Tipifarnib (Zarnestra)

目录号: A10935

FTase 抑制剂

Tipifarnib (Zarnestra)

Tipifarnib (Zarnestra) Chemical Structure

CAS NO. 192185-72-1

Tipifarnib (Zarnestra)是一种法尼基转移酶抑制剂,可在激酶途径变得过度活跃之前的翻译后修饰步骤中抑制Ras激酶。

库存: 现货

规格 价格 数量
5 mg
¥ 567.00
10 mg
¥ 1,008.00
25 mg
¥ 3,150.00
100 mg
¥ 5,600.00
10mM * 1mL in DMSO
¥ 1,442.00
Warning 产品仅用于科学研究,不针对患者销售,望谅解.

产品详情

Tipifarnib (Zarnestra)是一种法尼基转移酶抑制剂,可在激酶途径变得过度活跃之前的翻译后修饰步骤中抑制Ras激酶。
靶点信息
FTase
0.6 nM
In vitro (25°C) DMSO 14 mg/mL (28.6 mM)
Water Insoluble
Ethanol Insoluble
In vivo 15% Captisol+citrate vehicle 4 mg/mL
* <1 mg/ml means slightly soluble or insoluble.
* Please note that Adooq tests the solubility of all compounds in-house, and the actual solubility may differ slightly from published values. This is normal and is due to slight batch-to-batch variations.
Concentration / Solvent Volume / Mass 1 mg 5 mg 10 mg
0.1 mM 20.43 mL 102.17 mL 204.33 mL
0.5 mM 4.09 mL 20.43 mL 40.87 mL
1 mM 2.04 mL 10.22 mL 20.43 mL
5 mM 0.41 mL 2.04 mL 4.09 mL

*The above data is based on the productmolecular weight 489.4 . Batch specific molecular weights may vary from batch to batch due to solvent of hydration, which will affect the solvent volumes required to prepare stock solutions.

目录号 A10935
作用机制 Inhibitor (抑制剂)
M. Wt 489.4
Formula C27H22Cl2N4O
Purity >99%
Storage

Store lyophilized at -20ºC, keep desiccated.
In lyophilized form, the chemical is stable for 36 months.
In solution, store at -20ºC and use within 3 months to prevent loss of potency. Aliquot to avoid multiple freeze/thaw cycles.

CAS No. 192185-72-1
Synonyms IND 58359, R115777
SMILES CN1C=NC=C1[C@@](C2=CC=C(C=C2)Cl)(C3=CC4=C(C=C3)N(C(=O)C=C4C5=CC(=CC=C5)Cl)C)N

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