220) is an extremely potent , highly selective and orally active Gastrin/CCK-B antagonist with an IC50 value of 0.1 nM, has inhibitory effect on Gastrin/CCK-A activity with an IC50 of 502 nM. 了解更多 -
Pridopidine
Catalog No. A22009 D2R antagonistPridopidine, a dopamine (DA) stabilizer, acts as a low affinity dopamine D2 receptor (D2R) antagonist. 了解更多 -
Eplivanserin
Catalog No. A21967 5-HT2 receptor antagonistEplivanserin is a potent, selective and orally available 5-HT2 receptor antagonist, with an IC50 of 5.8 nM in rat cortical membrane, and a Kd of 1.14 nM. 了解更多 -
4-Phenoxybenzylamine
Catalog No. A20959 4-Phenoxybenzylamine inhibits the function of the NS3 protein by stabilizing an inactive conformation with an IC50 of about 500 μM against FL NS3/4a. 了解更多 -
WAY-151932
Catalog No. A20821 vasopressin V2-receptor agonistWAY-151932 is a vasopressin V2-receptor agonist with IC50 of 80.3 nM and 778 nM in human-V2 binding and V1a binding assay. 了解更多 -
(E)-[6]-Dehydroparadol
Catalog No. A20817 (E)-[6]-Dehydroparadol, extracted from patent US 9272994, compound M15, shows growth inhibition and induction of apoptosis against human cancer cells with IC50 values of 43.02 μM in HCT-116 cell and 41.59 μM in H-1299 cell, respectively. 了解更多 -
Ertiprotafib
Catalog No. A20815 PTP1B/IKK-βinhibitor and dual PPARα and PPARβ agonistErtiprotafib is an inhibitor of PTP1B, IkB kinase β (IKK-β), and a dual PPARα and PPARβ agonist, with an IC50 of 1.6 μM for PTP1B, 400 nM for IKK-β, an EC50 of ~1 μM for PPARα/PPARβ. 了解更多 -
Amphethinile
Catalog No. A20814 anti-tubulin agentAmphethinile is an anti-tubulin agent. The affinity constant for the association (Ka) of Amphethinile with tubulin is 1.3 μM. 了解更多 -
Phenylbiguanide
Catalog No. A20812 5-HT3 receptor selective agonistPhenylbiguanide is a 5-HT3 receptor selective agonist with an EC50 of 3.0±0.1 μM. 了解更多 -
(-)-Aspartic acid
Catalog No. A20810 -
BMY-25271
Catalog No. A20809 -
Val-Cit-PAB-MMAE
Catalog No. A20808 drug-linker conjugate for ADCVal-Cit-PAB-MMAE is a drug-linker conjugate for ADC by using the anti-mitotic agent, monomethyl auristatin E (MMAE, a tubulin inhibitor), linked via the peptide Val-Cit-PAB. 了解更多 -
Deschloroclozapine
Catalog No. A20801 dual dopamine and serotonin receptor antagonistDeschloroclozapine is a dual dopamine and serotonin receptor antagonist with Kis of 200, 2500, 420, 39, 84, 40 nM for dopamine D1, D2,D4, and serotonin S2A, S2C, S3, respectively. 了解更多 -
Setogepram sodium salt
Catalog No. A20796 GPR40 agonistSetogepram sodium salt (PBI-4050 sodium salt) acts as an orally active agonist for GPR40 and as an antagonist or inverse agonist for GPR84. 了解更多 -
Aganepag
Catalog No. A20794 Prostanoid EP2 receptor agonistAganepag is a potent Prostanoid EP2 receptor agonist, with an EC50 of 0.19 nM, and shows no activity at EP4 receptor. Aganepag can be used in the research of wound healing, scar reduction, scar prevention and wrinkle treatment and prevention. 了解更多 -
trans-ACPD
Catalog No. A20779 metabotropic receptor agonisttrans-ACPD, a metabotropic receptor agonist, produces calcium mobilization and an inward current in cultured cerebellar Purkinje neurons. 了解更多 -
Solabegron
Catalog No. A20778 β3-adrenergic receptor agonistSolabegron (GW 427353) is a selective β3-adrenergic receptor agonist, stimulating cAMP accumulation in Chinese hamster ovary cells expressing the human β3-AR, with an EC50 value of 22 nM. 了解更多 -
SSR-241586
Catalog No. A20773 neurokinin receptors antagonistSSR-241586 is an antagonist of neurokinin receptors. SSR-241586 is shown to be active in the treatment of depression, schizophrenia, urinary trouble, emesis, and irritable bowel syndrome (IBS). 了解更多 -
Roluperidone
Catalog No. A20770 5-HT2/sigma 2 receptor antagonistRoluperidone, also known as MIN-101, CYR-101, and MT-210, is a 5-HT2A and sigma 2 receptor antagonist potentially for the treatment of schizophrenia. 了解更多
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