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Endocrinology / Hormones

产品 1 到 50 共 59个

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  1. SR-2211
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    SR-2211

    Catalog No. A13568
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    RORr 激动剂
    SR-2211选择性结合RORr（Ki = 105 nM），充当体外本构RORr活性的反向激动剂（IC50 = 320 nM）。 了解更多
  2. Cintirorgon (LYC-55716)
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    Cintirorgon (LYC-55716)

    Catalog No. A16863
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    RORγ 激动剂
    Cintirorgon (LYC-55716)是新型口服RAR相关孤儿受体γ（RORγ）激动剂。 了解更多
  3. AZD-0284
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    AZD-0284

    Catalog No. A18766
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    RORγ 激动剂
    AZD-0284 is a potent, selective, inverse agonist of the nuclear receptor RORγ for the potential treatment of Plaque psoriasis. 了解更多
  4. XY101
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    XY101

    Catalog No. A18437
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    RORγ inverse 激动剂
    XY101 is a potent, selective, metabolically stable and orally available RORγ inverse agonist with an IC50 of 30 nM and a Kd of 380 nM. 了解更多
  5. A-9758
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    A-9758

    Catalog No. A19078
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    RORγt inverse 激动剂
    A-9758 is a RORγ ligand and a potent, selective RORγt inverse agonist (IC50=5 nM), and exhibits robust potency against IL-17A release. 了解更多
  6. ROR agonist-1
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    ROR agonist-1

    Catalog No. A18569
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    ROR 激动剂
    ROR agonist-1 is a potent and orally bioavailable inverse agonist of the retinoic acid receptor-related orphan receptor C2 (RORC2), inhibition of IL-17A production from human primary TH 17 cells with a pIC50 of 7.5. 了解更多
  7. SR1078
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    SR1078

    Catalog No. A15245
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    ROR 激动剂
    SR1078是视黄酸受体相关的孤儿受体（ROR）RORα/γ的激动剂；增加RORα靶基因的转录；认为可以增加p53的稳定性。 了解更多
  8. SR3335
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    SR3335

    Catalog No. A15246
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    RORα 激动剂
    SR3335是一种选择性RORα合成配体，直接与RORα结合，但不与其他ROR结合，并且在基于细胞的测定中用作RORα的选择性部分反向激动剂。 了解更多
  9. SR1001
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    SR1001

    Catalog No. A13193
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    ROR 激动剂
    SR1001是选择性的ROR-α和ROR-γ反向激动剂；抑制TH17细胞分化并抑制自身免疫。 了解更多
  10. SR 144528
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    SR 144528

    Catalog No. A12376
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    CB2 inverse 激动剂
    SR 144528是一种选择性的外周大麻素受体反向激动剂，对大鼠脾脏和人重组CB2受体的Ki值为0.6 nM，对大鼠脑和人重组CB1受体的Ki值为400 nM。 了解更多
  11. AEZS-108
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    AEZS-108

    Catalog No. A13536
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    GnRH-1 激动剂
    AEZS-108是促性腺激素释放激素1受体（GnRH-1R）的肽激动剂，其与蒽环类抗生素阿霉素结合，具有潜在的抗肿瘤活性。 了解更多
  12. Leuprolide Acetate
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    Leuprolide Acetate

    Catalog No. A15143
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    GnRH 激动剂
    Leuprolide Acetate是GnRH类似物；醋酸亮丙瑞林在垂体GnRH受体上起激动剂的作用。 了解更多
  13. Triptorelin Acetate
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    Triptorelin Acetate

    Catalog No. A15997
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    GnRH 激动剂
    Triptorelin Acetate是一种促性腺激素释放激素激动剂（GnRH激动剂），用作乙酸盐或pamoate盐。 了解更多
  14. Goserelin Acetate
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    Goserelin Acetate

    Catalog No. A15959
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    GnRH 激动剂
    Goserelin Acetate是具有抗肿瘤活性的促黄体激素释放激素（LHRH）的合成十肽类似物。 了解更多
  15. Leuprorelin Acetate
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    Leuprorelin Acetate

    Catalog No. A17986
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    GnRH/LHRH receptor agonist
    Leuprorelin is a Gonadotropin-releasing hormone (GnRH, luteinizing hormone-releasing hormone, LHRH) receptor agonist. Suppresses estradiol, LH and FSH serum levels and represses the growth of experimental rat endometriosis. 了解更多
  16. Nafarelin Acetate
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    Nafarelin Acetate

    Catalog No. A17992
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    GnRH agonist
    Nafarelin is a gonadotropin-releasing hormone agonist (GnRH agonist) which acts as an analog of GnRH. 了解更多
  17. Goserelin
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    Goserelin

