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￥ 0.00 Neuronal Signaling
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(±)-Huperzine A
Catalog No. A21003 AChE inhibitor(??)-Huperzine A, an active Lycopodium alkaloid extracted from traditional Chinese herb, is a potent, selective and reversible acetylcholinesterase (AChE) inhibitor and has been widely used in China for the treatment of Alzheimer's disease (AD). 了解更多 -
Galanthamine hydrobromide
Catalog No. A10416 -
Rivastigmine tartrate
Catalog No. A11719 AChE 抑制剂Rivastigmine tartrate是一种双重胆碱酯酶抑制剂(ChEI)。它同时抑制丁酰胆碱酯酶(BChE)和乙酰胆碱酯酶(AChE)。 了解更多 -
Donepezil hydrochloride
Catalog No. A10330 -
Neostigmine bromide (Prostigmin)
Catalog No. A10635 -
Deoxyvasicine HCl
Catalog No. A13925 -
Acotiamide hydrochloride trihydrate
Catalog No. A15782 AChE 抑制剂Acotiamide hydrochloride trihydrate是一种在日本获准用于治疗餐后饱胀，上腹胀气和功能性消化不良引起的早饱的药物。 了解更多 -
Rivastigmine
Catalog No. A14096 -
Tacrine HCl Hydrate
Catalog No. A16970 AChE and BChE 抑制剂Tacrine hydrochloride hydrate是乙酰（AChE）和丁酰胆碱酯酶（BChE）的抑制剂，IC50分别为31 nM和25.6 nM。 了解更多 -
Fesoterodine fumarate (Toviaz)
Catalog No. A10386 -
5-hydroxymethyl tolterodine (PNU 200577)
Catalog No. A11166 muscarinic receptor 拮抗剂5-hydroxymethyl tolterodine (PNU 200577)是托特罗定的代谢产物，tolterodine是一种用于治疗尿失禁的毒蕈碱受体拮抗剂。 了解更多 -
Rocuronium bromide
Catalog No. A10803 -
Biperiden HCl
Catalog No. A10147 -
Tolterodine tartrate (Detrol LA)
Catalog No. A10937 -
Solifenacin succinate
Catalog No. A11215 muscarinic M3 receptor antagoinstSolifenacin succinate是毒蕈碱M3受体拮抗剂，用于治疗尿失禁。 了解更多 -
SVT-40776 (Tarafenacin)
Catalog No. A10808 -
Bethanechol chloride
Catalog No. A10180 Muscarinic receptor 激动剂Bethanechol chloride是拟副交感神经的胆碱氨基甲酸酯，可选择性刺激毒蕈碱受体，而不会对烟碱样受体产生任何影响。 了解更多 -
Gallamine triethiodide
Catalog No. A10417 -
Methscopolamine bromide
Catalog No. A10579 Methscopolamine bromide是一种竞争性抗毒蕈碱剂，可阻断乙酰胆碱与毒蕈碱型乙酰胆碱受体（mAChR M）的结合。 了解更多 -
Oxybutynin
Catalog No. A10684 Oxybutynin (Ditropan)是一种抗胆碱能药物，是一种竞争性的muscarinic acetylcholine receptorM1，M2，和M3拮抗剂，用于缓解尿道和膀胱疾病。 了解更多 -
Metanicotine
Catalog No. A11545 Nicotinic receptor 激动剂Metanicotine是一种神经元的尼古丁受体激动剂，对α4β2亚型具有高选择性（Ki = 26 nM）。选择性是α7受体（Ki = 36000 nM）的1,000倍以上。 了解更多 -
Catharanthine sulfate
Catalog No. A12161 Catharanthine sulfate是长春碱型生物碱前体，具有抗肿瘤活性。它通过离子通道阻断和脱敏来抑制AChR。 了解更多 -
Diphenidol HCl
Catalog No. A14244 -
Xanomeline oxalate
Catalog No. A13685 mAChR 激动剂Xanomeline oxalate是毒蕈碱型乙酰胆碱受体的有效激动剂（M1，M2，M3，M4和M5的EC50值分别为0.3、92.5、5、52和42 nM）。 了解更多 -
PF-3635659
Catalog No. A13548 -
Cevimeline hydrochloride hemihydrate
Catalog No. A15042 -
Umeclidinium bromide
Catalog No. A15268 Muscarinic receptor 拮抗剂Umeclidinium bromide (GSK573719A)是毒蕈碱受体拮抗剂，可用于治疗慢性阻塞性肺疾病（COPD）。 了解更多 -
Imidafenacin
Catalog No. A15490 M3 receptors 抑制剂Imidafenacin是一种有效的选择性M3受体抑制剂，Kb为0.317 nM。对M2受体的效力较低（IC50 = 4.13 nM）。 了解更多 -
TBPB
Catalog No. A14205 -
Revefenacin
Catalog No. A15986 -
Glycopyrrolate
Catalog No. A12641 -
Flavoxate
Catalog No. A12900 -
Acetylcholine iodide
Catalog No. A16390 Acetylcholine iodide是一种神经递质，存在于神经肌肉接头，植物神经节，副交感神经效应接头，交感神经效应接头的子集以及中枢神经系统的许多部位。 了解更多 -
Atropine methyl bromide
Catalog No. A18026 mAChR antagonistAtropine methyl bromide, a muscarinic receptor (mAChR) antagonist, is a quaternary ammonium salt of atropine and a mydriatic for dilation of the pupil during ophthalmic examination. It is introduced for relieving pyloric spasm in infants for its highly polar nature. It penetrates less readily into the central nervous system than atropine. 了解更多 -
Cevimeline hydrochloride
Catalog No. A18092 mAChR agonistCevimeline (Evoxac) Hcl is a parasympathomimetic and muscarinic agonist, with particular effect on M3 receptors; used in the treatment of dry mouth associated with sjogren's syndrome. 了解更多
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