微信关注
China
Total item
Cart Subtotal
￥ 0.00 “receptor”的搜索结果
-
(S)-Willardiine
Catalog No. A21957 AMPA/kainate receptors agonist(S)-Willardiine is a potent agonist of AMPA/kainate receptors with EC50 of 44.8 uM. 了解更多 -
Gaboxadol hydrochloride
Catalog No. A21730 GABAA receptors agonistGaboxadol hydrochloride (Lu 02-030 hydrochloride) is a selective agonist at GABAA receptors that contain α4-δ subunits, and has anxiolytic and sedative effects. 了解更多 -
O-Phospho-L-serine
Catalog No. A21159 group III mGluR receptors agonistO-Phospho-L-serine is the immediate precursor to L-serine in the serine synthesis pathway, and an agonist at the group III mGluR receptors (mGluR4, mGluR6, mGluR7, and mGluR8); O-Phospho-L-serine also acts as a weak antagonist for mGluR1 and a potent antagonist for mGluR2. 了解更多 -
Carbetocin
Catalog No. A18080 peripheral oxytocin receptors agonistCarbetocin (Lonactene; Duratocin) is an obstetric drug used to control postpartum hemorrhage and bleeding after giving birth; an agonist at peripheral oxytocin receptors. 了解更多 -
L-Glutamic acid monosodium salt
Catalog No. A16591 excitatory transmitter/agonistL-Glutamic acid monosodium salt acts as an excitatory transmitter and an agonist at all subtypes of glutamate receptors (metabotropic, kainate, NMDA, and AMPA). (S)-Glutamic acid shows a direct activating effect on the release of DA from dopaminergic terminals. 了解更多 -
(S)-Glutamic acid
Catalog No. A15458 glutamate receptors agonist(S)-Glutamic acid acts as an excitatory transmitter and an agonist at all subtypes of glutamate receptors (metabotropic, kainate, NMDA, and AMPA). 了解更多 -
Donitriptan
Catalog No. A13145 5-HT1B/1D receptors agonistDonitriptan is a potent, high efficacy agonist at 5-HT1B/1D receptors with pKis of 9.4 and 9.3, respectively. 了解更多 -
Almitrine mesylate
Catalog No. A18020 Peripheral chemoreceptor agonistAlmitrine mesylate, a peripheral chemoreceptor agonist, inhibits selectively the Ca2+-dependent K+ channel. 了解更多 -
Cevimeline (AF-102B)
Catalog No. A11372 Muscarinic agonistCevimeline (AF-102B) is a parasympathomimetic and muscarinic agonist, with particular effect on M3 receptors; used in the treatment of dry mouth associated with sjogren's syndrome. 了解更多 -
Baclofen
Catalog No. A18248 GABA agonistBaclofen is a GABA agonist specific for GABA-B receptors. Baclofen is a synthetic chlorophenyl-butanoic acid derivative used to treat spasms due to spinal cord damage and multiple sclerosis, muscle-relaxing It acts at spinal and supraspinal sites, reducing excitatory transmission. 了解更多 -
Cevimeline hydrochloride
Catalog No. A18092 mAChR agonistCevimeline (Evoxac) Hcl is a parasympathomimetic and muscarinic agonist, with particular effect on M3 receptors; used in the treatment of dry mouth associated with sjogren's syndrome. 了解更多 -
Dihydroergotamine Mesylate
Catalog No. A17764 Serotonin receptors agonistDihydroergotamine Mesylate, also known as DHE or Migranal, is an ergot alkaloid used to treat migraines. It has similar actions to the triptans, acting as an agonist to the serotonin receptors and causing vasoconstriction of the intracranial blood vessels, but also interacts centrally with dopamine and adrenergic receptors. 了解更多 -
Vilanterol
Catalog No. A13125 ultra-long-acting β? adrenoreceptor 激动剂Vilanterol是一种新的选择性β2-AR激动剂，PEC50值为10.37±0.05。 了解更多 -
BRL 37344 Na Salt
Catalog No. A13676 -
BRL 52537 HCl
Catalog No. A11210 Opioid Receptors 激动剂BRL 52537 hydrochloride是一种高度选择性和有效的κ阿片类激动剂（Ki = 0.24 nM）。比吗啡强25倍。 了解更多 -
GW3965 HCl
Catalog No. A11204 -
Glucocorticoid receptor agonist
Catalog No. A11431 Glucocorticoid receptor agonistGlucocorticoid receptor agonist is a potent Glucocorticoid receptor agonist. 了解更多 -
H4 Receptor antagonist 1
Catalog No. A18929 histamine H4 receptor inverse agonistH4 Receptor antagonist 1 is a potent and selective histamine H4 receptor inverse agonist, with an IC50 of 19 nM. 了解更多 -
Orexin 2 Receptor Agonist
Catalog No. A15982 -
TGR5-Receptor-Agonist
Catalog No. A13732 TGR5(GPCR19) 激动剂TGR5 Receptor Agonist是一种有效的TGR5（GPCR19）激动剂，在U2-OS细胞分析（pEC50 = 6.8）和黑素细胞（pEC50 = 7.5）中显示出增强的效力。 了解更多 -
Pardoprunox hydrochloride