    Catalog No. A21197
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    GnRH agonist
    Goserelin(ICI 118630) is an injectable gonadotropin releasing hormone superagonist (GnRH agonist). 了解更多
  18. Alarelin Acetate
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    Alarelin Acetate

    Catalog No. A20968
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    synthetic GnRH agonist
    Alarelin acetate is a synthetic GnRH agonist. 了解更多
  19. Betamethasone dipropionate
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    Betamethasone dipropionate

    Catalog No. A10130
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    Glucocorticoid Receptor 激动剂
    Betamethasone Dipropionate是糖皮质激素类固醇，具有抗炎和免疫抑制特性。 了解更多
  20. Prednisone (Adasone)
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    Prednisone (Adasone)

    Catalog No. A10752
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    Glucocorticoid Receptor 激动剂
    Prednisone (Adasone)可降低粘膜TNF-a的产生，肠道通透性和NF-kB表达水平。 了解更多
  21. GW-870086
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    GW-870086

    Catalog No. A18343
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    Glucocorticoid receptor agonist
    GW-870086 is a potent anti-inflammatory agent, acting as a glucocorticoid receptor agonist, with a pIC50 of 10.1 in A549 cells expressing NF-κB. 了解更多
  22. Beclometasone
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    Beclometasone

    Catalog No. A18177
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    glucocorticoid receptor agonist
    Beclometasone, also known as Beclomethasone, is an anti-inflammatory, synthetic glucocorticoid. It is used topically as an anti-inflammatory agent and in aerosol form for the treatment of asthma. 了解更多
  23. AZD5423
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    AZD5423

    Catalog No. A13249
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    nonsteroidal glucocorticoid receptor 激动剂
    AZD5423是新型的非甾体类糖皮质激素受体激动剂。 了解更多
  24. AZD2906
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    AZD2906

    Catalog No. A18936
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    glucocorticoid receptor agonist
    AZD2906 is a selective glucocorticoid receptor (GR) agonist, increases micronucleated immature erythrocytes in the bone marrow of rats. AZD2906 shows IC50s of 2.2, 0.3, 41.6 and 7.5 nM at GR in human, rat PBMC and human, rat whole blood, respectively. 了解更多
  25. Glucocorticoid receptor agonist
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    Glucocorticoid receptor agonist

    Catalog No. A11431
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    Glucocorticoid receptor agonist
    Glucocorticoid receptor agonist is a potent Glucocorticoid receptor agonist. 了解更多
  26. Dexamethasone acetate
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    Dexamethasone acetate

    Catalog No. A16494
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    glucocorticoid receptor agonist
    Dexamethasone acetate (Dexamethasone 21-acetate) is a glucocorticoid receptor agonist. 了解更多
  27. Beclometasone dipropionate
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    Beclometasone dipropionate

    Catalog No. A17254
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    glucocorticoid agonist
    Beclometasone dipropionate is a potent glucocorticoid agonist; it is a prodrug of the free form, beclometasone. 了解更多
  28. Fosdagrocorat
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    Fosdagrocorat

    Catalog No. A21303
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    dissociated glucocorticoid receptor agonist
    Fosdagrocorat (PF-04171327) is a dissociated glucocorticoid receptor agonist. 了解更多
  29. Dagrocorat
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    Dagrocorat

    Catalog No. A21312
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    glucocorticoid receptor agonist
    Dagrocorat (PF-00251802) is a novel and dissociated glucocorticoid receptor agonist. 了解更多
  30. (S)-Mapracorat
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    (S)-Mapracorat

    Catalog No. A21528
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    glucocorticoid receptor agonist
    (S)-Mapracorat is a selective and less active glucocorticoid receptor agonist. 了解更多
  31. Mapracorat
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    Mapracorat

    Catalog No. A21953
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    glucocorticoid receptor agonist
    Mapracorat is a novel non-steroidal selective glucocorticoid receptor agonist. 了解更多
  32. CGP-42112
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    CGP-42112

    Catalog No. A21575
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    Angiotensin-II subtype 2 receptor(AT2 R) agonist
    CGP-42112(CGP-42112A) is a potent Angiotensin-II subtype 2 receptor(AT2 R) agonist. 了解更多
  33. AVE 0991
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    AVE 0991

    Catalog No. A20997
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    angiotensin-(1-7) receptor agonist
    AVE 0991 is a nonpeptide and orally active angiotensin-(1-7) receptor agonist with an IC50 of 21 nM. 了解更多
  34. SR-12813
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    SR-12813

