“leukotriene receptor”的搜索结果
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LTD4 receptor 拮抗剂
MK-0679 (Verlukast)是有效的白三烯D4拮抗剂。
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CysLT1 receptor 拮抗剂
MK-571是有效的CysLT1(LTD4)白三烯受体反向激动剂,EC50值为1.3 nM。
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- Jung-Hung Chen, .et al. Transplacental transfer of acetaminophen in pregnant rats, Biomed Pharmacother, 2022, Oct;154:113613 PMID: 36058146
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CysLT1 receptor 拮抗剂
MK-571 sodium salt是一种选择性的口服活性CysLT1受体拮抗剂。它阻断LTD4而不是LTC4与人和豚鼠肺膜的结合,Ki值分别为0.22 nM和2.1 nM。
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BLT2 receptors 拮抗剂
LY 255283是一种有效的 BLT2 receptors 拮抗剂。
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LTR antagonist
AS-35 is an orally effective, potent and selective antagonist of leukotrienes, antagonizes LTC4-, LTD4 and LTE4-induced contractions of the ileum with IC50 values of 8 nM, 4 nM and 3 nM, respectively, and has antiallergic activities.
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LTR antagonist
Montelukast (trade name Singulair) is a leukotriene receptor antagonist (LTRA) used for the maintenance treatment of asthma and to relieve symptoms of seasonal allergies.
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