Opioid Receptors

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  1. Trimebutine maleate

    Catalog No. A18115
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    ?- opioid receptor agonist
    Trimebutine Maleate is a drug with antimuscarinic and weak mu opioid agonist effects. Trimebutine Maleate modulates the calcium and potassium channels, relieves abdominal pain in patients with irritable bowel syndrome. 了解更多
  2. Cebranopadol (GRT-6005)

    Catalog No. A12670
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    Opioid Receptor 激动剂
    Cebranopadol是一种有效的伤害感受器/孤儿蛋白FQ肽(NOP)和阿片受体激动剂。作用于人NOP,MOP,KOP 和δ-阿片肽(DOP)受体,Ki/EC50 分别为 0.9 nM/13 nM,0.7 nM/1.2 nM,2.6 nM/17 nM,18 nM/110 nM。 了解更多
  3. Alvimopan monohydrate

    Catalog No. A14992
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    ?-opioid receptor 激动剂
    Alvimopan monohydrate是一种外围作用的类阿片受体(PAM-OR,IC50 = 1.7 nM)拮抗剂,可促进术后肠胃的恢复。 了解更多
  4. Alvimopan dihydrate

    Catalog No. A14991
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    ?-opioid receptor 激动剂
    Alvimopan dihydrate (LY 246736,ADL 8-2698)是一种外周作用的类阿片受体(PAM-OR,IC50 = 1.7 nM)拮抗剂,可促进术后胃肠道恢复。 了解更多
  5. ADL5747

    Catalog No. A13479
    δ opioid receptor 激动剂
    ADL5747是一种选择性的非肽类δ opioid激动剂。 了解更多
  6. ADL5859 HCl

    Catalog No. A11072
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    Opioid Receptor 激动剂
    ADL5859 HCl是高效的选择性δ阿片受体激动剂,Ki值为0.84 nM,ED50值为20 nM。 了解更多
  7. MCOPPB 3HCl

    Catalog No. A10561
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    NOP receptor 激动剂
    MCOPPB 3HCl是一种用作伤害感受器受体的有效和选择性激动剂的化合物,pKi为10.07。 了解更多
  8. BRL 52537 HCl

    Catalog No. A11210
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    Opioid Receptors 激动剂
    BRL 52537 hydrochloride是一种高度选择性和有效的κ阿片类激动剂(Ki = 0.24 nM)。比吗啡强25倍。 了解更多
  9. Nalfurafine hydrochloride

    Catalog No. A12579
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    opioid κ-selective 激动剂
    Nalfurafine hydrochloride是一种κ-opioid激动剂。 了解更多
  10. Nalmefene hydrochloride

    Catalog No. A13843
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    dopamine receptor 激动剂
    Nalmefene hydrochloride是opioid receptor拮抗剂。 了解更多
  11. U-69593

    Catalog No. A14187
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    κ1-opioid receptor 激动剂
    U-69593是有效的选择性κ1阿片受体激动剂(EC50 = 80-109 nM)。在体内有活性。抗伤害感受。 了解更多
  12. TRV130 HCl (Oliceridine)

    Catalog No. A15444
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    u-opioid receptor 激动剂
    TRV130 HCl (Oliceridine)是一种新型的μ-opioid 受体(MOR)G蛋白偏向配体。诱导强大的G蛋白信号传导(pEC50 = 8.1),效力和功效与吗啡相似,但β-arrestin募集和受体内在化作用要低得多。 了解更多
  13. DPI-3290

    Catalog No. A13699
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    opioid receptors agonist
    DPI-3290 (Org 41793) is a potent and specific opioid receptors agonist with Ki values of 0.18 nM, 0.46 nM, and 0.62 nM for δ-, μ-, and κ-opioid receptors, respectively. 了解更多
  14. CYT-1010 hydrochloride

    Catalog No. A21348
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    mu-opioid receptor agonist
    CYT-1010 hydrochloride is a mu-opioid receptor agonist extracted from patent WO2013173730A2, with EC50s of 13.1 nM and 0.0053 nM on beta-arrestin recruitment and inhibition of cAMP production, respectively. 了解更多
  15. AR-M 1000390 hydrochloride

    Catalog No. A21911
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    δ opioid receptor agonist
    AR-M 1000390 hydrochloride is an exceptionally selective, potent δ opioid receptor agonist with an EC50 of 7.2??0.9 nM for δ agonist potency. 了解更多

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