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MRK-016
Catalog No. A12046 GABAA α5 receptor agonistMRK-016 is a selective, orally bioavailable inverse agonist of GABAA α5 receptor, with an EC50 of 3 nM for GABAA α5, and Kis of 0.83, 0.85, 0.77?and 1.4?nM for human?GABAA?α1β3γ2, GABAA?α2β3γ2, GABAA?α3β3γ2, and GABAA?α5β3γ2, respectively; MRK-016 also readily penetrates the CNS. 了解更多 -
Motixafortide
Catalog No. A22276 CXCR4 antagonistMotixafortide (BKT140 4-fluorobenzoyl) is a novel CXCR4 antagonist with an IC50 vakue of ??1 nM. 了解更多 -
Oct3/4-inducer-1
Catalog No. A22642 Oct3/4 inducerOct3/4-inducer-1 (compound 2) is a potent Oct3/4 inducer. Oct3/4-inducer-1 promotes expression and stabilization of Oct3/4, and enhances its transcriptional activity in diverse human somatic cells. 了解更多 -
PAβN dihydrochloride
Catalog No. A22016 efflux pump inhibitorPAβN dihydrochloride (MC-207110 dihydrochloride) is an efflux pump inhibitor. 了解更多 -
AM-92016 hydrochloride
Catalog No. A20472 IK blockerAM-92016 hydrochloride is a specific blocker of rectifier potassium current (IK). 了解更多 -
DC1SMe
Catalog No. A20181 DC1Sme, a DC1 derivative, exhibits IC50 values of 22 pM, 10 pM, 32 pM and 250 pM for Ramos, Namalwa, HL60/s and COLO 205 cancer cells, respectively. DC1, a simplified analogue of CC-1065, is an antibody conjugate of cytotoxic DNA alkylators for the targeted treatment of cancer. 了解更多 -
(S,R,S)-AHPC-PEG6-C4-Cl
Catalog No. A20169 (S,R,S)-AHPC-PEG6-C4-Cl is a small molecule HaloPROTAC that incorporates the (S,R,S)-AHPC based VHL ligand and 6-unit PEG linker. (S,R,S)-AHPC-PEG6-C4-Cl is capable of inducing the degradation of GFP-HaloTag7 in cell-based assays. 了解更多 -
Polymyxin B nonapeptide
Catalog No. A20168 Polymyxin B nonapeptide is a cyclic peptide obtained from Polymyxin B by proteolytic removal of its terminal amino acyl residue. Polymyxin B nonapeptide is less toxic, lacks bactericidal activity, and retains its ability to render gram-negative bacteria susceptible to several antibiotics by permeabilizing their outer membranes. 了解更多 -
EOAI3402143
Catalog No. A20166 DUB inhibitorEOAI3402143 is a deubiquitinase (DUB) inhibitor, which inhibits dose-dependently inhibits Usp9x/Usp24 and Usp5. 了解更多 -
FK1052 hydrochloride
Catalog No. A20164 5-HT3 /5-HT4 receptor dual antagonistFK1052 hydrochloride is a potent 5-HT3 and 5-HT4 receptor dual antagonist. 了解更多 -
Heterocyclyl carbamate derivative 1
Catalog No. A20163 Heterocyclyl carbamate derivative 1 is a heterocyclyl carbamate derivative that may be used for the research of inflammatory and neurological diseases. 了解更多 -
BET-IN-2
Catalog No. A20162 -
Thalidomide-O-amido-PEG3-C2-NH2
Catalog No. A20161 E3 ligase ligand-linker conjugateThalidomide-O-amido-PEG3-C2-NH2 is a synthesized E3 ligase ligand-linker conjugate that incorporates the Thalidomide based cereblon ligand and 3-unit PEG linker used in PROTAC technology. 了解更多 -
PROTAC BET Degrader-1
Catalog No. A20016 BET degraderPROTAC BET Degrader-1 is a potent BET degrader based on PROTAC, decreasing BRD2, BRD3, and BRD4 protein levels at low concentration. 了解更多 -
