主页 /
搜索结果：“jwh 250”

“jwh 250”的搜索结果

Quick View
Cilnidipine

Catalog No. A10215
Quick View

添加到收藏
Calcium channel blocker

Cilnidipine是提供血管平滑肌中L型电压门控钙通道和交感神经末梢N型钙通道的双重阻滞剂。了解更多

Bulk Inquiry Free Sample
Quick View
Glyburide

Catalog No. A10433
Quick View

添加到收藏
K+ channel and CFTR Cl- channel blocker

Glyburide (Glibenclamide) 是一种抗糖尿病化合物，是一类磺脲类药物。了解更多

Bulk Inquiry Free Sample
Quick View
Pindolol

Catalog No. A13422
Quick View

添加到收藏
Beta adrenergic receptor blocker

Pindolol是一种非选择性β阻断剂，具有部分β肾上腺素能受体激动剂活性。了解更多

Bulk Inquiry
Quick View
QX 314 chloride

Catalog No. A13760
Quick View

添加到收藏
Sodium channel Blocker

QX 314 chloride是利多卡因的膜不可渗透的季衍生物，一种电压激活的Na+通道阻滞剂。了解更多

Bulk Inquiry Free Sample
Quick View
Phentolamine HCl

Catalog No. A13421
Quick View

添加到收藏
α-Adrenergic blocker

Phentolamine HCl是一种AR(α肾上腺素能)阻滞剂。了解更多

Bulk Inquiry
Quick View
Cinnarizine

Catalog No. A16455
Quick View

添加到收藏
calcium channel blocker

Cinnarizine是哌嗪的药物衍生物，其特征在于抗组胺药和钙通道阻滞剂。了解更多

Bulk Inquiry
Quick View
A 803467

Catalog No. A11234
Quick View

添加到收藏
Sodium channel Blocker

A 803467是NaV1.8通道的选择性阻滞剂（hNaV1.8，hNaV1.3，hNaV1.7，hNaV1.5和hNaV1.2通道的IC50值分别为8、2450、6740、7340和7380 nM）。了解更多

Bulk Inquiry Free Sample
Quick View
TRAM-34

Catalog No. A12783
Quick View

添加到收藏
Potassium Channel Blocker

TRAM-34是中等电导Ca2+激活的K+通道（KCa3.1）（Kd = 20 nM）的高度选择性阻滞剂。在KV，BKCa，KCa2，Na+，CRAC和Cl-通道上具有200-1500倍的选择性。抑制有丝分裂刺激对淋巴细胞的激活。了解更多

Product Citations (2)

Bulk Inquiry Free Sample
- Samuel Drinkall, .et al. The two pore potassium channel THIK-1 regulates NLRP3 inflammasome activation, Glia, 2022, Jul;70(7):1301-1316 PMID: 35353387
- Cheong Hoon Seo, .et al. Altered K Ca 3.1 expression following burn injury and the therapeutic potential of TRAM-34 in post-burn hypertrophic scar formation, Transl Res, 2021, Apr 24 PMID: 33905948
Quick View
Procainamide HCl

Catalog No. A14240
Quick View

添加到收藏
Sodium channel blocker/DNMT 抑制剂

Procainamide HCl是钠通道阻滞剂，又是DNA甲基转移酶抑制剂。了解更多

Bulk Inquiry
Quick View
Encainide HCl

Catalog No. A13898
Quick View

添加到收藏
Sodium channel blocker

Encainide hydrochloride是一种钠通道阻滞剂，具有Ic类抗心律不齐的作用。Encainide是一种非手性抗心律失常药和苯甲酰苯胺衍生物。了解更多

Bulk Inquiry
Quick View
GSK-2193874

Catalog No. A14201
Quick View

添加到收藏
TRPV4 blocker

GSK2193874被确定为选择性的口服活性TRPV4阻滞剂，可通过重组TRPV4通道和天然内皮TRPV4电流抑制Ca(2+)流入。了解更多

Bulk Inquiry
Quick View
Gap 26

Catalog No. A14865
Quick View

添加到收藏
Gap junction blocker

Gap 26是连接蛋白模拟肽，对应于连接蛋白43的残基63-75，其是间隙连接阻断剂。了解更多

Bulk Inquiry
Quick View
Cannabichromene

Catalog No. A15497
Quick View

添加到收藏
TRPA1 activatior/TRPM8 blocker

Cannabichromene是一种主要的非精神植物大麻素，可抑制内源性大麻素失活并激活瞬时受体电位锚蛋白1（TRPA1）。内源性大麻素和TRPA1均可调节肠胃蠕动。了解更多

Bulk Inquiry