“bone morphogenetic proteins bmp”的搜索结果
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BMP 抑制剂
Dorsomorphin 2HCl (BML-275)是BMP信号传导的选择性小分子抑制剂,可促进胚胎干细胞的心肌发生。Dorsomorphin通过抑制骨形态发生蛋白信号转导逆转乳腺癌起始细胞的间质表型。
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- Kameshima S, .et al. Eukaryotic elongation factor 2 (eEF2) kinase/eEF2 plays protective roles against glucose deprivation-induced cell death in H9c2 cardiomyoblasts, Apoptosis, 2019, Feb 8 PMID: 30737648
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BMP 抑制剂
K02288是一种有效的选择性I型BMP受体抑制剂,对ALK2,ALK1和ALK6的IC50为1.1、1.8、6.4 nM。
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BMP receptor 抑制剂
ML347是一种选择性BMP受体抑制剂。
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BMP receptor 抑制剂
LDN-212854是一种ALK2偏爱的BMP I型受体激酶抑制剂。
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ALK2 抑制剂
DMH-1是骨形态发生蛋白(BMP)ALK2受体的选择性抑制剂(IC50 = 108 nM)。
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- Teresa Rayon, .et al. Species-specific pace of development is associated with differences in protein stability, Science, 2020, Sep 18;369(6510):eaba7667 PMID: 32943498
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osteoclastic bone resorption 抑制剂
Zoledronic acid, 破骨细胞抑制剂,通过抑制甲羟戊酸途径诱导破骨细胞凋亡。
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LDN193189 HCl是ldn193189的盐酸盐。LDN193189是一种高效的小分子BMP抑制剂,可抑制BMP I型受体ALK2(IC50:5 nM),ALK3(IC50:30 nM)和ALK6(TGFβ1/ BMP信号转导)以及随后的SMAD磷酸化。
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- Brandon J.Peiffer, .et al. Activation of BMP Signaling by FKBP12 Ligands Synergizes with Inhibition of CXCR4 to Accelerate Wound Healing, Cell Chem Biol, 2019, 26, 1-10
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Neuroprotectant
Dimebon dihydrochloride是一种非选择性的抗组胺药,具有增强认知能力。
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ALK 抑制剂
LDN193189是一种高效的小分子BMP抑制剂,可抑制BMP I型受体ALK2(IC50=5 nM),ALK3(IC50=30 nM)和ALK6(TGFβ1/BMP信号转导)以及随后的SMAD磷酸化。
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- Trang Thi Huyen Dang, .et al. BMP10 positively regulates myogenic differentiation in C2C12 myoblasts via the Smad 1/5/8 signaling pathway, Mol Cell Biochem, 2021, May;476(5):2085-2097 PMID: 33517521
- Shizu Aikawa, .et al. Autotaxin-lysophosphatidic acid-LPA 3 signaling at the embryo?\epithelial boundary controls decidualization pathways, EMBO J, 2017, Jul 14; 36(14): 2146-2160 PMID: 28588064
- HIROTAKA SOMEYA, .et al. Thymosin beta 4 is associated with RUNX2 expression through the Smad and Akt signaling pathways in mouse dental epithelial cells, Int J Mol Med, 2015, May; 35(5): 1169-1178 PMID: 25739055
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TGF-beta/Smad 抑制剂
GW788388是有效的,口服活性的,选择性的转化生长因子β受体I(TGF-βR1)(激活素受体样激酶5,ALK5)抑制剂,无细胞试验中IC50为18 nM,也抑制TGF-βII型受体和activin II型受体活性,但不抑制BMP II型受体。
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