“azd”的搜索结果

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  1. Glycine

    Catalog No. A17936
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    NMDA antagonist
    AZD-4282, also known as aminoacetic acid and glycine, is a N-methyl-D-aspartate (NMDA) receptor antagonist potentially for the treatment of neuropathic pain. 了解更多
  2. Ispronicline (TC-1734, AZD-3480)

    Catalog No. A14183
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    nAChR 激动剂
    Ispronicline (TC-1734,AZD-3480)是神经元烟碱乙酰胆碱受体部分激动剂。Ispronicline是亚型选择性的,主要与a4b2亚型结合。它具有抗抑郁、益智和神经保护作用。 了解更多
  3. AZD3839 free base

    Catalog No. A21606
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    BACE1 inhibitor
    AZD3839 (free base) is a potent and selective BACE1 inhibitor with IC50 of 23.6 uM, about 14-fold selectivity over BACE2, also a β-secretase enzyme inhibitor. 了解更多
  4. Lanabecestat

    Catalog No. A12282
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    BACE1 inhibitor
    Lanabecestat (AZD3293) is a potent, highly permeable, orally active and blood-brain barrier penetrating BACE1 inhibitor with a Ki of 0.4 nM. 了解更多
  5. AZD1283

    Catalog No. A15443
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    P2Y12 receptor 拮抗剂
    AZD1283是P2Y12受体的有效拮抗剂,EC50为3.0 ug/kg/min,TI> 10;结合IC50为11 nM。 了解更多
  6. AZD5423

    Catalog No. A13249
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    nonsteroidal glucocorticoid receptor 激动剂
    AZD5423是新型的非甾体类糖皮质激素受体激动剂。 了解更多
  7. AZD3839

    Catalog No. A12825
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    BACE1 抑制剂
    AZD3839是人类BACE1的有效选择性抑制剂,Ki为26.1 nM。 了解更多
  8. Ticagrelor (AZD6140)

    Catalog No. A11238
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    P2Y12 拮抗剂
    Ticagrelor (AZD6140)是第一个可逆结合的口服P2Y(12)受体拮抗剂,可阻断ADP诱导的血小板聚集。 了解更多

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