    Catalog No. A16125
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    PXR 激动剂
    SR-12813是孕烷X受体（PXR）激动剂。 了解更多
  35. Diphenyleneiodonium chloride
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    Diphenyleneiodonium chloride

    Catalog No. A13359
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    GPR3 激动剂/NOS/ NADPH oxidases 抑制剂
    Diphenyleneiodonium是一种有效的不可逆的巨噬细胞抑制剂NOS2（iNOS）和内皮细胞NOS3（eNOS）抑制剂。 了解更多
  36. MBX-2982
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    MBX-2982

    Catalog No. A12634
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    GPR119 激动剂
    MBX-2982是针对2型糖尿病的潜在一流疗法，其靶向G蛋白偶联受体119（GPR119），该受体与已知刺激葡萄糖依赖性胰岛素分泌的生物活性脂质相互作用。 了解更多
  37. AR-231453
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    AR-231453

    Catalog No. A13716
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    GPR119 激动剂
    AR-231453是GPR119的一种有效的，选择性的小分子药物，可增强葡萄糖依赖性胰岛素分泌和胰高血糖素样肽1（GLP-1）的释放。 了解更多
  38. APD668
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    APD668

    Catalog No. A14342
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    GPR119 激动剂
    APD668是有效的GPR119激动剂，hGPR119和ratGPR119的EC50分别为2.7 nM和33 nM。 了解更多
  39. AMG 837 calcium hydrate
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    AMG 837 calcium hydrate

    Catalog No. A13468
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    GPR40/FFA1 激动剂
    AMG-837 calcium hydrate是一种口服生物有效的GPR40激动剂。 了解更多
  40. 6-OAU
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    6-OAU

    Catalog No. A15507
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    GPR84 激动剂
    6-OAU是GPR84的替代激动剂；在PI分析中，在HEK293细胞中存在Gqi5嵌合体时，可激活人GPR84，EC50为105 nM。 了解更多
  41. APD597 (JNJ-38431055)
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    APD597 (JNJ-38431055)

    Catalog No. A15452
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    GPR119 激动剂
    APD597 (JNJ-38431055)是一种GPR119激动剂，旨在治疗2型糖尿病，hGPR119的EC50为46 nM。 了解更多
  42. GSK137647A
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    GSK137647A

    Catalog No. A14542
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    FFA4/GPR120 激动剂
    GSK137647A是一种选择性FFA4激动剂，对人，小鼠和大鼠FFA4的pEC50分别为6.3、6.2和6.1。 了解更多
  43. TUG-770
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    TUG-770

    Catalog No. A12994
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    FFA1/GPR40 激动剂
    TUG-770是用于治疗2型糖尿病的高度有效的游离脂肪酸受体1（FFA1/GPR40）激动剂。 了解更多
  44. TC-G-1008
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    TC-G-1008

    Catalog No. A16364
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    GPR39 激动剂
    TC-G-1008是一种GPR39（锌受体）激动剂（大鼠和人类受体的EC50值分别为0.4和0.8 nM）。 了解更多
  45. Andarine (GTX-007)
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    Andarine (GTX-007)

    Catalog No. A10076
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    Androgen Receptor 激动剂
    Andarine (GTX-007)是研究性的选择性雄激素受体调节剂（SARM）。 了解更多
  46. Nestoron
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    Nestoron

    Catalog No. A15184
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    progesterone receptor 激动剂
    Nestoron是一种19-去孕激素衍生物和甾体孕激素，被用作激素避孕药。孕酮受体的高亲和力激动剂。 了解更多
  47. Tanaproget
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    Tanaproget

    Catalog No. A15256
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    Progesterone receptor 激动剂
    Tanaproget是一种新型的非甾体孕激素受体激动剂，与参考甾体孕激素相比，它可以更高的相对亲和力与各种物种的PR结合。 了解更多
  48. Medroxyprogesterone Acetate
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    Medroxyprogesterone Acetate

    Catalog No. A11625
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    progesterone receptor 激动剂
    Medroxyprogesterone acetate是一种孕激素，是人激素黄体酮的合成变异体，也是一种强效的黄体酮受体激动剂。 了解更多
  49. Nomegestrol acetate
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    Nomegestrol acetate

    Catalog No. A21829
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    progesterone receptor agonist
    Nomegestrol acetate is a potent, highly selective progestogen, which is characterized as a full agonist at the progesterone receptor, with no or minimal binding to other steroid receptors, including the androgen and glucocorticoid receptors. 了解更多
  50. TAK-875 (Fasiglifam)
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    TAK-875 (Fasiglifam)

    Catalog No. A11018
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    GPR 激动剂
    TAK-875 (Fasiglifam)是一种有效的，选择性的GPR40激动剂。 了解更多

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