Catalog No. A21624 partial dopamine D2 and D3 receptor agonistPardoprunox hydrochloride is a novel partial dopamine D2 and D3 receptor agonist and serotonin 5-HT1A receptor agonist, D2 (pKi = 8.1) and D3 receptor (pKi = 8.6) partial agonist and 5-HT1A receptor (pKi = 8.5) full agonist. 了解更多 -
Cutamesine
Catalog No. A21152 sigma 1 receptor agonistCutamesine (SA4503; AGY-94806) is a selective sigma 1 receptor(??1R) agonist; high affinity for the sigma 1 receptor subtype labeled by (+)-[3H]pentazocine (IC50= 17.4??1.9 nM); 100-fold less affinity for the sigma 2 receptor. 了解更多 -
Cariprazine
Catalog No. A21202 D3 receptor and D2 receptor partial agonistCariprazine is a novel antipsychotic drug candidate that exhibits high affinity for the D3 (Ki=0.085 nM) and D2 (Ki=0.49 nM) receptors, and moderate affinity for the 5-HT1A receptor (Ki=2.6 nM). 了解更多 -
Dihydrexidine
Catalog No. A21949 D1-like dopamine receptor (D1/D5) agonistDihydrexidine (DAR-0100) is a high potent, selective and full efficacy D1-like dopamine receptor (D1/D5) agonist with an IC50 of 10 nM for D1 receptor. Dihydrexidine exhibits potent antiparkinsonian activity. 了解更多 -
Ditolylguanidine
Catalog No. A21268 Sigma receptor agonistDitolylguanidine (1,3-Di-o-tolylguanidine) is an agonist of sigma receptor (??1/??2 receptor). 了解更多 -
Lobeline hydrochloride
Catalog No. A17333 nicotinic receptor agonistLobeline hydrochloride, a nicotinic receptor agonist, acting as a potent antagonist at both α3β2 and α4β2 neuronal nicotinic receptor subtypes. 了解更多 -
N6-Cyclohexyladenosine
Catalog No. A21008 A1 receptor agonistN6-Cyclohexyladenosine is a selective A1 receptor agonist (EC50 = 8.2 nM). 了解更多 -
Aripiprazole (D8)
Catalog No. A22004 human 5-HT1A receptor partial agonistAripiprazole D8 (OPC-14597 D8) is the deuterium labeled Aripiprazole, which is a human 5-HT1A receptor partial agonist with a Ki of 4.2 nM. 了解更多 -
Ro 10-5824 dihydrochloride
Catalog No. A21986 dopamine D4 receptor partial agonistRo 10-5824 dihydrochloride is a selective dopamine D4 receptor partial agonist, with Ki of 5.2 nM. 了解更多 -
Mapracorat
Catalog No. A21953 glucocorticoid receptor agonistMapracorat is a novel non-steroidal selective glucocorticoid receptor agonist. 了解更多 -
MT-7716 free base
Catalog No. A21928 non-peptide nociceptin receptor (NOP) agonistMT-7716 free base (W-212393) is a selective non-peptide nociceptin receptor (NOP) agonist and promising potential treatment drug for alcohol abuse and relapse prevention. 了解更多 -
AR-M 1000390 hydrochloride
Catalog No. A21911 δ opioid receptor agonistAR-M 1000390 hydrochloride is an exceptionally selective, potent δ opioid receptor agonist with an EC50 of 7.2??0.9 nM for δ agonist potency. 了解更多 -
Vilazodone D8
Catalog No. A21876 SSR inhibitor / 5-HT1A receptor partial agonistVilazodone D8 is the a deuterium labeled vilazodone, which is a combined serotonin specific reuptake inhibitor (SSRI) and 5-HT1A receptor partial agonist. 了解更多 -
SKF 82958
Catalog No. A21866 -
Nomegestrol acetate
Catalog No. A21829 progesterone receptor agonistNomegestrol acetate is a potent, highly selective progestogen, which is characterized as a full agonist at the progesterone receptor, with no or minimal binding to other steroid receptors, including the androgen and glucocorticoid receptors. 了解更多 -
PF-5190457
Catalog No. A21784 ghrelin receptor inverse agonistPF-5190457 is a potent and selective ghrelin receptor inverse agonist with a pKi of 8.36. 了解更多 -
SKF-82958 hydrobromide
Catalog No. A21763 D1/D5 receptor full agonistSKF-82958 hydrobromide is a D1/D5 receptor full agonist. 了解更多
联系我们
United StatesAdooq Bioscience
Toll Free: (866) 930-6790
Fax: +1-323-606-8156
Email: sales@adooq.com
Not your Region? View all Distributors
FILTER BY:
Filtering:
- 作用机制: Agonist (激动剂) 删除该内容
购物选项
- 分类
-
- Apoptosis (1)
- Cell Metabolism (19)
- Autophagy Signaling (4)
- Immunology & Inflammation (6)
- GPCR / G Protein (158)
- Neuronal Signaling (25)
- Proteases (2)
- Membrane Transporters/Ion Channels (3)
- Endocrinology / Hormones (26)
- PROTACs (1)
- Others (3)
- Natural Products (1)
- Ready to Use Solution (22)
- Products On Sale (35)
- 靶点
ADOOQ 产品质量保证
We promise all products to perform as described.