SMYD2-IN-1
Catalog No. A19908 SMYD2 inhibitorSMYD2-IN-1 is a SMYD2 inhibitor extracted from patent WO2016166186A1, compound example 1.1, has an IC50 of 4.45 nM. 了解更多 -
Nitroaspirin
Catalog No. A19145 Nitroaspirin (NCX 4016) is a nitric oxide (NO) donor and a nitro-derivative of Aspirin, which combines with Nitroaspirin to inhibit cyclooxygenase. Nitroaspirin (NCX 4016) has antithrombotic and anti-platelet properties and acts as a direct and irreversible inhibitor of COX-1. 了解更多 -
Pparδ agonist 2
Catalog No. A13262 PPARδ agonistPparδ agonist 2 is a PPARδ agonist extracted from patent WO 2016057656 A1. 了解更多 -
MethADP sodium salt
Catalog No. A21603 -
CRA-026440
Catalog No. A12179 -
Glycolic acid oxidase inhibitor 1
Catalog No. A13016 glycolate oxidase inhibitorGlycolic acid oxidase inhibitor 1 is a glycolate oxidase inhibitor, extracted from patent EP0021228A1, in Table IV. 了解更多 -
HPGDS inhibitor 2
Catalog No. A18390 H-PGDS 抑制剂HPGDS inhibitor 2 is a highly potent and selective hematopoietic prostaglandin D synthase (H-PGDS) inhibitor with an IC50 of 9.9 nM. 了解更多 -
CB1 antagonist 2
Catalog No. A18810 CB1 antagonistCB1 antagonist 2 is caimabinoid 1 (CB1) antagonist extracted from patent WO2016184310A1, compound 3, inhibits CB1 in vivo with an IC50 of 25.5 nM. 了解更多 -
UDM-001651
Catalog No. A18843 PAR4 antagonistUDM-001651 is a potent , selective and orally active Protease-Activated Receptor 4 (PAR4) Antagonist with in Vivo Antithrombotic Efficacy (IC50 = 2.4 nM). 了解更多 -
Bromodomain IN-1
Catalog No. A18845 Bromodomain inhibitorBromodomain IN-1 is a Bromodomain inhibitor extracted from patent WO2016069578A1, compound 4 . 了解更多 -
cIAP1 Ligand-Linker Conjugates 15
Catalog No. A19016 PROTAC linkercIAP1 Ligand-Linker Conjugates 15 incorporates an IAP ligand for the E3 ubiquitin ligase, and a PROTAC linker. cIAP1 Ligand-Linker Conjugates 15 can be used to design SNIPERs. 了解更多 -
RV01
Catalog No. A19104 ALDH2 inhibitorRV01 is an analogue of resveratrol, inhibits DNA damage, reduces acetaldehyde dehydrogenase 2 (ALDH2) mRNA expression induced by ethanol, and exhibits hydroxyl radical scavenging activity. RV01 decreases iNOS expression, with anti-neuroinflammatory activity. 了解更多 -
NRA-0160
Catalog No. A20128 Dopamine D4 receptor antagonistNRA-0160 is a selective dopamine D4 receptor antagonist, with a Ki value of 0.48 nM and with negligible affinity for dopamine D2 receptor (Ki: >10000 nM), D3 receptor (Ki: 39 nM), rat 5-HT2A receptor (Ki: 180 nM) and rat α1 adrenoceptor (Ki: 237 nM). 了解更多 -
Bepridil hydrochloride
Catalog No. A18016 calcium channel blockerBepridil hydrochloride (CERM 1978) is a calcium channel blocker, with antianginal activity. 了解更多 -
VU6005806
Catalog No. A18488 M4 modulatorVU6005806 (AZN-00016130) is a potent muscarnic acethylcholine receptor subtype 4 (M4) positive allosteric modulator (PAM), with EC50s of 94 nM, 28 nM, 87 nM and 68 nM for human, rat, dog and cyno M4, respectively. Used in the research of neuropsychiatric disorders. 了解更多
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