“TRV130 HCl”的搜索结果

20 个项目

每页

设置降序顺序
  1. Fexofenadine HCl

    Catalog No. A11859
    Quick View
    COX 抑制剂/histamine H1 receptor 激动剂
    Fexofenadine Hydrochloride是一种抗组胺药,可抑制Cox-1,Cox-2,并且是组胺H1受体激动剂,IC50为246 nM。 了解更多
  2. A-438079 HCl

    Catalog No. A12597
    Quick View
    P2X7 receptor 拮抗剂
    A-438079 HCl是一种竞争性P2X7受体拮抗剂(抑制人重组P2X7细胞系中Ca2+流入的pIC50 = 6.9)。在其他P2受体上没有活性(IC50 > 10 uM)。 了解更多
  3. GW791343 HCl

    Catalog No. A11107
    Quick View
    P2X7 modulator
    GW791343 HCl充当人P2X7的负变构调节剂(pIC50 = 6.9-7.2)和大鼠P2X7的正变构调节剂。 了解更多
  4. ABT-418 HCl

    Catalog No. A13688
    Quick View
    nAChR 激动剂
    ABT-418 HCl是神经元烟碱型乙酰胆碱受体激动剂。 了解更多
  5. Tropisetron HCL

    Catalog No. A14375
    Quick View
    5-HT3 receptor 拮抗剂
    Tropisetron HCL是选择性的5-HT3受体拮抗剂和α7烟碱样受体激动剂,对5-HT3受体的IC50为70.1±0.9 nM。 了解更多
  6. Deoxyvasicine HCl

    Catalog No. A13925
    Quick View
    AChE 抑制剂
    Desoxypeganine hydrochloride是一种AChE(乙酰胆碱酯酶)抑制剂,已用于治疗阿尔茨海默氏痴呆症。 了解更多
  7. Diphenidol HCl

    Catalog No. A14244
    Quick View
    M2/M3 拮抗剂
    Diphenidol HCl是毒蕈碱M2和M3受体的有效拮抗剂,pKb为6.72和7.02。 了解更多
  8. Adiphenine HCl

    Catalog No. A11716
    Quick View
    AChR抑制剂
    Adiphenine Hydrochloride是烟碱受体抑制剂,IC50为15μM,用作解痉药物。 了解更多
  9. Tacrine HCl Hydrate

    Catalog No. A16970
    Quick View
    AChE and BChE 抑制剂
    Tacrine hydrochloride hydrate是乙酰(AChE)和丁酰胆碱酯酶(BChE)的抑制剂,IC50分别为31 nM和25.6 nM。 了解更多
  10. GW791343 trihydrochloride

    Catalog No. A21204
    Quick View
    P2X7 allosteric modulator
    GW791343 3Hcl is a P2X7 allosteric modulator; exhibits species-specific activity and acts as a negative allosteric modulator of human P2X7 (pIC50 = 6.9 - 7.2). 了解更多
  11. 5-Iodo-A-85380 2HCl

    Catalog No. A13639
    Quick View
    nAChR 激动剂
    5-Iodo-A-85380 2HCl是针对a4b2和a6b2烟碱乙酰胆碱受体的强效亚型选择性激动剂。 了解更多
  12. Dimebon 2HCl

    Catalog No. A10312
    Quick View
    Neuroprotectant
    Dimebon dihydrochloride是一种非选择性的抗组胺药,具有增强认知能力。 了解更多
  13. Cevimeline hydrochloride

    Catalog No. A18092
    Quick View
    mAChR agonist
    Cevimeline (Evoxac) Hcl is a parasympathomimetic and muscarinic agonist, with particular effect on M3 receptors; used in the treatment of dry mouth associated with sjogren's syndrome. 了解更多
  14. Tacrine HCl

    Catalog No. A17374
    Quick View
    AChE & butyrylcholinesterase inhibitor
    Tacrine is a derivative of aminoacridine that functions as an inhibitor of both acetylcholinesterase (AChE) and butyrylcholinesterase (IC50s = 31 and 26.5 nM, respectively). 了解更多
  15. Mecamylamine Hydrochloride

    Catalog No. A17884
    Quick View
    nAChR antagonist
    Mecamylamine hydrochloride is a nAChR antagonist previously used to treat hypertension. It displays a wide variety of activities, including reducing depression-like behaviors in subjects with Tourette's syndrome and improving rates of smoking cessation. 了解更多
  16. Pitofenone Hydrochloride

    Catalog No. A17053
    Quick View
    Antispasmodic Agent
    Pitofenone Hydrochloride是抗痉化合物。它是乙酰胆碱酯酶活性的有效抑制剂。 了解更多
  17. Phenoxybenzamine hydrochloride

    Catalog No. A10719
    Quick View
    α-adrenergic (AR) 拮抗剂/CaM 抑制剂
    Phenoxybenzamine hydrochloride是一种细胞可渗透的,非特异性的,不可逆的α-肾上腺素(AR)拮抗剂,也可作为CaM抑制剂。 了解更多
  18. Ticlopidine HCl

    Catalog No. A11690
    Quick View
    Ticlopidine是一种二磷酸腺苷(ADP)受体抑制剂。它通过阻断ADP受体来改变血小板膜的功能,从而抑制血小板聚集。这防止了糖蛋白IIb/IIIa的构象变化,从而使血小板与血纤蛋白原结合。 了解更多
  19. Biperiden HCl

    Catalog No. A10147
    Quick View
    Muscarinic receptor antagonist
    Biperiden HCl是毒蕈碱受体拮抗剂,对M1亚型表现出一定的选择性。 了解更多
  20. SKF 89976A HCl

    Catalog No. A10849
    Quick View
    GABA uptake 抑制剂
    SKF 89976A HCl是一种有效的GABA吸收抑制剂,hGAT-1,rGAT-2,hGAT-3和hBGT-1的IC50分别为0.13、550、944和7210μM。 了解更多

20 个项目

每页

设置降序顺序
Rewards